Target Details
| UniProt AC | P27815 |
|---|---|
| Gene Symbol | PDE4A |
| Protein Name | 3',5'-cyclic-AMP phosphodiesterase 4A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF18100 (PDE4_UCR) PF00233 (PDEase_I) |
Summary
- Multi-target molecules 1,354
- Clinical molecules 3
- Avg pChEMBL 7.5
KEGG Pathways (5)
Active Molecules (1,354)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AIXOQQISNZECEU
|
7.2 | IC50 | 4 | — | |
ARCWEVSTONGWAK
|
7.2 | IC50 | 4 | — | |
FOVVRXVNPNCZHA
|
7.2 | IC50 | 4 | — | |
GAGQVLMOQSRDFQ
|
7.2 | IC50 | 4 | — | |
GAKWNBHAIWCEJO
|
7.2 | IC50 | 4 | — | |
GLUBDWKKNWGCBI
|
7.2 | IC50 | 4 | — | |
HKZHBMYWZFUQLG
|
7.2 | IC50 | 4 | — | |
QMORCHDFEGGWJD
|
7.2 | IC50 | 4 | — | |
ZWNFGCDZTYYBMZ
|
7.2 | IC50 | 4 | — | |
DWSJBSVHCVJEDX
|
7.2 | IC50 | 6 | — | |
MRBFFQVXMIGKST
|
7.2 | IC50 | 4 | — | |
XKCQUKPXCRLNRV
|
7.2 | IC50 | 4 | — | |
JZEAUROSINLLHT
|
7.1 | Ki | 4 | — | |
KBXMDPUEKMYINB
|
7.1 | Ki | 4 | — | |
PUQBWQLJPRIWLI
|
7.1 | IC50 | 4 | — | |
QMKYQHDOILEPNO
|
7.1 | Ki | 4 | — | |
RYIOVUIVRIACQM
|
7.1 | IC50 | 4 | — | |
SKFXNUMASAKKIC
|
7.1 | IC50 | 4 | — | |
SWBBTMGPRSGPCD
|
7.1 | IC50 | 4 | — | |
WUCGXMCXJRLPEJ
|
7.1 | IC50 | 2 | — | |
BAWGMUZVOXOKPF
|
7.1 | IC50 | 4 | — | |
IMOZEMNVLZVGJZ
|
7.1 | IC50 | 4 | — | |
XDBHURGONHZNJF
|
7.1 | IC50 | 4 | — | |
YWYBNQHTZBGHTD
|
7.1 | IC50 | 3 | — | |
AXLQEQVMYULXDD
|
7.1 | IC50 | 4 | — | |
DZODJYSTBGCNLF
|
7.1 | IC50 | 4 | — | |
NXVKRJCXXZXAES
|
7.1 | IC50 | 4 | — | |
SHZQSAWXMAJSSI
|
7.1 | IC50 | 4 | — | |
UZHICMGVAYPCLG
|
7.1 | IC50 | 4 | — | |
WDFOZMDHGRGPRF
|
7.1 | IC50 | 5 | — | |
NZSGGOJDVRRWTL
|
7.1 | IC50 | 5 | — | |
UTBNQNSSWODNLN
|
7.1 | IC50 | 4 | — | |
FTIDRMNTTJHUPO
|
7.1 | IC50 | 5 | — | |
HUUANGGGQAYPDU
|
7.1 | IC50 | 4 | — | |
KWUKMXYLCKXYFJ
|
7.1 | IC50 | 4 | — | |
LNZCEULLEVKFQA
|
7.1 | IC50 | 4 | — | |
LZCQFJKUAIWHRW
|
7.1 | IC50 | 6 | — | |
NMVLJLKIUKOKSB
|
7.1 | IC50 | 4 | — | |
OSGFQUPLDZBTPO
|
7.1 | IC50 | 4 | — | |
PDJCJBJJRNNEMG
|
7.1 | IC50 | 4 | — | |
QFAHXLIVMRUENH
|
7.1 | IC50 | 4 | — | |
RZAZJXDVOFZLKI
|
7.1 | IC50 | 4 | — | |
SJQXOZSDYOZKJF
|
7.1 | IC50 | 4 | — | |
TZLDNYQGARHUED
|
7.1 | IC50 | 4 | — | |
VOETXZPBUOBDCC
|
7.1 | IC50 | 4 | — | |
VVVNSVYXTOMPJW
|
7.1 | IC50 | 4 | — | |
XKBPHTUNGWWCLP
|
7.1 | IC50 | 4 | — | |
AJQZCACDXGLQGS
|
7.1 | IC50 | 4 | — | |
IMOZEMNVLZVGJZ
|
7.1 | IC50 | 4 | — | |
QHWJXFZLSVHSGH
|
7.1 | IC50 | 4 | — |