Target Details
| UniProt AC | P29317 |
|---|---|
| Gene Symbol | EPHA2 |
| Protein Name | Ephrin type-A receptor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF14575 (EphA2_TM) PF25599 (Ephrin_CRD) PF01404 (Ephrin_lbd) PF00041 (fn3) PF07714 (PK_Tyr_Ser-Thr) PF00536 (SAM_1) |
Summary
- Multi-target molecules 540
- Clinical molecules 37
- Avg pChEMBL 6.74
KEGG Pathways (5)
Associated Diseases (1)
Active Molecules (540)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UGEJLCNSVIVALC
|
7.2 | Ki | 41 | — | |
WPHKIQPVPYJNAX
|
7.2 | Ki | 81 | — | |
HKSZLNNOFSGOKW
|
7.1 | IC50 | 408 | — | |
PPCIDOUXWYIBPO
|
7.1 | IC50 | 6 | — | |
UMBFDGUGXMOMHX
|
7.1 | IC50 | 12 | — | |
GALVWTFFXPRMQM
|
7.1 | Ki | 20 | — | |
LGHBDVLAHHANMX
|
7.1 | Ki | 53 | — | |
NWAUBAGBGOPJLF
|
7.1 | Ki | 51 | Yes | |
XBYVOPRDASFDMY
|
7.1 | Ki | 42 | — | |
ZGDSBEUMPIMXBM
|
7.1 | Ki | 42 | — | |
ANZRNHPEVLXURS
|
7.1 | Kd | 2 | — | |
ZGBAJMQHJDFTQJ
|
7.0 | Kd | 15 | — | |
ULCIVHLQFMURQB
|
7.0 | Kd | 2 | — | |
ZLHFILGSQDJULK
|
7.0 | Kd | 37 | Yes | |
QPDPAWXTOAVKLC
|
7.0 | Kd | 2 | — | |
DZSUJUOJJJCWGG
|
7.0 | Ki | 55 | Yes | |
FQYLJBVSYHZWLT
|
7.0 | Ki | 35 | Yes | |
KTEIFNKAUNYNJU
|
7.0 | Kd | 114 | — | |
MQRDVGBWWVWMEN
|
7.0 | Ki | 47 | — | |
NFKMFNBKEOQNPZ
|
7.0 | Ki | 43 | — | |
NFMGZVPRGVERNN
|
7.0 | Ki | 44 | — | |
NRGYZNJPCGRCLV
|
7.0 | Ki | 52 | — | |
QJIVDCJIPGAKQZ
|
7.0 | Ki | 25 | — | |
QKPLUKMJEKRAJD
|
7.0 | Ki | 30 | Yes | |
XHORJSJFHVABEA
|
7.0 | Ki | 49 | — | |
XOOAAYRIVATZNM
|
7.0 | Ki | 55 | — | |
YEHCNYAQEBQCCS
|
7.0 | Ki | 74 | — | |
WPXVVAWAHQHJPF
|
7.0 | IC50 | 41 | — | |
DKZYXHCYPUVGAF
|
7.0 | Kd | 112 | — | |
MWKSRKSEWLRPBL
|
7.0 | IC50 | 1075 | — | |
FCDUXQUQGSKWMD
|
6.9 | Kd | 2 | — | |
FLEAYYMORDPWAJ
|
6.9 | Ki | 90 | — | |
HKZKELVPGXJIMW
|
6.9 | Ki | 41 | — | |
NRZYTPAJGVTKIM
|
6.9 | Ki | 38 | — | |
OTVCFDOYUHREFJ
|
6.9 | Ki | 26 | — | |
OWFXKTOLFUQPDJ
|
6.9 | Ki | 36 | — | |
ZVPDNRVYHLRXLX
|
6.9 | Ki | 35 | Yes | |
NHHQJBCNYHBUSI
|
6.8 | Kd | 220 | — | |
KRAYLQVJPUMBPE
|
6.8 | Kd | 2 | — | |
GSXRCPJTNIGKSZ
|
6.8 | Ki | 43 | — | |
MVCOAUNKQVWQHZ
|
6.8 | IC50 | 54 | Yes | |
ODPGGGTTYSGTGO
|
6.8 | Kd | 153 | — | |
PYXQMJSGJIJHJT
|
6.8 | Ki | 28 | — | |
RWEHAHIEUDLKGT
|
6.8 | Ki | 33 | — | |
KTEIFNKAUNYNJU
|
6.8 | Ki | 48 | — | |
WKDACQVEJIVHMZ
|
6.8 | Kd | 46 | — | |
SPMVMDHWKHCIDT
|
6.7 | Kd | 30 | — | |
AIQDZMUPVYDVLB
|
6.7 | Ki | 48 | — | |
BIKYDWLMTPRSQL
|
6.7 | Ki | 50 | — | |
HCNIBOQWDVOZKF
|
6.7 | Ki | 26 | — |