Target Details
| UniProt AC | P29317 |
|---|---|
| Gene Symbol | EPHA2 |
| Protein Name | Ephrin type-A receptor 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF14575 (EphA2_TM) PF25599 (Ephrin_CRD) PF01404 (Ephrin_lbd) PF00041 (fn3) PF07714 (PK_Tyr_Ser-Thr) PF00536 (SAM_1) |
Summary
- Multi-target molecules 540
- Clinical molecules 37
- Avg pChEMBL 6.74
KEGG Pathways (5)
Associated Diseases (1)
Active Molecules (540)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SUXYGJZMCWKJJI
|
9.2 | IC50 | 26 | Yes | |
AQSSMEORRLJZLU
|
9.0 | Kd | 34 | Yes | |
JTWMOWRMSZZHDR
|
8.6 | IC50 | 13 | — | |
CXBBWVXSZINRCS
|
8.5 | Ki | 41 | — | |
ZBNZXTGUTAYRHI
|
8.5 | Kd | 102 | Yes | |
SEJGTFPOEJWEGG
|
8.4 | Kd | 149 | — | |
VAARYSWULJUGST
|
8.3 | Kd | 119 | Yes | |
OWRXHGAFWZFFCW
|
8.2 | Ki | 113 | — | |
PHXJVRSECIGDHY
|
8.2 | Kd | 59 | — | |
SFCBIFOAGRZJNX
|
8.1 | Kd | 22 | — | |
XKFTZKGMDDZMJI
|
8.1 | Kd | 64 | Yes | |
KNARVZUUCLIBGV
|
8.0 | Ki | 33 | — | |
GXEGTVQATHKFDH
|
8.0 | IC50 | 10 | Yes | |
HYWXBDQAYLPMIX
|
8.0 | IC50 | 3 | Yes | |
XHBVYDAKJHETMP
|
8.0 | IC50 | 24 | Yes | |
UOOZSMNSBYVUGZ
|
7.9 | Ki | 32 | — | |
YDOPLCNFRXOHCC
|
7.9 | Ki | 28 | — | |
VREZKFPACUPTJS
|
7.9 | IC50 | 5 | — | |
YOBIWCLAYQWPPW
|
7.9 | IC50 | 23 | — | |
ZCCPLJOKGAACRT
|
7.9 | IC50 | 599 | — | |
CXQHYVUVSFXTMY
|
7.9 | Kd | 154 | — | |
YXARVHZXTQVAOP
|
7.9 | IC50 | 11 | — | |
BNRXMSGHPVYSDK
|
7.8 | IC50 | 24 | — | |
XCHWBXBDZRJVDP
|
7.8 | Ki | 51 | — | |
VKBFHTIUXUCYRQ
|
7.8 | Ki | 66 | — | |
DZUFTTMDQLYMBE
|
7.7 | IC50 | 10 | Yes | |
LQSGDXCDNZWTJN
|
7.7 | IC50 | 17 | — | |
UBPYILGKFZZVDX
|
7.7 | Kd | 130 | Yes | |
ALKJNCZNEOTEMP
|
7.7 | Kd | 55 | — | |
HHCBMISMPSAZBF
|
7.7 | IC50 | 23 | — | |
JSDGKSMNPHJDFK
|
7.7 | Ki | 35 | — | |
MCCCQFAOMZMZKE
|
7.7 | Ki | 52 | — | |
ULHGAQSVFPOUDY
|
7.7 | Ki | 43 | — | |
WFTZMAAMCVPJJT
|
7.7 | Ki | 26 | — | |
XJSFDMGICAWQFS
|
7.7 | Ki | 60 | — | |
XYXLUJQBBIBJFV
|
7.7 | Ki | 36 | — | |
UQRCJCNVNUFYDX
|
7.6 | Kd | 27 | — | |
DGSMEFWSLXFLQA
|
7.6 | IC50 | 2 | — | |
DKNUPRMJNUQNHR
|
7.5 | Kd | 33 | — | |
CFIBXVQLBVNOHW
|
7.5 | Ki | 64 | — | |
XKFTZKGMDDZMJI
|
7.5 | Ki | 56 | — | |
XLFYOIVELARSKP
|
7.5 | Ki | 33 | — | |
NWEIPABWNQPRCZ
|
7.5 | IC50 | 7 | Yes | |
PTVPBWWDGZSEAF
|
7.4 | Ki | 63 | — | |
ZXLFIHLBHMLHFJ
|
7.4 | Ki | 31 | — | |
AAWZYZGJDOSLSU
|
7.3 | IC50 | 4 | — | |
ABXIBRWZRWHJCZ
|
7.3 | IC50 | 3 | — | |
AENQVVCMBGUAQO
|
7.3 | IC50 | 2 | — | |
AKMSPGIAHZAWSW
|
7.3 | IC50 | 3 | — | |
ALVFQMWHUJBCDD
|
7.3 | IC50 | 2 | — |