Target Details
| UniProt AC | P29120 |
|---|---|
| Gene Symbol | PCSK1 |
| Protein Name | Neuroendocrine convertase 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01483 (P_proprotein) PF00082 (Peptidase_S8) PF12177 (Proho_convert) PF16470 (S8_pro-domain) |
Summary
- Multi-target molecules 11
- Clinical molecules 0
- Avg pChEMBL 8.2
Associated Diseases (2)
Active Molecules (11)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RARQEZVPGNQDRL
|
9.1 | Ki | 5 | — | |
YGMAIAXBJLVVLI
|
9.1 | Ki | 5 | — | |
UXEFAKYOWKPLSZ
|
8.8 | Ki | 4 | — | |
YIMSHXFWBSXLKW
|
8.8 | Ki | 4 | — | |
NHBJTTGFHCHQHS
|
8.7 | Ki | 6 | — | |
QMAXHSLPLMYIPN
|
8.4 | Ki | 6 | — | |
CLTYJDDMFQEKEL
|
8.4 | Ki | 6 | — | |
ACPMDCNBPZRQGO
|
7.3 | Ki | 4 | — | |
HCRNWNCAUNWLJZ
|
7.3 | Ki | 4 | — | |
LEEIZVYTIHJJNF
|
7.2 | Ki | 4 | — | |
KWHYASXOKFJBKD
|
7.2 | Ki | 4 | — |