Target Details
| UniProt AC | P27815 |
|---|---|
| Gene Symbol | PDE4A |
| Protein Name | 3',5'-cyclic-AMP phosphodiesterase 4A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF18100 (PDE4_UCR) PF00233 (PDEase_I) |
Summary
- Multi-target molecules 1,354
- Clinical molecules 3
- Avg pChEMBL 7.5
KEGG Pathways (5)
Active Molecules (1,354)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CNUGPCOZBJLIPA
|
6.7 | Ki | 4 | — | |
TYNNSCONBDUZBR
|
6.7 | Ki | 3 | — | |
AEBMOHIQXLCEDW
|
6.7 | Kd | 4 | — | |
CCNKVJUYQNQLPA
|
6.7 | IC50 | 4 | — | |
HISOEZAKLIMKIM
|
6.7 | Ki | 3 | — | |
IAUVQCNEDYDUSQ
|
6.7 | IC50 | 4 | — | |
JVZRSLGGZJREPI
|
6.7 | IC50 | 4 | — | |
RDNSHMMDOPSGFK
|
6.7 | IC50 | 4 | — | |
GAEOGEGXFOXKPH
|
6.7 | IC50 | 2 | — | |
ALFFQKBGWVKNSX
|
6.7 | IC50 | 3 | — | |
INDKHRIZOIEPIG
|
6.7 | IC50 | 2 | — | |
LKEVYMKDZMOTIM
|
6.7 | IC50 | 4 | — | |
NCXMJHMMJDZCEU
|
6.7 | IC50 | 4 | — | |
SPFPGSNCBFECSG
|
6.7 | IC50 | 2 | — | |
VSPGQUIYSBELGU
|
6.7 | IC50 | 4 | — | |
WGNLOXWSSSBKEK
|
6.7 | IC50 | 4 | — | |
JAEWRBICXOTWPT
|
6.7 | IC50 | 3 | — | |
LKZVGVHQSZSUFD
|
6.7 | IC50 | 4 | — | |
NDNYOPPCSGVZBY
|
6.7 | Ki | 4 | — | |
PWMBXCDZJSOTQB
|
6.7 | IC50 | 3 | — | |
QKTDYBBFKUXEOZ
|
6.7 | IC50 | 4 | — | |
WKIZWUJJDQILGH
|
6.7 | Ki | 3 | — | |
YDMASVAOSHOQRV
|
6.7 | Ki | 3 | — | |
FDOVMJSEGUQXQX
|
6.6 | IC50 | 4 | — | |
MOAIZPXPGWDXLJ
|
6.6 | IC50 | 4 | — | |
SOADCYOVHFISSX
|
6.6 | Ki | 3 | — | |
AXDLVMJAHYFBBA
|
6.6 | IC50 | 4 | — | |
BLUWLSQGJDRYLP
|
6.6 | IC50 | 3 | — | |
LGRMMJXKINGJFV
|
6.6 | IC50 | 4 | — | |
RJKWLGFYXTZMOU
|
6.6 | Ki | 3 | — | |
VRAURXTWLCTALJ
|
6.6 | IC50 | 4 | — | |
XXWSOEGOQFQTGV
|
6.6 | IC50 | 4 | — | |
YCEYKGZVRQVUNW
|
6.6 | IC50 | 4 | — | |
ZJALLMLKMUILFI
|
6.6 | IC50 | 4 | — | |
BFIFPXOXHAKNOH
|
6.6 | Ki | 3 | — | |
HGOQXTQGKPHGEY
|
6.6 | IC50 | 3 | — | |
MMUMOZBVLCNXNZ
|
6.6 | IC50 | 4 | — | |
RRKOMNZJZUGUEB
|
6.6 | IC50 | 4 | — | |
AVUQEUZIEFWTDC
|
6.6 | IC50 | 4 | — | |
GXORHWSQSORRGH
|
6.6 | IC50 | 4 | — | |
JNAXCAWEEVGSCX
|
6.6 | IC50 | 3 | — | |
NMGSQEBMRHQDOG
|
6.6 | IC50 | 4 | — | |
QKYCKCRBBBMXMF
|
6.6 | IC50 | 4 | — | |
RFWRTNNKLHHJRZ
|
6.6 | IC50 | 4 | — | |
XSKYWHOHKNAVIC
|
6.6 | IC50 | 4 | — | |
LYQNYINZEXWAQG
|
6.6 | IC50 | 4 | — | |
VSRMODZJMVEUKM
|
6.6 | IC50 | 4 | — | |
JJVMWANXAMHGPS
|
6.6 | IC50 | 4 | — | |
JTOAFEMFMSGNAF
|
6.6 | IC50 | 4 | — | |
LZZFXVQBLDVWTK
|
6.6 | IC50 | 4 | — |