Target Details
| UniProt AC | P27815 |
|---|---|
| Gene Symbol | PDE4A |
| Protein Name | 3',5'-cyclic-AMP phosphodiesterase 4A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF18100 (PDE4_UCR) PF00233 (PDEase_I) |
Summary
- Multi-target molecules 1,354
- Clinical molecules 3
- Avg pChEMBL 7.5
KEGG Pathways (5)
Active Molecules (1,354)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GOBQSCBEINUNFL
|
9.6 | IC50 | 24 | — | |
PTKJWJVATJSROG
|
9.6 | Kd | 4 | — | |
SOWPFNZYANAGNV
|
9.6 | IC50 | 4 | — | |
VNHHTXGKKXMXGW
|
9.6 | IC50 | 4 | — | |
IIXVILNNIWHUJI
|
9.5 | IC50 | 4 | — | |
JCWCKXNSHPKKEK
|
9.5 | IC50 | 4 | — | |
PXYPUNRFIKKXFX
|
9.5 | IC50 | 4 | — | |
QGELAKDHJSCTHV
|
9.5 | IC50 | 4 | — | |
SRUGDVLQDNLYGA
|
9.5 | IC50 | 4 | — | |
ZKJSUXYYCBKKHN
|
9.5 | IC50 | 4 | — | |
ZZIYTDPDYPNEHS
|
9.5 | IC50 | 3 | — | |
AFCWMWBOATWMJV
|
9.5 | IC50 | 24 | — | |
DKSKKVAOIPURFT
|
9.5 | IC50 | 24 | — | |
HRXLYMCUTJFRLZ
|
9.5 | IC50 | 4 | — | |
NZTAZJDYGSXAMS
|
9.5 | IC50 | 4 | — | |
LWGNZANWYDVSLC
|
9.5 | IC50 | 4 | — | |
JJOFHTMQOOJCKZ
|
9.5 | IC50 | 4 | — | |
JJOFHTMQOOJCKZ
|
9.5 | IC50 | 4 | — | |
MQQMKMLATGRCEW
|
9.5 | IC50 | 4 | — | |
NXKMKQNQJSICGX
|
9.4 | IC50 | 4 | — | |
ACPLWVLQDOXSMT
|
9.4 | IC50 | 4 | — | |
OHIUQAZROSYCMC
|
9.4 | IC50 | 3 | — | |
BPCBVEZGCYQKMS
|
9.4 | IC50 | 4 | — | |
IONUQMBLUOOOBQ
|
9.4 | IC50 | 4 | — | |
LCJPYDPFBGENCI
|
9.4 | IC50 | 4 | — | |
QHEUBKNOJMYNLT
|
9.4 | IC50 | 4 | — | |
SDOZEKMFHJJCPN
|
9.4 | IC50 | 4 | — | |
SPOLCPORTSDTGD
|
9.4 | IC50 | 4 | — | |
YDLQPURWTSDWCC
|
9.4 | IC50 | 4 | — | |
IEUGAGUQAUJRBX
|
9.4 | IC50 | 4 | — | |
SBFUKORMVPEKAI
|
9.4 | IC50 | 4 | — | |
ZYQHRABKRQWTBJ
|
9.3 | IC50 | 2 | — | |
PSYPBAHXIIVDCJ
|
9.3 | IC50 | 4 | — | |
WOQMDRAFIAHCIG
|
9.3 | IC50 | 4 | — | |
JTGRNMGEASTCHA
|
9.3 | IC50 | 4 | — | |
QUYNJXWGUKWZLL
|
9.3 | IC50 | 6 | — | |
VYFKDGSQQMQLMD
|
9.3 | IC50 | 4 | — | |
AASKIWUYRYLTIE
|
9.3 | IC50 | 4 | — | |
CSNUCLKQPKBQNG
|
9.3 | IC50 | 4 | — | |
CSNUCLKQPKBQNG
|
9.3 | IC50 | 4 | — | |
NRTPACQHCGILGF
|
9.3 | IC50 | 4 | — | |
OPMPGFFLKCUJGU
|
9.3 | IC50 | 4 | — | |
YDDOKULECCVFMB
|
9.3 | IC50 | 3 | — | |
XNCDYFQUBJDZGN
|
9.3 | IC50 | 4 | — | |
XNCDYFQUBJDZGN
|
9.3 | IC50 | 4 | — | |
GZOUIMXMENCWQZ
|
9.3 | IC50 | 4 | — | |
GZOUIMXMENCWQZ
|
9.3 | IC50 | 4 | — | |
PSYPBAHXIIVDCJ
|
9.3 | IC50 | 4 | — | |
RSLMMIUFYJQNAI
|
9.3 | IC50 | 4 | — | |
LWGNZANWYDVSLC
|
9.3 | IC50 | 4 | — |