Target Details
| UniProt AC | P28347 |
|---|---|
| Gene Symbol | TEAD1 |
| Protein Name | Transcriptional enhancer factor TEF-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01285 (TEA) PF17725 (YBD) |
Summary
- Multi-target molecules 211
- Clinical molecules 0
- Avg pChEMBL 7.26
KEGG Pathways (3)
Associated Diseases (1)
Active Molecules (211)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZDNOXXCLYNWLQC
|
6.8 | IC50 | 3 | — | |
KMMLWTJOWPPZLE
|
6.8 | IC50 | 3 | — | |
OKZNWIMTGZSWTI
|
6.8 | IC50 | 3 | — | |
CAORLWHRUGUSCD
|
6.8 | IC50 | 4 | — | |
LSSHXGKZWQPQOF
|
6.8 | IC50 | 3 | — | |
WRNUURQTNJCUCD
|
6.8 | IC50 | 3 | — | |
KXCKTSLTRHZBEF
|
6.8 | IC50 | 4 | — | |
PNHFKELIFBUTPW
|
6.8 | IC50 | 4 | — | |
LCJVJLBBFQAZCD
|
6.7 | IC50 | 2 | — | |
PQYZEJLNRTWTIU
|
6.7 | IC50 | 3 | — | |
STFNGTPHVKXUJX
|
6.7 | IC50 | 2 | — | |
WOHSOQGAUZKYLE
|
6.7 | IC50 | 2 | — | |
WRNUURQTNJCUCD
|
6.7 | IC50 | 3 | — | |
WXFBUGGCMXZIKK
|
6.7 | IC50 | 2 | — | |
DJGXOJSWOLDZPW
|
6.7 | IC50 | 4 | — | |
NWGUMSQMFYGSDM
|
6.7 | IC50 | 3 | — | |
PYYJLQOPDWLFDU
|
6.7 | IC50 | 2 | — | |
REXPRRRRXYZDCK
|
6.7 | IC50 | 2 | — | |
JLFVYIWUQHPMTB
|
6.7 | Kd | 2 | — | |
KWESWHHLPBOTRP
|
6.7 | IC50 | 3 | — | |
RIHGSIDKHRTLDB
|
6.7 | IC50 | 3 | — | |
UWHSYKJHXZYVDN
|
6.7 | IC50 | 4 | — | |
AAYVOUUBHRKCMZ
|
6.6 | IC50 | 4 | — | |
YZJALBBGXPGUIR
|
6.6 | IC50 | 3 | — | |
KCBOHOYGPCMZDC
|
6.6 | IC50 | 2 | — | |
MVXOBHJTQLGDOM
|
6.6 | IC50 | 4 | — | |
AYKBOWZOVIGZTC
|
6.5 | IC50 | 3 | — | |
JHIZAIITMHMHIB
|
6.5 | IC50 | 3 | — | |
LFYHYFAZHQOTIH
|
6.5 | IC50 | 3 | — | |
GCTSHJXOIFKTDC
|
6.5 | IC50 | 2 | — | |
PYFGVIHNOQRQLL
|
6.5 | IC50 | 3 | — | |
RRBNTBZUGZSZPY
|
6.5 | IC50 | 2 | — | |
YSVJQHXFMCJKHN
|
6.5 | IC50 | 3 | — | |
AHFREZBUCJRIGB
|
6.5 | IC50 | 3 | — | |
ZGJPWRMOZWWOSI
|
6.5 | IC50 | 3 | — | |
LBTWZXYXMWBYRV
|
6.5 | IC50 | 2 | — | |
JJKYNQHCVCQSIQ
|
6.5 | IC50 | 2 | — | |
GAQQHLRNBQSZHG
|
6.4 | IC50 | 2 | — | |
IQJIEOZLFQRBHD
|
6.4 | IC50 | 3 | — | |
FRCDQCXLBBSGID
|
6.4 | IC50 | 2 | — | |
RBVJNRCZCPPSFR
|
6.4 | IC50 | 3 | — | |
GGUMXPSCDHUNCC
|
6.4 | IC50 | 3 | — | |
HFNZVULXLWCEFN
|
6.3 | IC50 | 3 | — | |
NLYHECMWOMFTEC
|
6.3 | IC50 | 4 | — | |
RDTQVSHPKHPGRR
|
6.3 | IC50 | 2 | — | |
RMELHUQGBBCNHR
|
6.3 | IC50 | 3 | — | |
VMZAMOYHCUWUAW
|
6.3 | IC50 | 2 | — | |
FZJYLOPMTVKGCB
|
6.2 | IC50 | 2 | — | |
KQYBGLQZIUDBIA
|
6.2 | IC50 | 3 | — | |
GPQJFLRSELKULV
|
6.2 | IC50 | 3 | — |