Target Details
| UniProt AC | P27815 |
|---|---|
| Gene Symbol | PDE4A |
| Protein Name | 3',5'-cyclic-AMP phosphodiesterase 4A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF18100 (PDE4_UCR) PF00233 (PDEase_I) |
Summary
- Multi-target molecules 1,354
- Clinical molecules 3
- Avg pChEMBL 7.5
KEGG Pathways (5)
Active Molecules (1,354)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QIWNIPLAZVSPFF
|
7.1 | IC50 | 4 | — | |
RPLYWOYMTQLVSU
|
7.1 | IC50 | 4 | — | |
XQHOSMPOYDBZSO
|
7.1 | IC50 | 4 | — | |
BVTDODKZHFYENY
|
7.1 | IC50 | 4 | — | |
MSBSDSBWEIIBIS
|
7.1 | IC50 | 4 | — | |
OAMNKRXFJCQPJW
|
7.1 | IC50 | 4 | — | |
OUGXJJANWCSNJV
|
7.1 | IC50 | 4 | — | |
CHXCBEJGWFGXHC
|
7.1 | Ki | 4 | — | |
CNTOLDSXODWVGI
|
7.1 | IC50 | 4 | — | |
IERONGKSISNSFX
|
7.1 | IC50 | 4 | — | |
IPVSYDHNAKLEPK
|
7.1 | IC50 | 4 | — | |
ISPIFLJDLBSAFD
|
7.1 | IC50 | 4 | — | |
MPPQGDQFACBNCH
|
7.1 | IC50 | 3 | — | |
VDPHNQHKTFMQPH
|
7.1 | IC50 | 4 | — | |
YOXYJRZVIGXUHE
|
7.1 | Ki | 4 | — | |
QTNUWEKKZHSUQO
|
7.1 | IC50 | 4 | — | |
QWJILALUSUNXBN
|
7.1 | IC50 | 4 | — | |
SVFGSUZGISHPNJ
|
7.1 | IC50 | 4 | — | |
UWRKNNZXJMQNKG
|
7.1 | IC50 | 3 | — | |
DXBKTQMADALMPE
|
7.0 | IC50 | 4 | — | |
SAWDLJNAAJBRMX
|
7.0 | IC50 | 4 | — | |
UBTDNVISINZMMM
|
7.0 | IC50 | 4 | — | |
UMKXDGBAQDPHBC
|
7.0 | IC50 | 2 | — | |
ZJOMIFCTGFIUAW
|
7.0 | Kd | 4 | — | |
AQWXGANUJJZTGU
|
7.0 | IC50 | 3 | — | |
CWTRJWKDYPPKFI
|
7.0 | IC50 | 4 | — | |
WUJVRGUFPADWHY
|
7.0 | IC50 | 4 | — | |
NGYRPPIHPQIGEZ
|
7.0 | IC50 | 4 | — | |
IOCQLERZNMLYQW
|
7.0 | IC50 | 4 | — | |
CJBXVGVOXRYTRI
|
7.0 | IC50 | 4 | — | |
DDKQRPGJIVXWMQ
|
7.0 | Ki | 4 | — | |
FDESCELZSWKTDU
|
7.0 | IC50 | 3 | — | |
JRMFKYXKAZWHKF
|
7.0 | IC50 | 3 | — | |
VYBRGTIPSBPGKI
|
7.0 | IC50 | 4 | — | |
CFBUZOUXXHZCFB
|
7.0 | IC50 | 4 | — | |
FJLVGNYIAHIESD
|
7.0 | Ki | 4 | — | |
FWTNYXVPIAEBOQ
|
7.0 | IC50 | 5 | — | |
GZVHGBGPVKLJDQ
|
7.0 | IC50 | 4 | — | |
IHTDRAFPVZMGCQ
|
7.0 | IC50 | 6 | — | |
MRBFFQVXMIGKST
|
7.0 | IC50 | 4 | — | |
NMHVGUIPQDKNJJ
|
7.0 | IC50 | 4 | — | |
ODTMPGUGTQXMBN
|
7.0 | IC50 | 4 | — | |
OZDUMOKVDZODEB
|
7.0 | IC50 | 4 | — | |
YRCIXIVWTRGEHV
|
7.0 | IC50 | 4 | — | |
ZFPQQBRXDLRJDH
|
7.0 | IC50 | 4 | — | |
BDIWEEUPORVMSZ
|
7.0 | IC50 | 4 | — | |
IESKAFPEEMSDOP
|
7.0 | Ki | 3 | — | |
PYGGWLWYZUEZDS
|
7.0 | IC50 | 4 | — | |
RJSXJUGBWBWHSB
|
7.0 | IC50 | 4 | — | |
XMTOCICLPIPODV
|
7.0 | IC50 | 3 | — |