Target Details
| UniProt AC | P27815 |
|---|---|
| Gene Symbol | PDE4A |
| Protein Name | 3',5'-cyclic-AMP phosphodiesterase 4A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF18100 (PDE4_UCR) PF00233 (PDEase_I) |
Summary
- Multi-target molecules 1,354
- Clinical molecules 3
- Avg pChEMBL 7.5
KEGG Pathways (5)
Active Molecules (1,354)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MESVEPTYRCXMJY
|
9.3 | IC50 | 4 | — | |
MESVEPTYRCXMJY
|
9.3 | IC50 | 4 | — | |
VUOPSDKSUZFGMP
|
9.3 | IC50 | 4 | — | |
WLXXHGAJJHJBAL
|
9.3 | IC50 | 4 | — | |
YKYDPWLKXOYPEP
|
9.3 | IC50 | 6 | — | |
ZQTAUZWIZMXKIL
|
9.3 | IC50 | 3 | — | |
ZQTAUZWIZMXKIL
|
9.3 | IC50 | 4 | — | |
PSYPBAHXIIVDCJ
|
9.2 | IC50 | 4 | — | |
HVYYDLJKIQKWSE
|
9.2 | IC50 | 4 | — | |
HVYYDLJKIQKWSE
|
9.2 | IC50 | 4 | — | |
OEZADIAHVKNQKD
|
9.2 | IC50 | 5 | — | |
MNDBXUUTURYVHR
|
9.2 | IC50 | 4 | — | |
DNDNLFXKQSTINI
|
9.2 | IC50 | 5 | — | |
WOGGATDLFJQWMW
|
9.2 | IC50 | 4 | — | |
WQULMASHBWSKLG
|
9.2 | IC50 | 4 | — | |
XPEZNWWCRUWHBE
|
9.2 | IC50 | 4 | — | |
DNDNLFXKQSTINI
|
9.2 | IC50 | 5 | — | |
KWSQCXSDPNEXCF
|
9.2 | IC50 | 4 | — | |
QWPPDUCOFLWBIF
|
9.2 | IC50 | 4 | — | |
ZKVBVKZJTSAZMU
|
9.2 | IC50 | 4 | — | |
SFPJVJIEXHMQRQ
|
9.2 | IC50 | 4 | — | |
YXWJKHHWHLVVOJ
|
9.2 | IC50 | 4 | — | |
XYZVJIGJAYGNHT
|
9.2 | IC50 | 6 | — | |
HYNHXXLRHDXNIA
|
9.2 | IC50 | 4 | — | |
PVROZLBFLOWVPM
|
9.2 | IC50 | 7 | — | |
UXVOVBOPSKMAOQ
|
9.2 | IC50 | 4 | — | |
XIMHZMKMSZOFRT
|
9.2 | IC50 | 4 | — | |
FCAARBOTCCXTNL
|
9.1 | IC50 | 4 | — | |
XIKHPFHYUYLQDN
|
9.1 | IC50 | 4 | — | |
PSUSMJVQHFLIDF
|
9.1 | IC50 | 2 | — | |
XMTRXGNILNKCCU
|
9.1 | IC50 | 4 | — | |
VLKCAQJYGYQIJK
|
9.1 | IC50 | 4 | — | |
BEYCUVURKUGSEQ
|
9.1 | IC50 | 2 | — | |
CGAFBDBSTQEQKJ
|
9.1 | IC50 | 4 | — | |
DTJGUSJXWUZZHK
|
9.1 | IC50 | 4 | — | |
PSEOWXHNKGQICS
|
9.1 | IC50 | 4 | — | |
YJWCQZYAZNXTHY
|
9.1 | IC50 | 4 | — | |
AQTLNSKLZWRJEV
|
9.1 | IC50 | 2 | — | |
AOGQPQXZFOWMDY
|
9.1 | IC50 | 4 | — | |
DLEKOQWTRJCXHT
|
9.1 | IC50 | 4 | — | |
QVYRETZFMPQHEC
|
9.1 | IC50 | 4 | — | |
UBPADFUJANMBLR
|
9.1 | IC50 | 4 | — | |
AUOKKBJDDQDYTE
|
9.1 | IC50 | 5 | — | |
CECBGQCBSIBXFA
|
9.1 | IC50 | 3 | — | |
FXOUERUVWLMXDR
|
9.1 | IC50 | 4 | — | |
LSFNKAAKCFVCEP
|
9.1 | IC50 | 7 | — | |
MFVDHDWORIHHOB
|
9.1 | IC50 | 4 | — | |
NQABHMIQSRWDFD
|
9.1 | IC50 | 4 | — | |
NDDDEPJKVOFKNS
|
9.0 | IC50 | 4 | — | |
NSYYFQMQNAQQGB
|
9.0 | IC50 | 4 | — |