Target Details
UniProt ACP28223
Gene SymbolHTR2A
Protein Name5-hydroxytryptamine receptor 2A
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 4,720
  • Clinical molecules 66
  • Avg pChEMBL 7.56
Top Co-occurrence Targets
Active Molecules (4,720)
InChIKey pChEMBL Type Targets Clinical
TWLLJXZOTXAUCG 9.7 Ki 2
BKJQLMPFZFHIMJ 9.7 Ki 3
NRFJXDLMBKNOHP 9.7 Ki 3
QMVRSBUQOIXYIF 9.7 Ki 2
WWYFNHKUOJLBQO 9.7 Ki 2
BORKNTMJLZXUGM 9.7 Ki 3
CJYNZADQWSGLAG 9.7 Ki 2
LEDYBEGWCAWDCY 9.7 Ki 3
QBSWOTCICIQFIN 9.7 Ki 2
VUIPRPLRHSZXDX 9.7 Ki 3
XMXHEBAFVSFQEX 9.7 Ki 17
HMETZCGOVJHJBJ 9.7 Ki 4
RRPGXEGJQQVUTA 9.7 IC50 2
KSEHPHIHVMQGKQ 9.7 Ki 2
QAIRIJOUTULBTI 9.7 Ki 2
VARRTAZUISVFHX 9.7 Ki 2
AAELEHAFAYIZRH 9.6 Ki 5
DAUSNPVLXKKGNQ 9.6 Ki 3
DAUSNPVLXKKGNQ 9.6 Ki 3
OLRVQVYEXPCJPP 9.6 Ki 3
QYNVBLKTSBFRTP 9.6 Ki 3
DSNSWHGDQTZOTM 9.6 Ki 4
VZKXQURASTWIAW 9.6 Ki 4
FHTQWEHAVYFMHP 9.6 Ki 4
MIDQPNSXCMMZSS 9.6 Ki 4
QGVGRVIBOJVENZ 9.6 Ki 4
WIJVLCXKSPDTFW 9.6 Ki 4
BNPYZAAZLNWAPS 9.6 Ki 3
JQDBXOHJKFSLAO 9.6 Ki 2
JQDBXOHJKFSLAO 9.6 Ki 2
MUUOYNXCYHNXFB 9.6 IC50 2
XRBRXMZIBLYNRX 9.6 Ki 2
HCKNVBJJLXPUBM 9.6 IC50 2
SOMWRASUKKDBSH 9.6 Ki 4
VVQHIMSSYISPOD 9.6 Ki 2
YHEZQOSUVDWMEX 9.6 Ki 3
ZNLRXSLTHYHDNL 9.6 IC50 2
DBRVEHQLZZEVFX 9.6 Ki 5
CGVZEZGEEUBAEK 9.6 Ki 3
GGJYDEZYCACGIQ 9.6 IC50 2
PNDDOSJAKNIYIV 9.6 Ki 4
SWKDCCLYHAYMLD 9.6 Ki 2
XCZLLQDTFNFIDZ 9.6 Ki 2
ZCAJFFDMFGAKNN 9.6 Ki 2
DXQITHRANRYTGO 9.5 Ki 2
LCZMXKRXXCYHBB 9.5 Ki 5
RGWGDYMUCXDODX 9.5 Ki 4
CJCHZXCLUYLXJM 9.5 Ki 3
GHUSLXGCIAVXOA 9.5 Ki 2
GYVLPHYAFKCJIG 9.5 Ki 4
2D structure