Target Details
| UniProt AC | P27815 |
|---|---|
| Gene Symbol | PDE4A |
| Protein Name | 3',5'-cyclic-AMP phosphodiesterase 4A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF18100 (PDE4_UCR) PF00233 (PDEase_I) |
Summary
- Multi-target molecules 1,354
- Clinical molecules 3
- Avg pChEMBL 7.5
KEGG Pathways (5)
Active Molecules (1,354)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YUSMVVYYGMJNLB
|
7.6 | IC50 | 4 | — | |
ZDUSDAZRVNATDN
|
7.6 | IC50 | 4 | — | |
XJLNUYAEDMBFAZ
|
7.6 | IC50 | 3 | — | |
XWBNVRGWNULCLK
|
7.6 | IC50 | 4 | — | |
ACVHTZRYROUGLO
|
7.5 | IC50 | 4 | — | |
HVVGNLROCIOALI
|
7.5 | IC50 | 4 | — | |
KSRRPXVKALLJHV
|
7.5 | IC50 | 4 | — | |
SDXDROLDNVOSMH
|
7.5 | IC50 | 3 | — | |
SIJLGTONYCHCNA
|
7.5 | IC50 | 4 | — | |
SKSQSCQKTAQENI
|
7.5 | IC50 | 4 | — | |
GHYMFLJYUUFYNZ
|
7.5 | IC50 | 4 | — | |
JNDBRXMEQJISOU
|
7.5 | IC50 | 4 | — | |
SCIDSYICJROITB
|
7.5 | IC50 | 4 | — | |
YDSNGCAFYIQMNI
|
7.5 | IC50 | 4 | — | |
SRLHMGKYTUHFKW
|
7.5 | IC50 | 4 | — | |
AYHYIRASVWMGJI
|
7.5 | IC50 | 4 | — | |
DKLXINMEXJFCET
|
7.5 | IC50 | 6 | — | |
FGESEXRYOVBTIB
|
7.5 | IC50 | 4 | — | |
PKFGHAIJIHZQFD
|
7.5 | IC50 | 4 | — | |
PPHAWIZVVUURJO
|
7.5 | IC50 | 8 | Yes | |
SEZOJNSDVQCGGH
|
7.5 | IC50 | 4 | — | |
UVOMWHXGFUBTQK
|
7.5 | IC50 | 4 | — | |
XAEPFDVBAVYYLP
|
7.5 | IC50 | 4 | — | |
ZDMBKIHGRXLNRP
|
7.5 | IC50 | 4 | — | |
KGVHJHCDZZCOPP
|
7.5 | Ki | 4 | — | |
LBNIQKADHDXTKV
|
7.5 | IC50 | 4 | — | |
RDXNYSSQQZEEJF
|
7.5 | IC50 | 4 | — | |
VVRXUNSKFAKWSF
|
7.5 | IC50 | 6 | — | |
WKINNFHNVQMBKZ
|
7.5 | IC50 | 5 | — | |
FGYNRNOOSHCFPR
|
7.5 | IC50 | 4 | — | |
LTQPXIUEDFTWNR
|
7.5 | IC50 | 3 | — | |
NSHNYBPSXRQLAS
|
7.5 | IC50 | 2 | — | |
OFWLISQOQVGMBV
|
7.5 | IC50 | 4 | — | |
OTWDFHFFUNOBLA
|
7.5 | IC50 | 4 | — | |
PADQBOCDWXQDKL
|
7.5 | IC50 | 4 | — | |
PEGGCQCFFVKPAO
|
7.5 | IC50 | 4 | — | |
UBOJZLRKEYASPJ
|
7.5 | IC50 | 3 | — | |
UBOJZLRKEYASPJ
|
7.5 | IC50 | 4 | — | |
UJDRSYOCCUNRBX
|
7.5 | IC50 | 4 | — | |
VUISAJWDMBCIQP
|
7.5 | IC50 | 4 | — | |
WZZXQGHMUNKNST
|
7.5 | IC50 | 4 | — | |
BDZYIKRXVZUNQN
|
7.5 | IC50 | 3 | — | |
HBUJRYNMNPGQOW
|
7.5 | IC50 | 4 | — | |
MTKJJVQIOIGEFS
|
7.5 | IC50 | 4 | — | |
PIGDEODSCDFZBD
|
7.5 | IC50 | 4 | — | |
TUHZURBDZPBKQB
|
7.5 | IC50 | 3 | — | |
UGZDKECEYYYBSI
|
7.5 | IC50 | 4 | — | |
XRUNGFIMYAZVGB
|
7.5 | Ki | 4 | — | |
AUHPGOLYFSHALS
|
7.5 | IC50 | 4 | — | |
LIYOPOWLJZJRAK
|
7.5 | IC50 | 4 | — |