Target Details
| UniProt AC | P29317 |
|---|---|
| Gene Symbol | EPHA2 |
| Protein Name | Ephrin type-A receptor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF14575 (EphA2_TM) PF25599 (Ephrin_CRD) PF01404 (Ephrin_lbd) PF00041 (fn3) PF07714 (PK_Tyr_Ser-Thr) PF00536 (SAM_1) |
Summary
- Multi-target molecules 540
- Clinical molecules 37
- Avg pChEMBL 6.74
KEGG Pathways (5)
Associated Diseases (1)
Active Molecules (540)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KJLBXUKNKUWCED
|
7.3 | IC50 | 2 | — | |
KKYPRNBBPBRJQX
|
7.3 | Ki | 40 | — | |
KLCMTXVLRHGAEO
|
7.3 | IC50 | 3 | — | |
KNAPWFDGXYXHLO
|
7.3 | IC50 | 3 | — | |
KOHLHBQFFZUSET
|
7.3 | IC50 | 2 | — | |
KOSFAPNTMAEMEM
|
7.3 | IC50 | 3 | — | |
KPUHDJMEVYIACF
|
7.3 | IC50 | 3 | — | |
KSFMKTNHEIDMFI
|
7.3 | IC50 | 2 | — | |
KSQYAAKEJFJFOV
|
7.3 | IC50 | 3 | — | |
KTADNURCUXHCJM
|
7.3 | IC50 | 4 | — | |
KTBQYTJFMLOVMP
|
7.3 | IC50 | 5 | — | |
KYGRLSQAAKVRBS
|
7.3 | IC50 | 3 | — | |
KZIOAIIQBIYJTQ
|
7.3 | IC50 | 4 | — | |
LLUVEMMROYJZEI
|
7.3 | IC50 | 3 | — | |
LUAHOZHPDVOBIY
|
7.3 | IC50 | 4 | — | |
MAJPXTGDUCKEGK
|
7.3 | IC50 | 2 | — | |
MFZHNTIFSFFVQH
|
7.3 | IC50 | 3 | — | |
NJQIBYWJBXKSRO
|
7.3 | IC50 | 4 | — | |
NJQIBYWJBXKSRO
|
7.3 | IC50 | 5 | — | |
NJUOOEIYXARLMK
|
7.3 | IC50 | 3 | — | |
NQRHMWLUXWPKIS
|
7.3 | IC50 | 3 | — | |
NTVIDJBDSIQHHB
|
7.3 | IC50 | 4 | — | |
NWWPZALFLBATKW
|
7.3 | IC50 | 3 | — | |
OEGXYNWEJSFYPO
|
7.3 | IC50 | 5 | — | |
OGSIXPVUAMTENQ
|
7.3 | IC50 | 4 | — | |
OIGAOMAHSFGBDQ
|
7.3 | IC50 | 3 | — | |
OSKITHVLDNYNOG
|
7.3 | IC50 | 3 | — | |
OUPSOAXLJSDWRF
|
7.3 | IC50 | 3 | — | |
OXOZNJXEGUXWOO
|
7.3 | IC50 | 5 | — | |
PDSTVLMICZJXNC
|
7.3 | IC50 | 2 | — | |
PDWKXNAYFBPNOH
|
7.3 | IC50 | 3 | — | |
PFWWSXZJVNFSKD
|
7.3 | IC50 | 3 | — | |
PGROYXXCSUBAOJ
|
7.3 | IC50 | 2 | — | |
PKMKYIJSZRWDDY
|
7.3 | IC50 | 2 | — | |
PLPFTGVPIXWCIC
|
7.3 | IC50 | 3 | — | |
PQDLFPSEZJTCDS
|
7.3 | IC50 | 3 | — | |
PWNBTHIQJMPMTI
|
7.3 | IC50 | 4 | — | |
PYAFRFDCPSOBJI
|
7.3 | IC50 | 3 | — | |
PZXCQEQVQAFMLY
|
7.3 | IC50 | 3 | — | |
QFHBQKXGJZQISJ
|
7.3 | IC50 | 3 | — | |
QHJQGPXGMHCLDZ
|
7.3 | IC50 | 3 | — | |
QHTZGTDGFHTCOG
|
7.3 | IC50 | 3 | — | |
QOEMXTGSYTXSBD
|
7.3 | IC50 | 4 | — | |
QOLKGXDWVMWHLS
|
7.3 | IC50 | 3 | — | |
QPCXTIGWORLPNS
|
7.3 | IC50 | 3 | — | |
QPNYAXXXUXFKDG
|
7.3 | IC50 | 4 | — | |
QTMIYSYKAIPGKO
|
7.3 | IC50 | 3 | — | |
QYJJHEKFWCNKKZ
|
7.3 | IC50 | 2 | — | |
RFGYFZFUMBQSCW
|
7.3 | IC50 | 6 | — | |
RGUFKCMSOMSTHM
|
7.3 | IC50 | 3 | — |