Target Details
| UniProt AC | P27815 |
|---|---|
| Gene Symbol | PDE4A |
| Protein Name | 3',5'-cyclic-AMP phosphodiesterase 4A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF18100 (PDE4_UCR) PF00233 (PDEase_I) |
Summary
- Multi-target molecules 1,354
- Clinical molecules 3
- Avg pChEMBL 7.5
KEGG Pathways (5)
Active Molecules (1,354)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VKLSPPITZQCVKV
|
8.0 | Ki | 4 | — | |
XWLNXPBGFLZPDR
|
8.0 | IC50 | 4 | — | |
ZGBRFHWLOXQCMR
|
8.0 | IC50 | 4 | — | |
DSCLXJMGAQHPPO
|
8.0 | IC50 | 4 | — | |
IEIYCAUGLWVZTR
|
8.0 | IC50 | 4 | — | |
OPBIZTGCIJZSGG
|
8.0 | IC50 | 4 | — | |
YOCIPGYKDZCTFU
|
8.0 | IC50 | 4 | — | |
AIIYPFJZLRJGEL
|
8.0 | IC50 | 3 | — | |
PHIVEUQACADDGU
|
8.0 | IC50 | 4 | — | |
YXSFWZAMZUKSOK
|
8.0 | IC50 | 4 | — | |
VSOPHYORBVNBMU
|
7.9 | IC50 | 4 | — | |
DNQXAUUOWTUBLN
|
7.9 | IC50 | 4 | — | |
WKUVVAFTNFZIQC
|
7.9 | IC50 | 4 | — | |
CICKNGAWODWCEX
|
7.9 | IC50 | 4 | — | |
GUBLWTBQTNDNFO
|
7.9 | IC50 | 4 | — | |
JREKQRFHYGBRFX
|
7.9 | IC50 | 4 | — | |
KTHGYZDOEYNTKY
|
7.9 | IC50 | 4 | — | |
PJUUZPXCNUJBPS
|
7.9 | IC50 | 3 | — | |
YEUSBANVZAFKBV
|
7.9 | IC50 | 4 | — | |
ZFSNOVAGVJZIOT
|
7.9 | IC50 | 4 | — | |
ZJWBPIDGEVCEHP
|
7.9 | IC50 | 4 | — | |
XPVCYAAXXRUYDT
|
7.9 | IC50 | 3 | — | |
ABVXSVHDNRZRGD
|
7.9 | IC50 | 4 | — | |
HYFGDONYQPRTJU
|
7.9 | IC50 | 4 | — | |
ITLJCTJVLVIKBE
|
7.9 | IC50 | 4 | — | |
KPHBKZYONHHTQY
|
7.9 | IC50 | 4 | — | |
KYKHXPMUZAMXTE
|
7.9 | Kd | 4 | — | |
MLWIHJQIPLXJNU
|
7.9 | IC50 | 4 | — | |
NWSUWPQBMXRCDD
|
7.9 | IC50 | 4 | — | |
PAISFAPTLJTHAX
|
7.9 | IC50 | 4 | — | |
SCHCQOLPISHKOS
|
7.9 | IC50 | 4 | — | |
SEWBUIWTHYNBNC
|
7.9 | IC50 | 4 | — | |
SEWBUIWTHYNBNC
|
7.9 | IC50 | 4 | — | |
TVGJNNOUNWXDCO
|
7.9 | IC50 | 4 | — | |
DDWDVJRARZITDU
|
7.9 | IC50 | 4 | — | |
FMDFPSUREAEZOZ
|
7.9 | IC50 | 4 | — | |
JLQBUJOOXOEDTB
|
7.9 | IC50 | 4 | — | |
JSVIBRYXRHAZKZ
|
7.9 | IC50 | 4 | — | |
POOZXNMBPQYVQV
|
7.9 | IC50 | 6 | — | |
XUMPDYRHXWOEDT
|
7.9 | IC50 | 3 | — | |
DPHDSIQHVGSITN
|
7.8 | IC50 | 4 | — | |
PHOOWFUDCZCEGK
|
7.8 | IC50 | 4 | — | |
VKYWOZPNAQYXPJ
|
7.8 | IC50 | 4 | — | |
YFSKDXWVNPXSTG
|
7.8 | IC50 | 4 | — | |
FZWZAVQJUANPKQ
|
7.8 | IC50 | 4 | — | |
GRFHQTKEAOBDST
|
7.8 | IC50 | 3 | — | |
SEAKUVPPGRMOIJ
|
7.8 | IC50 | 4 | — | |
SRRULVNTICTTGE
|
7.8 | IC50 | 4 | — | |
WBVHJGBFCGWOMH
|
7.8 | IC50 | 4 | — | |
COQGBMKNVJUVAB
|
7.8 | IC50 | 4 | — |