Target Details
| UniProt AC | P27815 |
|---|---|
| Gene Symbol | PDE4A |
| Protein Name | 3',5'-cyclic-AMP phosphodiesterase 4A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF18100 (PDE4_UCR) PF00233 (PDEase_I) |
Summary
- Multi-target molecules 1,354
- Clinical molecules 3
- Avg pChEMBL 7.5
KEGG Pathways (5)
Active Molecules (1,354)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BQOGBJWRPQNEJB
|
6.9 | IC50 | 4 | — | |
DVPHOJPLPMGUJK
|
6.9 | IC50 | 3 | — | |
OETGNFHLFFSJQQ
|
6.9 | IC50 | 4 | — | |
WONHLGXBIZZDTI
|
6.9 | IC50 | 4 | — | |
ZJGKERLRECRRHY
|
6.9 | IC50 | 4 | — | |
KKUKTBVEYAJFEF
|
6.9 | IC50 | 4 | — | |
NBNCEZNBWYPDFB
|
6.9 | IC50 | 4 | — | |
SHBSLLKGHHNCQK
|
6.9 | IC50 | 4 | — | |
TURCQYBAPKWUEP
|
6.9 | IC50 | 4 | — | |
HOOKGSVYZWYNRS
|
6.9 | IC50 | 4 | — | |
DDKUJFXMLKEDRM
|
6.9 | Ki | 4 | — | |
PYCQROXMJZTAEC
|
6.9 | Ki | 4 | — | |
SMJWZBPNUICRQK
|
6.9 | IC50 | 4 | — | |
XATDAGYWANUZJH
|
6.9 | IC50 | 4 | — | |
XRSMIHKFCVUXDP
|
6.9 | Ki | 3 | — | |
CMQJWHDXTPYSNM
|
6.8 | IC50 | 4 | — | |
HDSKSSPIAVPTNS
|
6.8 | IC50 | 3 | — | |
HPYBFHOINKPXAH
|
6.8 | IC50 | 4 | — | |
KDMOASCHWTZIML
|
6.8 | IC50 | 4 | — | |
PVBVRQMAUYVLOU
|
6.8 | IC50 | 4 | — | |
TXOWTJJUOMBYJF
|
6.8 | IC50 | 4 | — | |
ZGTKBCRXUMJCPQ
|
6.8 | IC50 | 4 | — | |
PKGAXGNVVMHTJZ
|
6.8 | IC50 | 4 | — | |
SGKGAGMPKNULQW
|
6.8 | IC50 | 4 | — | |
VNQSENKMPYKPJX
|
6.8 | IC50 | 4 | — | |
DNLRZCUCMQKICE
|
6.8 | Ki | 3 | — | |
BHLGGZNIHLIJNR
|
6.8 | IC50 | 4 | — | |
CWPNCIOMBLFPGU
|
6.8 | IC50 | 4 | — | |
HQKLMNBLQVGJKB
|
6.8 | IC50 | 4 | — | |
KLQIHSRSOJJAMH
|
6.8 | IC50 | 4 | — | |
LQFOHBHJWWQMHJ
|
6.8 | IC50 | 4 | — | |
OOBLUJRKRDCDBQ
|
6.8 | IC50 | 4 | — | |
QNZGJJKAOJFFSP
|
6.8 | IC50 | 4 | — | |
UWJAFRDFISOYFE
|
6.8 | IC50 | 4 | — | |
ZPKXBOPRMSHUDR
|
6.8 | IC50 | 4 | — | |
DYMRKAXKZNLFOP
|
6.8 | Ki | 3 | — | |
IKTHWSKYRJPRFX
|
6.8 | IC50 | 2 | — | |
AXZKFSDYFLRTKE
|
6.8 | IC50 | 4 | — | |
BBIPVJCGIASXJB
|
6.8 | Ki | 7 | — | |
BHEOYIGPFQUZIV
|
6.8 | IC50 | 4 | — | |
BYYHDFCCMVGVAV
|
6.8 | IC50 | 4 | — | |
CKHXIYDCQPVVOE
|
6.8 | Ki | 4 | — | |
HJMQDJPMQIHLPB
|
6.8 | IC50 | 6 | — | |
IAPZXUKYTCQQFE
|
6.8 | IC50 | 6 | — | |
IGKKHAVNSJKCCF
|
6.8 | IC50 | 4 | — | |
MKZVRIBEBCVKCP
|
6.8 | IC50 | 4 | — | |
MZCBWUQGZGDZAW
|
6.8 | IC50 | 4 | — | |
NCSNXSRDMMPNSI
|
6.8 | IC50 | 4 | — | |
NTYCZROBEUBTBF
|
6.8 | IC50 | 6 | — | |
OXMXRHWOUVHGDC
|
6.8 | IC50 | 4 | — |