Target Details
| UniProt AC | P27815 |
|---|---|
| Gene Symbol | PDE4A |
| Protein Name | 3',5'-cyclic-AMP phosphodiesterase 4A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF18100 (PDE4_UCR) PF00233 (PDEase_I) |
Summary
- Multi-target molecules 1,354
- Clinical molecules 3
- Avg pChEMBL 7.5
KEGG Pathways (5)
Active Molecules (1,354)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YWTCDMZVTLNYLN
|
8.3 | IC50 | 3 | — | |
JPPKVWKIBHEEGN
|
8.3 | IC50 | 3 | — | |
YYGZHVJDHMMABU
|
8.3 | IC50 | 4 | — | |
LAJDTVWSQMUYRE
|
8.3 | IC50 | 4 | — | |
BGOQUVGOCSMNKK
|
8.3 | IC50 | 3 | — | |
CWRSELIFKXREAE
|
8.3 | IC50 | 4 | — | |
FCCDJWUNWSSEGE
|
8.3 | IC50 | 4 | — | |
GLYPDLWNQYDRTQ
|
8.3 | IC50 | 4 | — | |
HLSOZRYDNZEYOT
|
8.3 | IC50 | 6 | — | |
KKINNZHENOWAFZ
|
8.3 | IC50 | 4 | — | |
OMBWXFIZADXIQW
|
8.3 | IC50 | 4 | — | |
ONVLPDRKPJLPDE
|
8.3 | IC50 | 4 | — | |
OZUNUTXZGBJXGF
|
8.3 | IC50 | 4 | — | |
UGEXFJGYLFXPNT
|
8.3 | IC50 | 3 | — | |
WOWBDVWWSBMFRA
|
8.3 | IC50 | 3 | — | |
IVSBLXFZMFGIAK
|
8.3 | IC50 | 4 | — | |
BKBBEYMNJXXDAQ
|
8.3 | IC50 | 2 | — | |
RQKJDWFZSBVQSW
|
8.3 | IC50 | 4 | — | |
BNUQRBLZFCEYSG
|
8.3 | IC50 | 3 | — | |
FKOVNYLAGQLEDI
|
8.3 | IC50 | 4 | — | |
RESYBSJMKXZFCE
|
8.3 | IC50 | 4 | — | |
VJEYWPJLEFUOTH
|
8.3 | IC50 | 4 | — | |
CDQAOTLTJJQBOP
|
8.2 | IC50 | 4 | — | |
CTIDVXFZTVGPIU
|
8.2 | IC50 | 4 | — | |
FYZBEANPACBLTJ
|
8.2 | IC50 | 4 | — | |
LZXLYACBALMEJP
|
8.2 | IC50 | 4 | — | |
GKHODUKSOBLBHU
|
8.2 | IC50 | 4 | — | |
CICKNGAWODWCEX
|
8.2 | IC50 | 4 | — | |
CIMWFDZKHUKERW
|
8.2 | IC50 | 4 | — | |
JJWKQXNHYDJXKF
|
8.2 | IC50 | 4 | — | |
NSYYFQMQNAQQGB
|
8.2 | IC50 | 4 | — | |
GWKPSIAHYYAQIR
|
8.2 | IC50 | 4 | — | |
IIYMHHZVTORHCY
|
8.2 | IC50 | 4 | — | |
JASNCWACDBPEJY
|
8.2 | IC50 | 4 | — | |
WUECXCBONAGRSA
|
8.2 | IC50 | 6 | — | |
BJHZUUZWVUANNB
|
8.2 | IC50 | 4 | — | |
KUWSQRWJCOFAGZ
|
8.2 | IC50 | 3 | — | |
VGRIHMHLBGLHHB
|
8.2 | IC50 | 4 | — | |
XHHHLXUOGDNSNR
|
8.2 | IC50 | 4 | — | |
AGNPWVFAZVESPJ
|
8.2 | IC50 | 4 | — | |
KBHCNHZXGQOFAJ
|
8.2 | IC50 | 4 | — | |
KSDNSDVILMJIKK
|
8.2 | IC50 | 6 | — | |
OVLZKANHBRXYRB
|
8.2 | IC50 | 4 | — | |
SHWIKYNKCMPTHS
|
8.2 | IC50 | 4 | — | |
YBCWUCNBLGPSSQ
|
8.2 | IC50 | 6 | — | |
QXMYNGZVAQOGPB
|
8.2 | IC50 | 4 | — | |
VERPTCRKINCACJ
|
8.2 | IC50 | 3 | — | |
VUKLRTNDLAMXGZ
|
8.2 | IC50 | 2 | — | |
ATETVUDHVLJVIY
|
8.2 | IC50 | 4 | — | |
DZAUSKKPHXFGNN
|
8.2 | IC50 | 6 | — |