Target Details
| UniProt AC | P27815 |
|---|---|
| Gene Symbol | PDE4A |
| Protein Name | 3',5'-cyclic-AMP phosphodiesterase 4A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF18100 (PDE4_UCR) PF00233 (PDEase_I) |
Summary
- Multi-target molecules 1,354
- Clinical molecules 3
- Avg pChEMBL 7.5
KEGG Pathways (5)
Active Molecules (1,354)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QPRTWWYGPSDGAQ
|
7.0 | IC50 | 4 | — | |
ZPTWZORADURFAJ
|
7.0 | Ki | 4 | — | |
KQTBOQXYPPPCCB
|
7.0 | IC50 | 4 | — | |
LRQBXHMVEXEFBO
|
7.0 | IC50 | 3 | — | |
DFLNUZZIKCRVBO
|
7.0 | IC50 | 4 | — | |
JCDIHRDMTWMTBI
|
7.0 | IC50 | 4 | — | |
JOGZVFZJMKTJPH
|
7.0 | Ki | 4 | — | |
SKGPWAOUHRCMEJ
|
7.0 | Ki | 4 | — | |
SLLFJRFQUSVCAS
|
7.0 | IC50 | 4 | — | |
USZAGAREISWJDP
|
7.0 | IC50 | 7 | — | |
WONHLGXBIZZDTI
|
7.0 | IC50 | 4 | — | |
ZSJIVPYJQSYHBN
|
7.0 | Ki | 4 | — | |
AHZYSVGQXRJFMW
|
7.0 | Ki | 4 | — | |
DCBILCYUFOEHGI
|
7.0 | IC50 | 4 | — | |
DLTIJXDCEGNJEW
|
7.0 | IC50 | 4 | — | |
HPVSARJVHJIZBV
|
7.0 | Ki | 3 | — | |
PPFGVIYVXGCXRU
|
7.0 | IC50 | 3 | — | |
WIQOYODZISEKQB
|
7.0 | Ki | 4 | — | |
MYBATSJXBUMOOH
|
6.9 | IC50 | 3 | — | |
OKGMHDVECIFLJL
|
6.9 | IC50 | 4 | — | |
PKUYHRMPDZBAFY
|
6.9 | IC50 | 4 | — | |
WRFHSMVYMIABFW
|
6.9 | IC50 | 4 | — | |
BPBJURKFWJXNTD
|
6.9 | IC50 | 4 | — | |
HTLIQNNZGMWTCP
|
6.9 | IC50 | 4 | — | |
WJEGHVYQRQOJAQ
|
6.9 | IC50 | 4 | — | |
AEZZPAQOEUQNBB
|
6.9 | IC50 | 6 | — | |
BHJUWEUNUCJYER
|
6.9 | IC50 | 4 | — | |
BXVGSZRVMMOLBC
|
6.9 | IC50 | 4 | — | |
CJDUNKLUUVJWIS
|
6.9 | IC50 | 4 | — | |
FSRCBTSVLQDXOV
|
6.9 | IC50 | 3 | — | |
JEAJHMPBGAMZKO
|
6.9 | IC50 | 4 | — | |
JSIJXGJOXVPSCW
|
6.9 | IC50 | 6 | — | |
KXLPTRRQYABNIU
|
6.9 | IC50 | 3 | — | |
LPZMRVKAJJEVKM
|
6.9 | IC50 | 4 | — | |
NKESBLJNJIVASL
|
6.9 | IC50 | 4 | — | |
PSVLGBSHWVNMKF
|
6.9 | IC50 | 4 | — | |
PVLQCKVDYPCWRJ
|
6.9 | IC50 | 4 | — | |
RNRARDKWHJJVFT
|
6.9 | IC50 | 4 | — | |
RRIHDUBWQABECL
|
6.9 | IC50 | 4 | — | |
WYPQDUGRCRAKKH
|
6.9 | IC50 | 6 | — | |
XUNHZDJAYPEEKV
|
6.9 | IC50 | 4 | — | |
MKNJREMNOZKXPS
|
6.9 | IC50 | 4 | — | |
XWVBOPKUSVZZPJ
|
6.9 | IC50 | 4 | — | |
COONGBDOJFYLER
|
6.9 | IC50 | 4 | — | |
COSOWSDUTHWTJU
|
6.9 | IC50 | 4 | — | |
CSNUCLKQPKBQNG
|
6.9 | IC50 | 4 | — | |
FXJNCIZGQFVQLF
|
6.9 | IC50 | 4 | — | |
MFLCJOGZEKCESC
|
6.9 | Ki | 3 | — | |
VMARDPGLTIIYGC
|
6.9 | IC50 | 4 | — | |
BQFSXRKNQWALDP
|
6.9 | IC50 | 4 | — |