Target Details
UniProt ACP28223
Gene SymbolHTR2A
Protein Name5-hydroxytryptamine receptor 2A
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00001 (7tm_1)
Summary
  • Multi-target molecules 4,720
  • Clinical molecules 66
  • Avg pChEMBL 7.56
Top Co-occurrence Targets
Active Molecules (4,720)
InChIKey pChEMBL Type Targets Clinical
YFIBOKLKHXZNEU 8.8 Ki 3
ZESRJSPZRDMNHY 8.8 Ki 5
HNFGNFPOEVJRAY 8.8 Ki 3
NFZVIQPFHKWWOS 8.8 Ki 2
TYMYSUSJLROMAC 8.8 Ki 2
YOQMDXGCJSLBBS 8.8 Ki 4
AVPWRHUUQUMMJK 8.8 Ki 4
BQDBKDMTIJBJLA 8.8 Ki 5
FQRIRCXYLMTNDU 8.8 Ki 4
GIALFYFYXHAZSV 8.8 Ki 3
HDOZVRUNCMBHFH 8.8 Ki 26 Yes
HLGKXVMBSLHNKH 8.8 Ki 4
MWUUTPCYIHCLOP 8.8 Ki 2
NVXLFLRKJMMSPG 8.8 Ki 2
OHIHGZWNDVVIBE 8.8 Ki 2
PHOFLKKBYFRIGR 8.8 Ki 3
RCWSDRYOQJIECB 8.8 Ki 4
RFRAMVDLVRFQPK 8.8 Ki 3
SLFGIOIONGJGRT 8.8 Ki 12
TULOEXKDPBREQC 8.8 Ki 3
UXHXPQAQESSLQQ 8.8 Ki 3
VUFNCLXJAJQINV 8.8 IC50 2
WBENNDOANVTGAH 8.8 Ki 2
YLZMZAMSWUDWOE 8.8 IC50 2
YQCPDRVHUVCVIN 8.8 Ki 2
HMILUIFVMYFSEQ 8.8 Ki 2
AYFAGRAOJPSHSH 8.8 Ki 19
BGMZUEKZENQUJY 8.8 Ki 3
BSOLCASXROXPRZ 8.8 Ki 9
BTICABKVLJBOCS 8.8 Ki 2
FFZUWXZVFRDGLT 8.8 Ki 3
IAJGHVPYWZBQQT 8.8 Ki 3
LCGBVEYGRZPQEM 8.8 Ki 3
LQYNONCEAYAGNN 8.8 Ki 5
MYUNZXXMZICHEZ 8.8 Ki 3
NJJMNKOVGYIOBG 8.8 Ki 4
ODNIEBFFNONVCK 8.8 Ki 3
PQWQIDDLFHUBOY 8.8 Ki 3
RCFZNHOLJFFNFW 8.8 Ki 2
SXEPPXITHUOXQU 8.8 IC50 2
USTBGZUJKCBYAR 8.8 Ki 2
UTVCJNNRVXMBSF 8.8 Ki 3
VLXOYOJCCCNIRP 8.8 Ki 3
XBWNTYFNUFPCHL 8.8 Ki 3
APOMSSAGEAOUGO 8.8 Ki 5
IYRFHZMJBBCIFA 8.8 Ki 4
KLCDGLISRKLICJ 8.8 Ki 2
NFPWRHWDAIDXGI 8.8 IC50 2
VWBQZTFOSGQJQU 8.8 Ki 3
VZHORDSFYCKLRO 8.8 Ki 4
2D structure