Target Details
| UniProt AC | P27815 |
|---|---|
| Gene Symbol | PDE4A |
| Protein Name | 3',5'-cyclic-AMP phosphodiesterase 4A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF18100 (PDE4_UCR) PF00233 (PDEase_I) |
Summary
- Multi-target molecules 1,354
- Clinical molecules 3
- Avg pChEMBL 7.5
KEGG Pathways (5)
Active Molecules (1,354)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XRVDXHQYLWXJOB
|
8.6 | IC50 | 4 | — | |
LZQQXWXCJOTIAP
|
8.6 | IC50 | 4 | — | |
LSCITVBMOOTYOS
|
8.6 | IC50 | 3 | — | |
BBTFKAOFCSOZMB
|
8.6 | IC50 | 5 | — | |
HOKIHKLKOZWCRY
|
8.6 | IC50 | 4 | — | |
LQSTXUKGXUCNPL
|
8.6 | IC50 | 4 | — | |
QSRJUMJDYNOQBS
|
8.5 | IC50 | 4 | — | |
FCIZPPJLBOLIRV
|
8.5 | IC50 | 5 | — | |
GVLQLBNMZUZFAS
|
8.5 | Ki | 4 | — | |
IXQHNBONEVULTL
|
8.5 | IC50 | 4 | — | |
JERXUPDBWDWFCF
|
8.5 | IC50 | 4 | — | |
OHSOWGXJKVARKN
|
8.5 | IC50 | 4 | — | |
XVFXPIPTQRSUTA
|
8.5 | IC50 | 4 | — | |
NMGSQEBMRHQDOG
|
8.5 | IC50 | 4 | — | |
RLKUDKVBRRKFID
|
8.5 | IC50 | 4 | — | |
XXAZCHDKOQBDMG
|
8.5 | IC50 | 4 | — | |
DZFTVPIHZOONHV
|
8.5 | IC50 | 4 | — | |
IXFIUOCIFSTVBK
|
8.5 | IC50 | 4 | — | |
OBKIBWWNAYXLEM
|
8.5 | IC50 | 4 | — | |
QWJORUKKCABZPO
|
8.5 | IC50 | 4 | — | |
ZOPYTZDTLDQKKZ
|
8.5 | IC50 | 4 | — | |
CPGLQQFUYMJRLF
|
8.4 | IC50 | 4 | — | |
IHICZLPILSZEIR
|
8.4 | IC50 | 4 | — | |
OADRFAYKJSEHSL
|
8.4 | IC50 | 4 | — | |
IJGCWHSMOTWWLO
|
8.4 | IC50 | 4 | — | |
OPCOERKUHFQVKE
|
8.4 | IC50 | 4 | — | |
ACCZCVFKTVIVJV
|
8.4 | IC50 | 4 | — | |
COSLZNSLGCSJBY
|
8.4 | IC50 | 4 | — | |
CZFXKMHZLIYHEV
|
8.4 | IC50 | 6 | — | |
FYEUTUDJCAUZQG
|
8.4 | IC50 | 4 | — | |
OZUHZRXDNSSAMN
|
8.4 | IC50 | 6 | — | |
PMDTUKRFGFOQKR
|
8.4 | IC50 | 4 | — | |
XARBLJKEGWJAGR
|
8.4 | IC50 | 4 | — | |
XIYCOQBLMCIMFX
|
8.4 | IC50 | 4 | — | |
PPRHBMORJBZDIK
|
8.4 | IC50 | 4 | — | |
RZJRUSAPSQVWEL
|
8.4 | IC50 | 4 | — | |
UXXSCNVCFOZAFY
|
8.4 | IC50 | 4 | — | |
IQKXFSXPCZEULC
|
8.4 | IC50 | 6 | — | |
MBBSPQBGJJWYLF
|
8.4 | IC50 | 4 | — | |
UTUUPXBCDMQYRR
|
8.4 | IC50 | 4 | — | |
CEIVKBVSJHEXIU
|
8.4 | IC50 | 2 | — | |
CNAIHJWGQFJIKX
|
8.3 | IC50 | 4 | — | |
IKADFHCDTYOPKD
|
8.3 | IC50 | 3 | — | |
AEVXMUCLERMJMB
|
8.3 | IC50 | 4 | — | |
DDVHCGNQPCSRQB
|
8.3 | IC50 | 3 | — | |
DDVHCGNQPCSRQB
|
8.3 | IC50 | 4 | — | |
DOKUUHZWXPIFPB
|
8.3 | IC50 | 4 | — | |
IMOBPVDSTURWHO
|
8.3 | IC50 | 4 | — | |
NUUIJDOADURGSD
|
8.3 | IC50 | 4 | — | |
VRUGXMNNKXUAGT
|
8.3 | IC50 | 4 | — |