Target Details
UniProt ACP28566
Gene SymbolHTR1E
Protein Name5-hydroxytryptamine receptor 1E
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 60
  • Clinical molecules 7
  • Avg pChEMBL 6.64
Top Co-occurrence Targets
Active Molecules (60)
InChIKey pChEMBL Type Targets Clinical
OPCCXGXGEHABFP 9.8 Kd 17
BCGWQEUPMDMJNV 9.0 IC50 30 Yes
QBRLVMQBZIFWTB 8.2 Ki 12
QZAYGJVTTNCVMB 8.2 Ki 17
VSWBSWWIRNCQIJ 8.0 Ki 23
BIXJFIJYBLJTMK 7.4 Ki 3
SPCIYGNTAMCTRO 7.4 Ki 15
BKRGVLQUQGGVSM 7.3 Ki 26 Yes
WVVSZNPYNCNODU 7.1 Ki 2
UNBRKDKAWYKMIV 7.0 Ki 12
VAYOSLLFUXYJDT 7.0 Ki 19
LXWHNYYETIMYQL 7.0 IC50 3
YZDFADGMVOSVIX 7.0 Ki 16
RLDFVSFNVOLFEU 6.9 Ki 5
YMHOBZXQZVXHBM 6.9 Ki 13
XEDHVZKDSYZQBF 6.9 Ki 7
DUKNIHFTDAXJON 6.8 Ki 11
CJKGAQSNLYKBKH 6.7 Ki 9
DUKNIHFTDAXJON 6.7 Ki 17
DUKNIHFTDAXJON 6.7 Ki 16
DUKNIHFTDAXJON 6.7 Ki 13
VNICFCQJUVFULD 6.7 Ki 15
DUKNIHFTDAXJON 6.5 Ki 12
HDOZVRUNCMBHFH 6.5 Ki 26 Yes
XRJGWSMTLAFHBN 6.5 Ki 21
MVWVFYHBGMAFLY 6.4 Ki 31 Yes
LQEATNFJCMVKAC 6.4 Ki 14
QXXXZTFUFKESQI 6.4 IC50 2
HCWQGDLBIKOJPM 6.4 Ki 12
WYWIFABBXFUGLM 6.4 Ki 17
GZKLJWGUPQBVJQ 6.4 Ki 24 Yes
ZUXABONWMNSFBN 6.4 Ki 29
ZSTKHSQDNIGFLM 6.4 Ki 22
DMULVCHRPCFFGV 6.3 Ki 16
DZXZPVGWRZCXDH 6.3 Ki 20
HGRHWEAUHXYNNP 6.3 Ki 16
ALTKABGEMCJWJH 6.3 Ki 15
ZKIAIYBUSXZPLP 6.3 Ki 29
HTDIOUCPOHFDQH 6.3 Ki 14
JWPAYBAIIARWMG 6.3 Ki 19
FXMWUTGUCAKGQL 6.2 Ki 10
JUQLTPCYUFPYKE 6.2 Ki 25
KKIMDKMETPPURN 6.2 Ki 8
XCGSFFUVFURLIX 6.2 Ki 17
DMDNERFCUCYCGM 6.2 IC50 9
VDRGNAMREYBIHA 6.2 Ki 11
RUJUSCZEDDAGAW 6.2 Ki 4
LUZRJRNZXALNLM 6.2 Ki 20
NZKYTYHIERLZBG 6.1 Ki 8
ALRBWNXPNRLJKC 6.1 Ki 10
2D structure