Target Details
| UniProt AC | P29317 |
|---|---|
| Gene Symbol | EPHA2 |
| Protein Name | Ephrin type-A receptor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF14575 (EphA2_TM) PF25599 (Ephrin_CRD) PF01404 (Ephrin_lbd) PF00041 (fn3) PF07714 (PK_Tyr_Ser-Thr) PF00536 (SAM_1) |
Summary
- Multi-target molecules 540
- Clinical molecules 37
- Avg pChEMBL 6.74
KEGG Pathways (5)
Associated Diseases (1)
Active Molecules (540)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ASUKBBADPXBJFR
|
7.3 | IC50 | 2 | — | |
AVADFQHEIADTFF
|
7.3 | IC50 | 3 | — | |
BADQNHXUQWKUBJ
|
7.3 | IC50 | 3 | — | |
BLDLZCARBOCFMX
|
7.3 | IC50 | 2 | — | |
BLPHPXYTDDFZER
|
7.3 | IC50 | 2 | — | |
BTGGKWOJEKOLEQ
|
7.3 | IC50 | 3 | — | |
CHESBDRRLQCAEW
|
7.3 | IC50 | 2 | — | |
CJQHDRRRDSNFOQ
|
7.3 | IC50 | 2 | — | |
CKIBKYNCWLLXRU
|
7.3 | IC50 | 3 | — | |
CMTRUERFSJKMJQ
|
7.3 | IC50 | 4 | — | |
CPDVUYTVYREKJG
|
7.3 | IC50 | 3 | — | |
DCHUHENWAKOFLF
|
7.3 | IC50 | 4 | — | |
DGJOZXUZTUDBOH
|
7.3 | IC50 | 2 | — | |
DLZJESFGQYKOIJ
|
7.3 | IC50 | 3 | — | |
DNTJORWEWRMHBN
|
7.3 | IC50 | 4 | — | |
DSXVRWQRFDVWBE
|
7.3 | IC50 | 2 | — | |
DVEHRUCQBHJWFA
|
7.3 | IC50 | 5 | — | |
FBKDSVZIPCLRHF
|
7.3 | IC50 | 3 | — | |
FEBOQCZDPJAXJB
|
7.3 | IC50 | 2 | — | |
FFDFDDSWSCPPMW
|
7.3 | IC50 | 3 | — | |
FIIMJONANOAMJA
|
7.3 | IC50 | 2 | — | |
FKFOSUXFCGMEJY
|
7.3 | IC50 | 3 | — | |
FSJDACURTSWGHC
|
7.3 | IC50 | 3 | — | |
FWOWVRMQIDGFHG
|
7.3 | IC50 | 3 | — | |
GFMZMGTWUAXGMZ
|
7.3 | IC50 | 4 | — | |
GQBGDMIPLRKLGO
|
7.3 | IC50 | 3 | — | |
GQHKXXVKPUENOH
|
7.3 | IC50 | 3 | — | |
GVKSFOCLIXUHCD
|
7.3 | IC50 | 2 | — | |
GVQHNFSUVYXILE
|
7.3 | IC50 | 3 | — | |
HFDJFCJNMFTWOT
|
7.3 | IC50 | 2 | — | |
HFTHZTJJBJKTGD
|
7.3 | IC50 | 3 | — | |
HKHCOFOLZLSONC
|
7.3 | IC50 | 3 | — | |
HKKAQXNDAFGPHA
|
7.3 | IC50 | 2 | — | |
HYOURUDRVAZLAG
|
7.3 | IC50 | 4 | — | |
HZQVPHRLYRINCU
|
7.3 | IC50 | 3 | — | |
IAULTELZJHNXGT
|
7.3 | IC50 | 3 | — | |
ICKYQMYVKOGDAJ
|
7.3 | IC50 | 4 | — | |
IFVXCNKRSUKURE
|
7.3 | IC50 | 4 | — | |
IFVXCNKRSUKURE
|
7.3 | IC50 | 5 | — | |
IHALJECVDZIKBK
|
7.3 | IC50 | 2 | — | |
IUMNCIHHFXUHBR
|
7.3 | IC50 | 3 | — | |
JAGHRSZQQGMOBS
|
7.3 | IC50 | 3 | — | |
JDSDNLQKCIMLFG
|
7.3 | IC50 | 3 | — | |
JHVXCKPKPWJTHM
|
7.3 | IC50 | 4 | — | |
JJHKGTMOROVPCK
|
7.3 | IC50 | 2 | — | |
JRGYGHIKWBYTFJ
|
7.3 | IC50 | 3 | — | |
JXWOGDLXVWLJMH
|
7.3 | IC50 | 3 | — | |
KGRQWBCQDURFIP
|
7.3 | IC50 | 3 | — | |
KHSJGHHCLKKKKU
|
7.3 | IC50 | 4 | — | |
KHSJGHHCLKKKKU
|
7.3 | IC50 | 5 | — |