Target Details
UniProt ACP28223
Gene SymbolHTR2A
Protein Name5-hydroxytryptamine receptor 2A
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 4,720
  • Clinical molecules 66
  • Avg pChEMBL 7.56
Top Co-occurrence Targets
Active Molecules (4,720)
InChIKey pChEMBL Type Targets Clinical
HKELRUMBUSUQHV 9.2 Ki 3
HSSOKZQOZIZVNW 9.2 Ki 2
KAAGJIUPRMXDTG 9.2 Ki 3
KWNJJPLLFRQMRI 9.2 Ki 4
LMPJCXOOACXKHV 9.2 Ki 4
LWEJANPMNUMGMB 9.2 Ki 4
NLQDMIUSBFMXRV 9.2 Ki 4
RRTOYKUQJIMLKS 9.2 Ki 2
SOJUVNZTSQSTPY 9.2 Ki 2
UFNOVPGGHCFBLJ 9.2 Ki 3
ULFZVKKURLBXLU 9.2 Ki 3
VJYQMOSNEVQNJR 9.2 Ki 3
VPEJCRRRTLASBZ 9.2 Ki 2
ZKEUFSFPGJUPGF 9.2 IC50 2
ZWZGWXZGAUJLHN 9.2 Ki 3
CERBCWPHTRCSMG 9.2 Ki 2
GKDBTHSYQZTDAJ 9.2 IC50 13
QQARGOMNAXCOKN 9.2 Ki 2
SMLCPNKOWBEDFF 9.2 Ki 3
MZBZALUTJALVLT 9.2 Ki 4
NCGLCBITYFKBDE 9.2 IC50 2
OLSNXEOXWIBURX 9.2 IC50 2
PJUZUZVUPDFYFD 9.2 IC50 2
RNYHWTXZYQHTBA 9.2 Ki 2
SYDFROBMNFAPBV 9.2 Ki 3
YMVIRCYNRMVMJQ 9.2 IC50 2
CESJQKNECLKVHF 9.2 Ki 3
CJGYRCCRCWSGRT 9.2 Ki 2
FQBBSOFRGNNFDV 9.2 Ki 3
KXAOPEMSBPZNPQ 9.2 Ki 5
KXEZUXJCVHYFBX 9.2 Ki 3
KYIGOCCCBXRHNJ 9.2 IC50 43
MOBOBORGXXJTLS 9.2 Ki 2
UHSHPGFICACACL 9.2 Ki 4
UZLABACTMPVNHT 9.2 Ki 2
WGCMIWIMQFOYOI 9.2 Ki 3
XEJNCXFNKSUHHY 9.2 Ki 5
FDLRDRBESBJAAV 9.2 Ki 3
KZTBTZPPFWBWTI 9.2 Ki 2
NPJOTTITGQHAPT 9.2 Ki 2
ORARZDXQXHHARR 9.2 Ki 4
ADVRGUCYVUJICT 9.2 Ki 2
GFQPGTMHAHWZHS 9.2 Ki 4
PNRXQZLTVQCRMF 9.2 Ki 3
VQEPYEWGKYAOBG 9.2 Ki 2
BTWSXWRYWXPDBK 9.2 Ki 2
BTWSXWRYWXPDBK 9.2 Ki 2
GZIHLYBPKBXRSW 9.2 Ki 3
NBMCMVKIOBKUGI 9.2 Ki 3
NTNOFWTZPPUTET 9.2 Ki 2
2D structure