Target Details
| UniProt AC | P27815 |
|---|---|
| Gene Symbol | PDE4A |
| Protein Name | 3',5'-cyclic-AMP phosphodiesterase 4A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF18100 (PDE4_UCR) PF00233 (PDEase_I) |
Summary
- Multi-target molecules 1,354
- Clinical molecules 3
- Avg pChEMBL 7.5
KEGG Pathways (5)
Active Molecules (1,354)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VPDYRGHPOFWFHI
|
8.8 | IC50 | 4 | — | |
ZJXFGGIJHFLWBE
|
8.8 | IC50 | 4 | — | |
ALGYAXVEWGTXDA
|
8.8 | IC50 | 6 | — | |
BVJRFNKHFQRJTE
|
8.8 | IC50 | 4 | — | |
CUYPGPQSXWUTLO
|
8.8 | IC50 | 4 | — | |
FNRUBUFCNWKZEI
|
8.8 | IC50 | 4 | — | |
IURSWTQMXOIIAU
|
8.8 | IC50 | 4 | — | |
SFPJVJIEXHMQRQ
|
8.8 | IC50 | 4 | — | |
VKQDIKWPKDHRJH
|
8.8 | IC50 | 4 | — | |
ANSXOWFFAFVDLN
|
8.8 | IC50 | 5 | — | |
HGDWTVWVCTUICT
|
8.8 | IC50 | 4 | — | |
VSUBBIZTQLTMFR
|
8.8 | IC50 | 4 | — | |
XONFIBGUKUGPPG
|
8.8 | IC50 | 2 | — | |
CABBMCIEXVVIDP
|
8.8 | IC50 | 4 | — | |
MIKQDQMGJFMIAZ
|
8.7 | IC50 | 4 | — | |
AVBSGRYHZMSEHV
|
8.7 | IC50 | 4 | — | |
DJQNRDCGWWXDHA
|
8.7 | IC50 | 4 | — | |
QWJORUKKCABZPO
|
8.7 | IC50 | 4 | — | |
DMPHLSBWKJKTKF
|
8.7 | IC50 | 6 | — | |
HLKIKTJQVCVTJG
|
8.7 | IC50 | 4 | — | |
JFCMFEVPHGDYMS
|
8.7 | IC50 | 4 | — | |
KJUXYSPBVYVNHD
|
8.7 | IC50 | 4 | — | |
OEADYOMRQYOJAO
|
8.7 | IC50 | 4 | — | |
OFNKSFVKBAHXFD
|
8.7 | IC50 | 4 | — | |
QMOPFHQOZKALTC
|
8.7 | IC50 | 4 | — | |
SLPPCYGGTCSDJX
|
8.7 | IC50 | 4 | — | |
SMWGOZGGMUJHKG
|
8.7 | IC50 | 4 | — | |
XQZSDSGBZZUHKR
|
8.7 | IC50 | 2 | — | |
KNVLHSLMSJUURQ
|
8.7 | IC50 | 4 | — | |
MESOMSSOOSHAJX
|
8.7 | IC50 | 4 | — | |
JPXAIORZGBCHIB
|
8.7 | IC50 | 5 | — | |
OMDWIQHGWHOABF
|
8.7 | IC50 | 4 | — | |
QIESARUEQVCDIR
|
8.7 | IC50 | 4 | — | |
QJLFNDIEDQOREP
|
8.7 | IC50 | 2 | — | |
IOHIGXZNGBFEFK
|
8.7 | IC50 | 4 | — | |
NSVZCMUAFBWPEB
|
8.7 | IC50 | 2 | — | |
SGGQQXATQWLMRQ
|
8.7 | IC50 | 4 | — | |
IMNGGIXQGKWJJB
|
8.6 | IC50 | 4 | — | |
MSCBHSUFDKFWDM
|
8.6 | IC50 | 4 | — | |
UHJAPZBOKPPKGD
|
8.6 | IC50 | 4 | — | |
JTGRNMGEASTCHA
|
8.6 | IC50 | 4 | — | |
CCJARLANHMJLNZ
|
8.6 | IC50 | 4 | — | |
GOUBCTXRBKJIBR
|
8.6 | IC50 | 4 | — | |
IPBKYRYKTIGBGW
|
8.6 | IC50 | 4 | — | |
JOFDTTXRCXFIGE
|
8.6 | IC50 | 4 | — | |
LQUSZPOBAPKYNT
|
8.6 | IC50 | 4 | — | |
UARYJPSKTPGAFA
|
8.6 | IC50 | 4 | — | |
WGWKCNVFLGOBOV
|
8.6 | IC50 | 4 | — | |
WPQCJAJFAOGVNJ
|
8.6 | IC50 | 6 | — | |
XZJUOKCCPBELOU
|
8.6 | IC50 | 4 | — |