Target Details
| UniProt AC | P27815 |
|---|---|
| Gene Symbol | PDE4A |
| Protein Name | 3',5'-cyclic-AMP phosphodiesterase 4A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF18100 (PDE4_UCR) PF00233 (PDEase_I) |
Summary
- Multi-target molecules 1,354
- Clinical molecules 3
- Avg pChEMBL 7.5
KEGG Pathways (5)
Active Molecules (1,354)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QCUHKLBHHWHXAM
|
7.3 | IC50 | 4 | — | |
SXBKTNMKNCEAEF
|
7.3 | IC50 | 4 | — | |
UHUZDJMHKDQSSG
|
7.3 | IC50 | 4 | — | |
WWBMDNVOUMWXEP
|
7.3 | IC50 | 4 | — | |
AZGFYUPSXODBAO
|
7.3 | IC50 | 4 | — | |
OSIAQFSEAYCSKV
|
7.3 | IC50 | 6 | — | |
PVJLIQXJOIAHCQ
|
7.3 | IC50 | 4 | — | |
ZHUOBYXGRFSJOZ
|
7.3 | IC50 | 4 | — | |
KDRNXUFBYVXQSL
|
7.3 | IC50 | 4 | — | |
RGIGHJGWQTVJGO
|
7.3 | IC50 | 4 | — | |
YGZXJQKMMJKRBV
|
7.3 | IC50 | 4 | — | |
FHCIKJABQDYUJK
|
7.3 | IC50 | 5 | — | |
HRVGXJYBJMMTEJ
|
7.3 | IC50 | 4 | — | |
JKGFOIGGPUTHIY
|
7.3 | IC50 | 3 | — | |
LYJGBGQLQMRKKF
|
7.3 | IC50 | 4 | — | |
MWBKSPAGZZMVNI
|
7.3 | IC50 | 4 | — | |
LJEWJUWTKPBRNQ
|
7.3 | IC50 | 4 | — | |
NOSXOAFVJDFCQR
|
7.3 | IC50 | 4 | — | |
NQDQONQTHUPPNR
|
7.3 | IC50 | 4 | — | |
OHZWWRAGTGIQOP
|
7.3 | IC50 | 4 | — | |
BDYDINKSILYBOL
|
7.3 | IC50 | 5 | — | |
GNWCRBFQZDJFTI
|
7.3 | IC50 | 4 | — | |
HBDOUVSVVYQJQQ
|
7.3 | IC50 | 4 | — | |
JFIPQLSQEHFZKL
|
7.3 | IC50 | 4 | — | |
MHCDVXQKXSNQPC
|
7.3 | IC50 | 4 | — | |
PAGIVPCQHJQBLJ
|
7.3 | IC50 | 4 | — | |
PVWGPCPZYAEPPN
|
7.3 | IC50 | 4 | — | |
TWKMZYIUVKFGDK
|
7.3 | IC50 | 3 | — | |
UWZTUNHQFYSEGU
|
7.3 | IC50 | 6 | — | |
ZKPQLHMITFDDQQ
|
7.3 | Ki | 4 | — | |
ZTRURMGGKLLTNK
|
7.3 | IC50 | 4 | — | |
GACGDQDYWVSBEL
|
7.3 | IC50 | 4 | — | |
HBRLPTMZNRCNBL
|
7.3 | IC50 | 4 | — | |
WGUXBENBNHCCQX
|
7.3 | IC50 | 4 | — | |
YFASTVZAZWFDOS
|
7.3 | Ki | 4 | — | |
CQGRVMWIHSGBNM
|
7.3 | IC50 | 4 | — | |
KOYGDVZTTWVMNV
|
7.3 | IC50 | 4 | — | |
OZHBSVBPSKZWMX
|
7.3 | IC50 | 4 | — | |
QHBGWNQSFRIXFV
|
7.3 | IC50 | 4 | — | |
YDLQPURWTSDWCC
|
7.3 | IC50 | 4 | — | |
YPVISLYCIGDNCE
|
7.3 | IC50 | 4 | — | |
MPXKKKYXZROOTK
|
7.3 | IC50 | 4 | — | |
NBMOZEZCSGFNAZ
|
7.3 | IC50 | 4 | — | |
UZJJLBYHSDGPBB
|
7.3 | IC50 | 4 | — | |
VTRNMYGATDHWOK
|
7.3 | IC50 | 4 | — | |
YQPSCZXPOGCSMA
|
7.3 | IC50 | 4 | — | |
ZJVFLBOZORBYFE
|
7.3 | IC50 | 4 | — | |
GGBPMJVCUHMAJB
|
7.3 | IC50 | 4 | — | |
URQYGZHYLQIBIU
|
7.3 | IC50 | 4 | — | |
COLQUUDNEIJASV
|
7.2 | IC50 | 4 | — |