Target Details
UniProt ACP28335
Gene SymbolHTR2C
Protein Name5-hydroxytryptamine receptor 2C
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 2,557
  • Clinical molecules 61
  • Avg pChEMBL 7.26
Top Co-occurrence Targets
Active Molecules (2,557)
InChIKey pChEMBL Type Targets Clinical
GIKPTWKWYXCBEC 10.7 Ki 3
CFIKNQMQZHORRL 10.5 Ki 2
AZGOVLGMSGAOMP 10.4 Ki 3
ZETKICHIMHKHIO 10.1 Ki 2
MUTLEZDXAUDNMD 10.0 Ki 2
SJJZDXFWNBMUPH 9.9 IC50 2
OPCCXGXGEHABFP 9.8 Kd 17
IYCYBBKOARJBGP 9.7 Ki 2
JEBVCVUBEGERDC 9.7 Ki 3
XAEAYQWCVVRSFL 9.7 Ki 2
BSOLCASXROXPRZ 9.7 Ki 9
RYUVUCIHNWDAGY 9.6 Ki 2
GIWWCFJNCWGLAP 9.6 Ki 3
GSPGZYOBUGBKTB 9.6 Ki 2
FKRREVSELFOLDT 9.5 Ki 3
SZWVUASESVZMCY 9.5 Ki 3
YIGHLUNEZLKMPP 9.5 Ki 2
CBYNVWMUBJNWTI 9.5 Ki 2
GJVPUHJMJVJTOE 9.5 Ki 3
NNRMMTGPLBXKIO 9.5 Ki 3
UQAOMNGDHNIWSW 9.5 Ki 2
SVWXMPDHBHJCLK 9.5 Ki 2
SNRJCGGWLRAQGG 9.4 Ki 2
HGGAPXYKOUETOQ 9.4 Ki 2
BVTYPXOYRUAGFD 9.4 Ki 2
CNYCTYLQOYVVNS 9.4 Ki 4
FTJNHAUXWUOACE 9.4 Ki 3
GJVPUHJMJVJTOE 9.4 Ki 3
QFPXEFZKXYSMPH 9.4 Ki 3
SYDFROBMNFAPBV 9.4 Ki 3
WGFMMFHWGQNJEB 9.4 Ki 3
ZZJYIKPMDIWRSN 9.4 Ki 11
MOBOBORGXXJTLS 9.4 Ki 2
ITBDDOYXQTUJHV 9.4 Ki 4
VQEPYEWGKYAOBG 9.3 Ki 2
VPLDGFXTWUCSIG 9.3 Ki 2
PTFCJDUGZIFGRV 9.3 Ki 2
XQDRWCFJBHLWPR 9.3 Ki 8 Yes
AGPTZOURDHRCAS 9.3 Ki 3
KLAHZRONIHBPPB 9.3 Ki 3
RCKUMMWWCMFKRU 9.3 Ki 3
SXBHICYVWPUTOA 9.3 Ki 3
VBVQALLSEUJYOK 9.3 Ki 3
HNRQZIBKSIMGFC 9.3 Ki 2
VHNFRNTVRLAIBR 9.3 IC50 2
VOGDBAZLGHXJBS 9.3 Ki 3
KQRKHYJZSCKWTF 9.2 Ki 2
XRYLGRGAWQSVQW 9.2 Ki 7
DXXXGJIMFKZHRL 9.2 Ki 5
NWDWRYLAZDYIBK 9.2 Ki 3
2D structure