Target Details
| UniProt AC | P27815 |
|---|---|
| Gene Symbol | PDE4A |
| Protein Name | 3',5'-cyclic-AMP phosphodiesterase 4A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF18100 (PDE4_UCR) PF00233 (PDEase_I) |
Summary
- Multi-target molecules 1,354
- Clinical molecules 3
- Avg pChEMBL 7.5
KEGG Pathways (5)
Active Molecules (1,354)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QDFKGLKTIPWNOS
|
6.6 | IC50 | 5 | — | |
QELHEVBSVCAUHV
|
6.6 | IC50 | 4 | — | |
UCCHUTIXGGVYOM
|
6.6 | IC50 | 5 | — | |
DJQNRDCGWWXDHA
|
6.6 | IC50 | 3 | — | |
FZXLJWUIPTZQQD
|
6.6 | Ki | 3 | — | |
GYKIIBHKVXZXBY
|
6.6 | IC50 | 4 | — | |
IJALVDBOEUTVBN
|
6.6 | IC50 | 4 | — | |
LHIGSNUVLANYIO
|
6.6 | IC50 | 2 | — | |
LLONFBHYVKPZCK
|
6.6 | IC50 | 4 | — | |
OATHQRZSVDHXRZ
|
6.6 | IC50 | 4 | — | |
GBWMEFKBLUNZIM
|
6.6 | IC50 | 2 | — | |
KAMHDCJXCXWDOJ
|
6.6 | IC50 | 2 | — | |
XGXOSJSGDNPEEF
|
6.6 | IC50 | 4 | — | |
KJLVJCFCBOJYEX
|
6.5 | IC50 | 3 | — | |
NULJNWINBNQZPW
|
6.5 | IC50 | 5 | — | |
UWTHGZFFTNZQDZ
|
6.5 | IC50 | 5 | — | |
YIASDUXALBOMQY
|
6.5 | IC50 | 4 | — | |
GLHZRBCLNXYTTF
|
6.5 | IC50 | 2 | — | |
OHQYEALDIFIKBY
|
6.5 | IC50 | 4 | — | |
PUJFXPWIBOJQHB
|
6.5 | IC50 | 12 | — | |
WNZKAFPJXSZWFJ
|
6.5 | IC50 | 6 | — | |
ALKGLLLPQJKCRV
|
6.5 | IC50 | 4 | — | |
CDAQIZGSCYILCB
|
6.5 | IC50 | 4 | — | |
DICYBSMLFAFOAP
|
6.5 | IC50 | 4 | — | |
GLQDANQNRADIEB
|
6.5 | IC50 | 4 | — | |
JVQZYDGQUZXTDQ
|
6.5 | IC50 | 3 | — | |
KNPLFFHAIBJZBG
|
6.5 | IC50 | 4 | — | |
NZKILVAZKDWRAR
|
6.5 | IC50 | 6 | — | |
PPHAWIZVVUURJO
|
6.5 | IC50 | 8 | Yes | |
PXTIJJMIHNFXAA
|
6.5 | IC50 | 4 | — | |
SJARNHOILQJSKN
|
6.5 | IC50 | 4 | — | |
CNIGFESSDPOCKS
|
6.5 | IC50 | 3 | — | |
DZMANEJEPAEVPF
|
6.5 | IC50 | 4 | — | |
LWYVEWRKCBNCFJ
|
6.5 | IC50 | 3 | — | |
XUANVLMFEXVBQF
|
6.5 | Ki | 3 | — | |
AWBDSVYVTQKKKJ
|
6.5 | IC50 | 4 | — | |
CZSPDYBKOUOJCH
|
6.5 | IC50 | 5 | — | |
HHUDRCZTUYRTSA
|
6.5 | IC50 | 4 | — | |
IQZZOLVGBYWFIM
|
6.5 | IC50 | 4 | — | |
LJJCYRVBDASIDX
|
6.5 | IC50 | 5 | — | |
MVBJBRFEZXJJLE
|
6.5 | IC50 | 4 | — | |
PHGIHHZUCQVJBM
|
6.5 | IC50 | 4 | — | |
UPMMDJIWRGVHSR
|
6.5 | IC50 | 6 | — | |
WHVLKHKNUNQGLI
|
6.5 | IC50 | 4 | — | |
XBAAJWHLDYXCQR
|
6.5 | IC50 | 4 | — | |
XWQHYCHXAAQZQB
|
6.5 | IC50 | 5 | — | |
JGZKXYWHNVBFJT
|
6.5 | IC50 | 4 | — | |
FBVRPENWLNLGLG
|
6.5 | IC50 | 4 | — | |
LERGZMBXLBAASW
|
6.5 | IC50 | 6 | — | |
MZWJIDRFXJVDGC
|
6.5 | IC50 | 4 | — |