Target Details
| UniProt AC | P27815 |
|---|---|
| Gene Symbol | PDE4A |
| Protein Name | 3',5'-cyclic-AMP phosphodiesterase 4A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF18100 (PDE4_UCR) PF00233 (PDEase_I) |
Summary
- Multi-target molecules 1,354
- Clinical molecules 3
- Avg pChEMBL 7.5
KEGG Pathways (5)
Active Molecules (1,354)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NJCCFDZQRIVPQK
|
8.2 | IC50 | 4 | — | |
UNFSVUGGDWHOPR
|
8.2 | IC50 | 4 | — | |
YJPWCVBJBWSWSU
|
8.2 | IC50 | 3 | — | |
IOOPRDTXOWLHHO
|
8.2 | IC50 | 4 | — | |
VNMFECKPJDGTEJ
|
8.2 | IC50 | 4 | — | |
XBELIXRJJBCGOR
|
8.2 | IC50 | 4 | — | |
CVDXFPBVOIERBH
|
8.2 | IC50 | 4 | — | |
FGLJIZXIRLUUJT
|
8.2 | IC50 | 4 | — | |
ZLYJLUCSZKDSRN
|
8.2 | IC50 | 4 | — | |
OBZABHIWBRSMRC
|
8.1 | IC50 | 4 | — | |
UGUNGNPFDJUJNI
|
8.1 | IC50 | 4 | — | |
VIWWIIFOLLGWED
|
8.1 | IC50 | 4 | — | |
TVPGHEMRNSSWKT
|
8.1 | IC50 | 4 | — | |
DCYZEFXLJGEMAA
|
8.1 | IC50 | 4 | — | |
JBMNQTIIWJVUPM
|
8.1 | IC50 | 4 | — | |
KMAXAJFXSIHYPS
|
8.1 | IC50 | 4 | — | |
OTTVHKKGMZTQQL
|
8.1 | IC50 | 4 | — | |
QSFOYCZPHALXMC
|
8.1 | IC50 | 4 | — | |
RKHLITOQHDGEOE
|
8.1 | IC50 | 4 | — | |
SPNSPIATZGICGL
|
8.1 | IC50 | 4 | — | |
SPNSPIATZGICGL
|
8.1 | IC50 | 4 | — | |
UHXRJGVYNNLRMG
|
8.1 | IC50 | 4 | — | |
UQHGEVKJBWBSGG
|
8.1 | IC50 | 2 | — | |
WXBVDTBUOVXWKY
|
8.1 | IC50 | 6 | — | |
DXYODODSZIQFFT
|
8.1 | IC50 | 2 | — | |
MYBHWAVLLSQXOM
|
8.1 | IC50 | 4 | — | |
SEPBFTDLZPYNPJ
|
8.1 | IC50 | 4 | — | |
PPRGGHMXTMLYEU
|
8.1 | IC50 | 3 | — | |
VNKRGOHAYGVCDA
|
8.1 | IC50 | 2 | — | |
VSLZRLVOASPJGZ
|
8.1 | IC50 | 4 | — | |
WDIRFWGTTLSFDP
|
8.1 | IC50 | 4 | — | |
AKNVUBOYOIBCCN
|
8.1 | IC50 | 4 | — | |
DIQPQAKBMJIODR
|
8.1 | IC50 | 3 | — | |
KLQIHSRSOJJAMH
|
8.1 | IC50 | 4 | — | |
MSGATJYNCMZCIQ
|
8.0 | IC50 | 4 | — | |
DLSHWTXXGZXIQU
|
8.0 | IC50 | 4 | — | |
BZYKZBJOZPFGGO
|
8.0 | IC50 | 4 | — | |
AKOYRAGTUVPQDO
|
8.0 | IC50 | 4 | — | |
BTKBSAYJTCJZMD
|
8.0 | IC50 | 4 | — | |
CESDTWPSVRIIIH
|
8.0 | IC50 | 4 | — | |
GFALNLVQJILPHP
|
8.0 | IC50 | 4 | — | |
HMKJSFGZWJJYNY
|
8.0 | IC50 | 4 | — | |
ILTIMOPOVHETED
|
8.0 | IC50 | 4 | — | |
LSQPGJAKGOVZCJ
|
8.0 | IC50 | 4 | — | |
MUZUXIDORXRNNG
|
8.0 | IC50 | 4 | — | |
NMGSQEBMRHQDOG
|
8.0 | IC50 | 4 | — | |
OLDNCOKMXZXSQN
|
8.0 | IC50 | 4 | — | |
OVLZKANHBRXYRB
|
8.0 | IC50 | 4 | — | |
QMLOEDCWTHEZJY
|
8.0 | IC50 | 5 | — | |
TVHKGMWQQAHKTC
|
8.0 | IC50 | 4 | — |