Target Details
UniProt ACP28472
Gene SymbolGABRB3
Protein NameGamma-aminobutyric acid receptor subunit beta-3
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 1,198
  • Clinical molecules 0
  • Avg pChEMBL 7.71
Top Co-occurrence Targets
Active Molecules (1,198)
InChIKey pChEMBL Type Targets Clinical
KIDPGPYNXRNUGP 9.3 Ki 3
NJUMMJUUDUYSKB 9.3 IC50 16
AJWPZYMLAILYCO 9.3 Ki 5
ANARVVNNNQSSPE 9.3 Ki 3
BYMDBFGHCDTBMT 9.3 IC50 16
FPRLTMYWIBRCQM 9.3 Ki 3
IUHKSTINHDUYRO 9.3 IC50 16
LWUDDYHYYNNIQI 9.3 Ki 7
UIKTZQCQKHUZHT 9.3 Ki 3
VJVAWKPXJCDEQG 9.3 IC50 16
COIHYICCVMGEJO 9.3 Ki 3
FNCCIRFBYGUBRQ 9.3 Ki 5
NTQIDFIQUNKLIH 9.3 Ki 5
QIWRIQRYIRGJCG 9.3 Ki 4
BPTASZCHRIMWEF 9.3 Ki 6
ZHPXUSDIAXKCGY 9.3 Ki 3
GMDXFYPWVIKBFF 9.3 Ki 4
LVJXDIPOLXCUPP 9.3 Ki 3
KJDDJAPSHCVDDC 9.2 Ki 3
FAEJWVCMADNLAQ 9.2 Ki 4
UPMDLTAPSSWEPU 9.2 Ki 4
BLJPKQXXDFIIFR 9.2 IC50 16
GIUPLTIPPKYWPM 9.2 Ki 3
LULPFCFGFHHBEZ 9.2 Ki 3
OABMKUYJAYGQHV 9.2 Ki 3
SPUDBCPXWITYDE 9.2 Ki 3
XHCCKQJTDGEMHT 9.2 Ki 3
XJMIBNLJFYSGAR 9.2 IC50 16
LYZCPNJIFQNJQM 9.2 Ki 3
MTOXGGJOEHOEJT 9.2 Ki 5
NZMJFRXKGUCYNP 9.2 Ki 6
FXXAEVWLAOMRSI 9.2 Ki 4
UJBOQYCZTOTBAN 9.2 Ki 4
BKIXSCDBYYIHQI 9.2 Ki 5
KVQKVRWATUWLAO 9.2 Ki 5
LICVBNQRZFPUHS 9.2 Ki 4
QZDWWRKBDPYMIP 9.2 Ki 6
JLCBYDSLJHLQQB 9.1 Ki 5
ISZRIZPRXUQOMU 9.1 Ki 5
BQDUNOMMYOKHEP 9.1 Ki 6
CNEHRQMKOUFFMX 9.1 Ki 3
DQKNTSFPZMVKNA 9.1 Ki 3
GXPHYMCBGKIIKN 9.1 Ki 3
ILFZZMYJRPZIPF 9.1 Ki 5
JFGUJXZLJIUVPZ 9.1 IC50 16
LYFROTHEKIFZAU 9.1 IC50 16
RYIVVNHBYBYXHF 9.1 IC50 16
SRAWBNFSMIHBEM 9.1 Ki 8
VZKRZUPJCVFVGR 9.1 IC50 16
LLHQBHOWDZNCNK 9.1 Ki 5
2D structure