Target Details
| UniProt AC | P27815 |
|---|---|
| Gene Symbol | PDE4A |
| Protein Name | 3',5'-cyclic-AMP phosphodiesterase 4A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF18100 (PDE4_UCR) PF00233 (PDEase_I) |
Summary
- Multi-target molecules 1,354
- Clinical molecules 3
- Avg pChEMBL 7.5
KEGG Pathways (5)
Active Molecules (1,354)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MJHYQMWSWMXYQH
|
7.5 | IC50 | 3 | — | |
BJEUCBFCNBFMLD
|
7.5 | IC50 | 4 | — | |
CEMQXLVYSIOKKQ
|
7.5 | IC50 | 4 | — | |
KUWALJOWQIFEPB
|
7.5 | IC50 | 3 | — | |
OYOKUCRYUNATTC
|
7.5 | IC50 | 4 | — | |
QBJZJLGONNMMNS
|
7.5 | IC50 | 4 | — | |
XQZMYDIWLZMXHX
|
7.5 | IC50 | 4 | — | |
JXDYJNOWRSRYDW
|
7.5 | IC50 | 4 | — | |
DTJNUDNOBCGTPD
|
7.4 | IC50 | 3 | — | |
GSXKMMPZFVRZAU
|
7.4 | IC50 | 4 | — | |
KHBZAHNRQJPBQK
|
7.4 | IC50 | 4 | — | |
MAXOLFIODKJKGF
|
7.4 | IC50 | 4 | — | |
OSRABMBLFJSDDJ
|
7.4 | IC50 | 6 | — | |
WYSBJUKHVQZOHC
|
7.4 | IC50 | 3 | — | |
XIVVDTJZCTVMFP
|
7.4 | IC50 | 4 | — | |
HMTGPYRFOCPERJ
|
7.4 | IC50 | 4 | — | |
JDQDGTOBHTWISP
|
7.4 | Ki | 4 | — | |
DBCKRBGYGMVSTI
|
7.4 | IC50 | 3 | — | |
DWGPOBJDCKSRHT
|
7.4 | IC50 | 4 | — | |
KFPBEJNFGNVRCD
|
7.4 | IC50 | 2 | — | |
NXQIEDDZYQXLGS
|
7.4 | IC50 | 3 | — | |
APQCTKWSIMEXKR
|
7.4 | IC50 | 4 | — | |
CMBMBGWFZPINMW
|
7.4 | IC50 | 4 | — | |
OUXBYUBGWJQGHZ
|
7.4 | IC50 | 4 | — | |
YALCOJRYUXNVOV
|
7.4 | IC50 | 4 | — | |
FRRBVAWAIKCZEF
|
7.4 | IC50 | 4 | — | |
KGLQCVFPIGHIAB
|
7.4 | IC50 | 4 | — | |
LKQLMGVBCLAGOJ
|
7.4 | IC50 | 6 | — | |
MWSUARADAXHTLM
|
7.4 | IC50 | 4 | — | |
OKFXGRLQLSKPJJ
|
7.4 | IC50 | 4 | — | |
PKNCMHIFSWTLHO
|
7.4 | IC50 | 4 | — | |
QWECFCKUHAMUOT
|
7.4 | IC50 | 4 | — | |
VOETXZPBUOBDCC
|
7.4 | IC50 | 4 | — | |
VOKPVPDGZJRVLI
|
7.4 | IC50 | 4 | — | |
YDADFGXXCHDXFC
|
7.4 | IC50 | 4 | — | |
ZKXQMGSFLNBQON
|
7.4 | IC50 | 4 | — | |
CEPZWKIBCFQSSQ
|
7.4 | IC50 | 4 | — | |
GQSMQGGJKLJVOI
|
7.4 | IC50 | 4 | — | |
HIZORNOKOHJTBO
|
7.4 | IC50 | 3 | — | |
APZGHLKUAICCAJ
|
7.4 | IC50 | 4 | — | |
DYHGFTMEUMYPOC
|
7.4 | IC50 | 4 | — | |
WGCLVKDICJNHNO
|
7.4 | IC50 | 4 | — | |
XOINTZNHWHXINB
|
7.4 | IC50 | 4 | — | |
PYEOZIHIJFSCOO
|
7.4 | IC50 | 4 | — | |
SMOWDUACKVMUAN
|
7.4 | IC50 | 3 | — | |
XNIYDLUVCSJKFF
|
7.4 | IC50 | 3 | — | |
MYPOVEUFNMJGML
|
7.4 | IC50 | 2 | — | |
QWJORUKKCABZPO
|
7.4 | IC50 | 4 | — | |
RXWLKROKFKZBEA
|
7.4 | IC50 | 4 | — | |
URXUAYQZIDJXGT
|
7.4 | IC50 | 4 | — |