Target Details
| UniProt AC | P29317 |
|---|---|
| Gene Symbol | EPHA2 |
| Protein Name | Ephrin type-A receptor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF14575 (EphA2_TM) PF25599 (Ephrin_CRD) PF01404 (Ephrin_lbd) PF00041 (fn3) PF07714 (PK_Tyr_Ser-Thr) PF00536 (SAM_1) |
Summary
- Multi-target molecules 540
- Clinical molecules 37
- Avg pChEMBL 6.74
KEGG Pathways (5)
Associated Diseases (1)
Active Molecules (540)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RNCWMUAJKHOSIS
|
7.3 | IC50 | 2 | — | |
RPLCLUCJTHAIOW
|
7.3 | IC50 | 4 | — | |
SBYHOEZLNRTZNU
|
7.3 | IC50 | 2 | — | |
SFASAOFVHLMKPH
|
7.3 | IC50 | 3 | — | |
SHQDTJIUTBSGPO
|
7.3 | IC50 | 3 | — | |
SHQICENFGOEXMY
|
7.3 | IC50 | 4 | — | |
STKWUQHKDUWIGO
|
7.3 | IC50 | 4 | — | |
SVJQCEUABCZTGM
|
7.3 | IC50 | 3 | — | |
SWQHCAPKAPNADM
|
7.3 | IC50 | 3 | — | |
TWMPXXRMSJFJSY
|
7.3 | IC50 | 3 | — | |
TXHOCWWJSGCZLC
|
7.3 | Ki | 18 | — | |
TYDHEVOVJOWAEX
|
7.3 | IC50 | 3 | — | |
UCKGFSDFZDKPJE
|
7.3 | IC50 | 3 | — | |
UHDUHDKGRPVSSW
|
7.3 | IC50 | 3 | — | |
UIODCBCHOOHDBJ
|
7.3 | IC50 | 3 | — | |
UJKCNZDTMJJLEP
|
7.3 | IC50 | 3 | — | |
UOVCGJXDGOGOCZ
|
7.3 | Ki | 59 | — | |
USQQETNBKWVAHU
|
7.3 | IC50 | 2 | — | |
USTBWYHTULQCGO
|
7.3 | IC50 | 2 | — | |
UTCBITIGWNRGAW
|
7.3 | IC50 | 3 | — | |
UULADMWDIINHOI
|
7.3 | IC50 | 2 | — | |
VBHNSELTUCCXDK
|
7.3 | IC50 | 3 | — | |
VBRGKAXLFVNGHF
|
7.3 | IC50 | 3 | — | |
VDNKDMALAXYLFZ
|
7.3 | IC50 | 3 | — | |
VETATMCQXNIHSE
|
7.3 | IC50 | 3 | — | |
VGKSTMJEMVAVLY
|
7.3 | IC50 | 3 | — | |
VNKOLNHCWLKONF
|
7.3 | IC50 | 3 | — | |
VOQVXZHQBTXEHV
|
7.3 | IC50 | 3 | — | |
VTKBQOHBYWWZNL
|
7.3 | IC50 | 3 | — | |
VWLDHVBJTHRWJI
|
7.3 | IC50 | 3 | — | |
VXJCKEGWFQFYGD
|
7.3 | IC50 | 4 | — | |
WEUDFLZPDBNRRQ
|
7.3 | IC50 | 2 | — | |
WPKITCNGCYKRNZ
|
7.3 | IC50 | 3 | — | |
WTOQAKRNPRFBML
|
7.3 | IC50 | 3 | — | |
WVXLPNDNCDLCQW
|
7.3 | IC50 | 2 | — | |
XYNKEFOTYHJQFS
|
7.3 | IC50 | 3 | — | |
YAEMBTULTQVMDI
|
7.3 | IC50 | 3 | — | |
YGRIEMSMFNEFKK
|
7.3 | IC50 | 2 | — | |
YJHVTCUKZLXENT
|
7.3 | IC50 | 2 | — | |
YVZZAELYZKUMKK
|
7.3 | IC50 | 3 | — | |
ZDTMGSSRQLKYTK
|
7.3 | IC50 | 5 | — | |
ZIKUMDQTYYWCRD
|
7.3 | IC50 | 2 | — | |
ZJFHLSCSEWIASA
|
7.3 | IC50 | 2 | — | |
ZJOIMYDGIVGAMA
|
7.3 | IC50 | 3 | — | |
ZKUNKJWGKBMFCR
|
7.3 | IC50 | 4 | — | |
ZPNITDGPLQDXIJ
|
7.3 | IC50 | 2 | — | |
ZPNSUJMOMIXELJ
|
7.3 | IC50 | 4 | — | |
ZTUNVYDNGSGYLT
|
7.3 | IC50 | 4 | — | |
ZVTLPVGUCZTBMB
|
7.3 | IC50 | 2 | — | |
QONPPIZSNSSCSK
|
7.2 | Ki | 45 | Yes |