Target Details
| UniProt AC | P29317 |
|---|---|
| Gene Symbol | EPHA2 |
| Protein Name | Ephrin type-A receptor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF14575 (EphA2_TM) PF25599 (Ephrin_CRD) PF01404 (Ephrin_lbd) PF00041 (fn3) PF07714 (PK_Tyr_Ser-Thr) PF00536 (SAM_1) |
Summary
- Multi-target molecules 540
- Clinical molecules 37
- Avg pChEMBL 6.74
KEGG Pathways (5)
Associated Diseases (1)
Active Molecules (540)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LCVIRAZGMYMNNT
|
6.7 | Kd | 20 | — | |
SFPWNTQWFFNJIH
|
6.7 | Ki | 48 | — | |
HHZIURLSWUIHRB
|
6.6 | Kd | 57 | Yes | |
BOBGABAXWFYHQX
|
6.6 | Ki | 9 | — | |
GWMATETWMAQOFL
|
6.6 | Ki | 36 | — | |
HKSZLNNOFSGOKW
|
6.6 | Ki | 118 | — | |
OOQJIJYKWXLQNC
|
6.6 | IC50 | 16 | Yes | |
YMIJUBCSOKSFRU
|
6.6 | Ki | 87 | — | |
ZCCJKVBTHCOISJ
|
6.6 | Ki | 46 | — | |
IUGBGEUCXVKGQK
|
6.6 | Kd | 13 | — | |
LCVIRAZGMYMNNT
|
6.6 | Kd | 4 | — | |
WMXDIPVFXWNELM
|
6.6 | IC50 | 14 | Yes | |
JRKYKAKARRYSSS
|
6.5 | IC50 | 14 | Yes | |
AWSQADBSXFTFKL
|
6.5 | Kd | 5 | — | |
DKSNLQYRZJKYOC
|
6.5 | Ki | 51 | — | |
HRZOUBQYVUXBNS
|
6.5 | Ki | 38 | — | |
KNACLJBHKVSTDL
|
6.5 | Ki | 40 | — | |
LYNBNVBMAGDJRW
|
6.5 | Ki | 81 | — | |
SEVCBWKJSOLMNQ
|
6.5 | Ki | 38 | — | |
APPXQUDJLJXULP
|
6.5 | IC50 | 47 | — | |
HHFBDROWDBDFBR
|
6.4 | Kd | 40 | Yes | |
XKZQZMSAWVDRSP
|
6.4 | IC50 | 39 | Yes | |
FAYAUAZLLLJJGH
|
6.4 | Ki | 36 | Yes | |
JXNMCDLXYWQTIW
|
6.4 | Ki | 13 | — | |
PUPCRRRSBUYJAD
|
6.4 | Ki | 44 | Yes | |
UWDBNTXEKYRMSG
|
6.4 | Ki | 26 | — | |
WVPSKSLAZQPAKQ
|
6.4 | Ki | 3 | — | |
ZWVZORIKUNOTCS
|
6.4 | Ki | 69 | — | |
CQBBMNXXVMOFCA
|
6.3 | Ki | 39 | — | |
DOLVPVSWTLFZMQ
|
6.3 | Ki | 17 | — | |
HVXKQKFEHMGHSL
|
6.3 | Kd | 21 | — | |
HXHAJRMTJXHJJZ
|
6.3 | Ki | 52 | Yes | |
OUKYUETWWIPKQR
|
6.3 | Kd | 31 | Yes | |
ABQLLFONNKQLLB
|
6.3 | IC50 | 4 | — | |
ABXIBRWZRWHJCZ
|
6.3 | IC50 | 5 | — | |
AFHNMWQBLLGGSP
|
6.3 | IC50 | 5 | — | |
AHIOWTSQFILAEW
|
6.3 | IC50 | 5 | — | |
AYWUHPUXKGVOSD
|
6.3 | IC50 | 3 | — | |
BDVHNGIDDSJCCD
|
6.3 | IC50 | 3 | — | |
BDXLOYXFMUPOIW
|
6.3 | IC50 | 2 | — | |
BLBVISQGOQQTND
|
6.3 | IC50 | 5 | — | |
BLZCIAZUKSOFTP
|
6.3 | IC50 | 2 | — | |
BQCYIIVLNTWNSU
|
6.3 | IC50 | 3 | — | |
BVPDJKPURONCRY
|
6.3 | IC50 | 4 | — | |
BYRDCUSCDUCHLA
|
6.3 | IC50 | 4 | — | |
CMTRUERFSJKMJQ
|
6.3 | IC50 | 5 | — | |
COWKEXRPFBNPOQ
|
6.3 | IC50 | 3 | — | |
CQIIIEIHBWOUOM
|
6.3 | IC50 | 2 | — | |
DACWWGSNTVRALQ
|
6.3 | IC50 | 2 | — | |
DBXVNVVGMHBBOC
|
6.3 | IC50 | 3 | — |