Target Details
| UniProt AC | P28566 |
|---|---|
| Gene Symbol | HTR1E |
| Protein Name | 5-hydroxytryptamine receptor 1E |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00001 (7tm_1) |
Summary
- Multi-target molecules 60
- Clinical molecules 7
- Avg pChEMBL 6.64
KEGG Pathways (5)
Active Molecules (60)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ORJIHHLJBCQRBS
|
6.1 | Ki | 6 | — | |
YOZGUJJGVBYZQY
|
6.1 | Ki | 7 | — | |
ASXGJMSKWNBENU
|
6.1 | Ki | 12 | Yes | |
LWNZEHWQIHUHGP
|
6.0 | Ki | 7 | — | |
WKZLNEWVIAGNAW
|
6.0 | Ki | 11 | — | |
DVALOPXWVWHIHY
|
6.0 | Ki | 10 | — | |
JRNUKVFYILMMLX
|
6.0 | Ki | 16 | — | |
QYVHPITUKBNDGT
|
6.0 | IC50 | 2 | — | |
QZUDBNBUXVUHMW
|
6.0 | Ki | 39 | Yes | |
YOGJZQGRTVMCPY
|
6.0 | IC50 | 17 | — |