Target Details
| UniProt AC | P27958 |
|---|---|
| Gene Symbol | N/A |
| Protein Name | Genome polyprotein |
| Organism | Hepatitis C virus genotype 1a (isolate H77) |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF07652 (Flavi_DEAD) PF01543 (HCV_capsid) PF01542 (HCV_core) PF01539 (HCV_env) PF01560 (HCV_NS1) PF01538 (HCV_NS2) PF01006 (HCV_NS4a) PF01001 (HCV_NS4b) PF01506 (HCV_NS5a) PF08300 (HCV_NS5a_1a) PF08301 (HCV_NS5a_1b) PF12941 (HCV_NS5a_C) PF22027 (NS3_helicase_C) PF02907 (Peptidase_S29) PF00998 (RdRP_3) |
Summary
- Multi-target molecules 315
- Clinical molecules 0
- Avg pChEMBL 7.76
Active Molecules (315)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DULIAOKIHPSTBZ
|
10.0 | Ki | 3 | — | |
JDMPXCANLSMISU
|
10.0 | Ki | 3 | — | |
SMGNMBKPAWFKGH
|
10.0 | Ki | 3 | — | |
VOMDFEZIJGRATE
|
10.0 | Ki | 3 | — | |
FEBJFCFXFXZCLS
|
9.7 | Ki | 3 | — | |
YCYCBCSJYGZXLL
|
9.6 | IC50 | 3 | — | |
CFMGTKRBVVZVBF
|
9.3 | IC50 | 4 | — | |
PFORZALCOLIZSP
|
9.3 | Ki | 3 | — | |
IQKDRVURUHCSRA
|
9.2 | IC50 | 4 | — | |
KRVBPGRPHRGDBE
|
9.2 | IC50 | 4 | — | |
XXXWQTLZEUCJPJ
|
9.1 | IC50 | 3 | — | |
AGVSXXLDLPSANO
|
9.1 | Ki | 3 | — | |
LOYIQGBTNJFCIL
|
9.1 | IC50 | 4 | — | |
IHPQWLFEUQBMFZ
|
9.1 | IC50 | 4 | — | |
KNQHCQDUNTWSPH
|
9.1 | IC50 | 4 | — | |
NWFWLEAQCNXLAB
|
9.0 | IC50 | 4 | — | |
NWNRFJLJFPUJSR
|
9.0 | IC50 | 4 | — | |
OIHIJLNMNDCCIY
|
9.0 | IC50 | 4 | — | |
RZCUJQGMLLHXFG
|
9.0 | IC50 | 4 | — | |
WFXFHGMKTRFARM
|
9.0 | IC50 | 4 | — | |
YHJYFWRWHAHNQA
|
9.0 | IC50 | 4 | — | |
XLLUDKOBZFHIKN
|
8.9 | IC50 | 4 | — | |
XFYOTNPRWVBFPP
|
8.9 | IC50 | 4 | — | |
MOJHZLPPVIASCY
|
8.8 | IC50 | 4 | — | |
NLCBQIDOYIYGHS
|
8.8 | IC50 | 4 | — | |
VXDRIGYTIFAUHJ
|
8.8 | IC50 | 4 | — | |
YNYFVDOGUKBANE
|
8.8 | IC50 | 4 | — | |
AMWXBFDFQCGDLH
|
8.8 | IC50 | 4 | — | |
GNMJIFOVLJTJGQ
|
8.8 | IC50 | 4 | — | |
LRSKPOKZPAQFRH
|
8.8 | IC50 | 4 | — | |
VCYVRAYCTRSTDK
|
8.8 | IC50 | 4 | — | |
NMFUHYFGDLXDAP
|
8.8 | IC50 | 3 | — | |
WXGVQUUZCZFRQM
|
8.8 | IC50 | 4 | — | |
CYWKRSLNXIMRQO
|
8.7 | IC50 | 4 | — | |
VMEBZEMJNJSXPG
|
8.7 | IC50 | 3 | — | |
DBKVPPPOBUUZEG
|
8.7 | IC50 | 4 | — | |
GZPOQDPGYRPDKE
|
8.7 | IC50 | 4 | — | |
ILEXPDKMDMRQKR
|
8.7 | IC50 | 4 | — | |
OPNNEDOKBVIBDQ
|
8.7 | IC50 | 4 | — | |
RHEVGRYWYIGWAV
|
8.7 | IC50 | 4 | — | |
SXFOFKRRPNGFMD
|
8.7 | IC50 | 3 | — | |
SYHBIJWOUCBHHI
|
8.7 | Ki | 2 | — | |
WFXFHGMKTRFARM
|
8.7 | IC50 | 4 | — | |
XONCCNBWLVICPL
|
8.7 | IC50 | 4 | — | |
XONCCNBWLVICPL
|
8.6 | IC50 | 4 | — | |
XRACUQUEKFCAJG
|
8.6 | IC50 | 3 | — | |
LTXGWCYRWMVHSW
|
8.6 | IC50 | 4 | — | |
CMGPWMKFYBSJKI
|
8.6 | IC50 | 4 | — | |
GGGMJNVXWGTZHR
|
8.6 | IC50 | 4 | — | |
HFIAXUYJXXCQEM
|
8.6 | IC50 | 4 | — |