Target Details
| UniProt AC | P27815 |
|---|---|
| Gene Symbol | PDE4A |
| Protein Name | 3',5'-cyclic-AMP phosphodiesterase 4A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF18100 (PDE4_UCR) PF00233 (PDEase_I) |
Summary
- Multi-target molecules 1,354
- Clinical molecules 3
- Avg pChEMBL 7.5
KEGG Pathways (5)
Active Molecules (1,354)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PSONXFNMYSRABR
|
9.0 | IC50 | 4 | — | |
FWWXAPNNHWGQDC
|
9.0 | IC50 | 4 | — | |
SFPJVJIEXHMQRQ
|
9.0 | IC50 | 4 | — | |
WYBLCAXPFFVGGM
|
9.0 | IC50 | 3 | — | |
BPBDCOLBZYWXHD
|
9.0 | IC50 | 24 | — | |
BQXOJMGGMXNMBL
|
9.0 | IC50 | 4 | — | |
DTJGUSJXWUZZHK
|
9.0 | IC50 | 4 | — | |
FMMIDZWTNQYEIY
|
9.0 | IC50 | 24 | — | |
GILOGFJUMQAJNQ
|
9.0 | IC50 | 4 | — | |
JRNMYGZUERYWCG
|
9.0 | IC50 | 4 | — | |
MAFMSYWPKNBAHN
|
9.0 | IC50 | 4 | — | |
RRRUXBQSQLKHEL
|
9.0 | IC50 | 4 | — | |
SFPJVJIEXHMQRQ
|
9.0 | IC50 | 4 | — | |
WOVJAODSYBKIRW
|
9.0 | IC50 | 3 | — | |
WPKUFAIEVOBXTL
|
9.0 | IC50 | 4 | — | |
WSISMBBKFDPNKB
|
9.0 | IC50 | 4 | — | |
XEPASQPUIOGOCW
|
9.0 | IC50 | 4 | — | |
XSLQVZKRYWJDJT
|
9.0 | IC50 | 4 | — | |
YTFBNFMILWHYAP
|
9.0 | Ki | 4 | — | |
ULFAYKSQGUIMBK
|
9.0 | IC50 | 4 | — | |
KLQWQRAVJHQKOI
|
9.0 | IC50 | 4 | — | |
DSHINXNFGWBHRA
|
9.0 | IC50 | 2 | — | |
FEGNNXIOTUDYKF
|
8.9 | IC50 | 4 | — | |
WDJVSROJMOYUQL
|
8.9 | IC50 | 4 | — | |
HKZQRKPXNBQUSQ
|
8.9 | IC50 | 4 | — | |
LUUUHUYQTLUIDG
|
8.9 | IC50 | 4 | — | |
NMWZIECWRMDJED
|
8.9 | IC50 | 5 | — | |
PYJYVNMGHSGIDT
|
8.9 | IC50 | 3 | — | |
CITPCSPDQMOFRH
|
8.9 | IC50 | 4 | — | |
IQLTUSGIDSAUEK
|
8.9 | IC50 | 4 | — | |
LDQZVKGBHAZGGR
|
8.9 | IC50 | 4 | — | |
SXTQYUHRUIQQLQ
|
8.9 | IC50 | 4 | — | |
VQMKXNJTGPRWCC
|
8.9 | IC50 | 4 | — | |
XYOGUDRZODERFH
|
8.9 | IC50 | 4 | — | |
GZMPVUPEEMXMQY
|
8.9 | IC50 | 4 | — | |
JXQLQPODTZFKHM
|
8.9 | IC50 | 2 | — | |
KRPGYDWKKKFLRX
|
8.9 | IC50 | 2 | — | |
MBNWGNWRHMXPDV
|
8.9 | IC50 | 4 | — | |
MFMSLIOHRZHOEC
|
8.9 | IC50 | 4 | — | |
CQKWNVYRCGKDPM
|
8.9 | IC50 | 4 | — | |
JXBLIAHYVCYDGO
|
8.9 | IC50 | 4 | — | |
LJNMTXMGPGCHPD
|
8.9 | IC50 | 4 | — | |
CQKMCWALCBFISY
|
8.8 | IC50 | 4 | — | |
DMPOYNQUJADULP
|
8.8 | IC50 | 5 | — | |
SDAANIJBPDIBMR
|
8.8 | IC50 | 4 | — | |
WOSZIGPPVCFSFK
|
8.8 | IC50 | 5 | — | |
YYGZHVJDHMMABU
|
8.8 | IC50 | 5 | — | |
DAHVRHNHMXYVKR
|
8.8 | IC50 | 4 | — | |
HKASZTPKFUJMFS
|
8.8 | IC50 | 4 | — | |
HQUIEUONYYTHEW
|
8.8 | IC50 | 5 | — |