Target Details
| UniProt AC | P27815 |
|---|---|
| Gene Symbol | PDE4A |
| Protein Name | 3',5'-cyclic-AMP phosphodiesterase 4A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF18100 (PDE4_UCR) PF00233 (PDEase_I) |
Summary
- Multi-target molecules 1,354
- Clinical molecules 3
- Avg pChEMBL 7.5
KEGG Pathways (5)
Active Molecules (1,354)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PPQXVSYEDVNMKT
|
6.8 | IC50 | 4 | — | |
TWWNJXWEOLLKJT
|
6.8 | IC50 | 4 | — | |
VVVNSVYXTOMPJW
|
6.8 | IC50 | 4 | — | |
WRHIKWNGCJVUOW
|
6.8 | IC50 | 6 | — | |
GSSCJTPNAQEUCB
|
6.8 | IC50 | 2 | — | |
GVRRXASZZAKBMN
|
6.8 | IC50 | 3 | — | |
HJORMJIFDVBMOB
|
6.8 | IC50 | 6 | — | |
RAFCFNZBQHYJSO
|
6.8 | IC50 | 4 | — | |
RQCIGHZUMYJCCJ
|
6.8 | IC50 | 3 | — | |
FVPAKTWMPJJNNZ
|
6.8 | IC50 | 4 | — | |
QGRFAJXJBYWDDZ
|
6.8 | Ki | 3 | — | |
ULQNAQGVZXNYDA
|
6.8 | IC50 | 3 | — | |
WXZZRVFNPNQGRD
|
6.8 | IC50 | 2 | — | |
FXGLUJHMJSFMFN
|
6.8 | IC50 | 6 | — | |
UBNAXKVAGIAFDG
|
6.8 | IC50 | 4 | — | |
UBYNBZKQYLBKFN
|
6.8 | IC50 | 4 | — | |
FGOAWTXGIORNAM
|
6.8 | IC50 | 3 | — | |
RHRMVOLUBKHHHM
|
6.8 | Ki | 3 | — | |
TYIBVHZITAXGDO
|
6.8 | Ki | 3 | — | |
CPRRZYUTSOZMLR
|
6.8 | IC50 | 4 | — | |
GGBSVVWNJGUOLN
|
6.8 | IC50 | 2 | — | |
HAWFVOHRJWLGGU
|
6.8 | IC50 | 4 | — | |
HTUFGGLEPYKOSR
|
6.8 | IC50 | 4 | — | |
SCAQJDLHHQAAFF
|
6.8 | Ki | 3 | — | |
ULKIELHDMWBCFZ
|
6.8 | IC50 | 6 | — | |
VMCWSNPVMPDJKY
|
6.8 | IC50 | 4 | — | |
HTZYCNVPJINMRJ
|
6.7 | Ki | 4 | — | |
URIRVYFWHKYUDQ
|
6.7 | IC50 | 6 | — | |
CRKMXHLUZCJURN
|
6.7 | IC50 | 3 | — | |
FJBUIEZNAFNOQA
|
6.7 | IC50 | 4 | — | |
SDZFOFNADNADKA
|
6.7 | IC50 | 4 | — | |
HJORMJIFDVBMOB
|
6.7 | IC50 | 6 | — | |
MMQKMLRIZHMIAU
|
6.7 | Ki | 4 | — | |
MXRZRMQHGDCNEC
|
6.7 | IC50 | 4 | — | |
UMUFOIVYCZZNQK
|
6.7 | IC50 | 4 | — | |
ALHMDZSGQSSLJK
|
6.7 | IC50 | 4 | — | |
ARYMSOFDUIIUNT
|
6.7 | IC50 | 4 | — | |
DUDAJACKYYHAFH
|
6.7 | IC50 | 4 | — | |
GNJIHIZQGDXYIS
|
6.7 | IC50 | 4 | — | |
GVUSQUVPOHOCQF
|
6.7 | IC50 | 4 | — | |
HLTNUUDVLLFYTN
|
6.7 | IC50 | 2 | — | |
RRRMTTFOHGYQIH
|
6.7 | IC50 | 6 | — | |
SMOBFXSXJCNBMQ
|
6.7 | IC50 | 4 | — | |
VOETXZPBUOBDCC
|
6.7 | IC50 | 4 | — | |
VWTOPXBUNQDCKW
|
6.7 | IC50 | 4 | — | |
VYLHRODYBXCVOV
|
6.7 | IC50 | 4 | — | |
WCKUPOIOQDQXOE
|
6.7 | IC50 | 5 | — | |
XLIGEVMSLRBZGG
|
6.7 | IC50 | 6 | — | |
ZHOCQFVWAAJXSH
|
6.7 | IC50 | 4 | — | |
ZPEFXFXPZVPLLR
|
6.7 | IC50 | 4 | — |