Target Details
| UniProt AC | P29317 |
|---|---|
| Gene Symbol | EPHA2 |
| Protein Name | Ephrin type-A receptor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF14575 (EphA2_TM) PF25599 (Ephrin_CRD) PF01404 (Ephrin_lbd) PF00041 (fn3) PF07714 (PK_Tyr_Ser-Thr) PF00536 (SAM_1) |
Summary
- Multi-target molecules 540
- Clinical molecules 37
- Avg pChEMBL 6.74
KEGG Pathways (5)
Associated Diseases (1)
Active Molecules (540)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZTASYFQODPYQIW
|
6.3 | IC50 | 4 | — | |
ZYDWOISDXFZQRM
|
6.3 | IC50 | 3 | — | |
MFAQYJIYDMLAIM
|
6.2 | Kd | 130 | Yes | |
GCBJDOWIQHMCMR
|
6.2 | Ki | 84 | — | |
VWMJHAFYPMOMGF
|
6.2 | Kd | 15 | — | |
YEPNVBNYCRGZRX
|
6.2 | Ki | 26 | — | |
MGGBYMDAPCCKCT
|
6.2 | Kd | 23 | — | |
WRLSAGKQYAORBC
|
6.2 | IC50 | 12 | — | |
ONIQOQHATWINJY
|
6.1 | Kd | 25 | — | |
IKLGYJACVCXYIL
|
6.1 | IC50 | 5 | — | |
SMPGEBOIKULBCT
|
6.1 | IC50 | 15 | — | |
GCYXEGSPUDSZJY
|
6.1 | Ki | 82 | — | |
GEGCXGMFUYJULA
|
6.1 | Ki | 30 | Yes | |
GMYYMEOGFRKSFS
|
6.1 | Ki | 29 | — | |
MHCPAORAYMTGCZ
|
6.1 | Ki | 37 | — | |
MLDQJTXFUGDVEO
|
6.1 | Ki | 85 | Yes | |
MULNSLQVKKUPJN
|
6.1 | Ki | 41 | — | |
UIARLYUEJFELEN
|
6.1 | Kd | 289 | Yes | |
YPDWGKSFVMASOZ
|
6.1 | Ki | 5 | — | |
GCIKSSRWRFVXBI
|
6.1 | Kd | 109 | Yes | |
HEPDAJRNJBNJAE
|
6.1 | IC50 | 15 | Yes | |
FNHKPVJBJVTLMP
|
6.1 | Kd | 29 | — | |
QQWUGDVOUVUTOY
|
6.0 | Kd | 231 | Yes | |
CSGQVNMSRKWUSH
|
6.0 | Kd | 21 | — | |
ATNQJIZWZJGBST
|
6.0 | IC50 | 4 | — | |
AYHZKTTUBQETRW
|
6.0 | IC50 | 3 | — | |
BACURHXRJBKWQO
|
6.0 | IC50 | 4 | — | |
BBSZLPWCQBIFJS
|
6.0 | IC50 | 4 | — | |
BZYUMECEYCQIQF
|
6.0 | IC50 | 3 | — | |
CJQXHWIFGRLKGH
|
6.0 | IC50 | 3 | — | |
CKTFKRFHQMIOAN
|
6.0 | IC50 | 5 | — | |
CMDXLFALYMWXLO
|
6.0 | IC50 | 4 | — | |
CXTBYZCZYIJFDG
|
6.0 | IC50 | 5 | — | |
DUNQTRHEGUIEHU
|
6.0 | IC50 | 4 | — | |
FCDDMXMTHQYQBS
|
6.0 | IC50 | 4 | — | |
FGQMTFNXIHXUTF
|
6.0 | IC50 | 3 | — | |
GBVHHGINCYVVRZ
|
6.0 | IC50 | 4 | — | |
GNMRWTTWRQISEY
|
6.0 | IC50 | 3 | — | |
GOMLGIJFTVXGSO
|
6.0 | IC50 | 4 | — | |
HDJUYMWWZOHAHK
|
6.0 | IC50 | 5 | — | |
IBKXZCOYYLYZQJ
|
6.0 | IC50 | 4 | — | |
IGXXJHAWUNOEDC
|
6.0 | IC50 | 5 | — | |
ILENFMLSOQJLGD
|
6.0 | IC50 | 4 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
JHBNNKDJEPHKTQ
|
6.0 | IC50 | 4 | — | |
JIBJCRRXQHEKJX
|
6.0 | IC50 | 5 | — | |
JXPMQIMIJGMOIG
|
6.0 | IC50 | 3 | — | |
KTJGGFYHAOWIMA
|
6.0 | IC50 | 4 | — | |
LARWQCXRXJJFLU
|
6.0 | IC50 | 3 | — | |
LCTKSVLGCZKLFJ
|
6.0 | IC50 | 3 | — |