Target Details
| UniProt AC | P29317 |
|---|---|
| Gene Symbol | EPHA2 |
| Protein Name | Ephrin type-A receptor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF14575 (EphA2_TM) PF25599 (Ephrin_CRD) PF01404 (Ephrin_lbd) PF00041 (fn3) PF07714 (PK_Tyr_Ser-Thr) PF00536 (SAM_1) |
Summary
- Multi-target molecules 540
- Clinical molecules 37
- Avg pChEMBL 6.74
KEGG Pathways (5)
Associated Diseases (1)
Active Molecules (540)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MFHPFBVKYHTFKA
|
6.0 | IC50 | 4 | — | |
MFJPJXJGMGXYLR
|
6.0 | IC50 | 3 | — | |
MIAAVOBHHDBHSW
|
6.0 | IC50 | 5 | — | |
MTJYFGYTUQVKPE
|
6.0 | IC50 | 4 | — | |
OMTQJDUOTIRCBU
|
6.0 | IC50 | 3 | — | |
OUEOJFCFMCXADD
|
6.0 | IC50 | 6 | — | |
PVTTWYOJLADNCZ
|
6.0 | IC50 | 4 | — | |
PWDUFJSWDUGFRW
|
6.0 | IC50 | 4 | — | |
PZRQHOBLMLLAAY
|
6.0 | IC50 | 4 | — | |
QEGLEPAPQKOMLB
|
6.0 | IC50 | 4 | — | |
QEIAACVSNFOMGZ
|
6.0 | IC50 | 4 | — | |
QQGZOWNAHJAXCG
|
6.0 | IC50 | 4 | — | |
RDFSWUCGNZTNGD
|
6.0 | IC50 | 4 | — | |
RPGBQFNDFPEOON
|
6.0 | Ki | 22 | — | |
RSQKKUZJTBAHBG
|
6.0 | IC50 | 5 | — | |
RUBSXJGCJAOKHK
|
6.0 | IC50 | 3 | — | |
RVMLSAUWFLLGAT
|
6.0 | IC50 | 5 | — | |
RYYNGWLOYLRZLK
|
6.0 | Ki | 104 | — | |
SROSEDFOBYVYCH
|
6.0 | IC50 | 3 | — | |
SYLHDCKBBWIRTH
|
6.0 | IC50 | 3 | — | |
TZKZSFJMVHBLGG
|
6.0 | IC50 | 3 | — | |
UAUVSHOAYLPSOU
|
6.0 | IC50 | 4 | — | |
UIBFVYOIDXCKPI
|
6.0 | IC50 | 4 | — | |
UJTDMNARLIOVGT
|
6.0 | IC50 | 4 | — | |
UPTQFQIWDCTNMU
|
6.0 | IC50 | 4 | — | |
VENHPOQTVRCHJV
|
6.0 | IC50 | 6 | — | |
VKCKBMWVXBACHI
|
6.0 | IC50 | 3 | — | |
VRXGZDANOSIHSR
|
6.0 | IC50 | 4 | — | |
WEAZKUYDPMNZPH
|
6.0 | IC50 | 3 | — | |
XCAOLOJNZVNRSK
|
6.0 | IC50 | 5 | — | |
XCMSAHCDUHXACI
|
6.0 | IC50 | 3 | — | |
XDESVXWYQFZXJJ
|
6.0 | IC50 | 4 | — | |
XJDLHHHTZRBRFC
|
6.0 | IC50 | 4 | — | |
XNWJPKXDERVJBQ
|
6.0 | IC50 | 3 | — | |
XRRHFQQSBXKXCI
|
6.0 | IC50 | 4 | — | |
ZEFUNPUAOZNDER
|
6.0 | IC50 | 4 | — | |
ZEFUNPUAOZNDER
|
6.0 | IC50 | 4 | — | |
ZFLUWPGMYIIBJD
|
6.0 | IC50 | 4 | — | |
ZHMULGIXCIACTQ
|
6.0 | IC50 | 2 | — | |
ZWBURYJEEIVZFT
|
6.0 | IC50 | 4 | — |