Target Details
| UniProt AC | P27815 |
|---|---|
| Gene Symbol | PDE4A |
| Protein Name | 3',5'-cyclic-AMP phosphodiesterase 4A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF18100 (PDE4_UCR) PF00233 (PDEase_I) |
Summary
- Multi-target molecules 1,354
- Clinical molecules 3
- Avg pChEMBL 7.5
KEGG Pathways (5)
Active Molecules (1,354)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FOXQXUPYSIQJFO
|
7.7 | IC50 | 4 | — | |
HVZVPGFXFPHGPA
|
7.7 | IC50 | 4 | — | |
LCTMXACJLVAYNA
|
7.7 | IC50 | 4 | — | |
MERWGYSKTWXXSP
|
7.7 | IC50 | 3 | — | |
NMKWYXGLIWTXRG
|
7.7 | IC50 | 4 | — | |
NZZVPKJQFQTLOP
|
7.7 | IC50 | 4 | — | |
OZUNUTXZGBJXGF
|
7.7 | IC50 | 4 | — | |
GRFHQTKEAOBDST
|
7.7 | IC50 | 3 | — | |
CSLQYGQMUXSECS
|
7.7 | IC50 | 4 | — | |
UBVKVEOYBYZYGM
|
7.7 | IC50 | 4 | — | |
URYVNEIOAZXYPR
|
7.7 | IC50 | 3 | — | |
VOILLODEUKMPEX
|
7.7 | IC50 | 4 | — | |
GTAREIVODMENMP
|
7.7 | IC50 | 4 | — | |
WSHHEXFRSSGSLG
|
7.7 | IC50 | 4 | — | |
WXDAFRGTHFUIST
|
7.7 | IC50 | 3 | — | |
DHCOPPHTVOXDKU
|
7.6 | IC50 | 3 | — | |
GJJMKGXNHORNRI
|
7.6 | IC50 | 3 | — | |
KDPKDOHAJHCGSZ
|
7.6 | IC50 | 4 | — | |
LDKCNCXJCVADEV
|
7.6 | IC50 | 5 | — | |
UPVVGSOGUOKFGS
|
7.6 | IC50 | 4 | — | |
WLRPIEXEHDHNIW
|
7.6 | IC50 | 2 | — | |
XKDMBJJSWDXWNU
|
7.6 | IC50 | 4 | — | |
FUWCYRLOJQXZEJ
|
7.6 | IC50 | 4 | — | |
ZQTGMZNEQOGOQC
|
7.6 | IC50 | 4 | — | |
HXVNESZNUYSKMT
|
7.6 | IC50 | 3 | — | |
AMLLKGOZJKLVGB
|
7.6 | IC50 | 4 | — | |
FRHMLRQQIOCJKU
|
7.6 | IC50 | 4 | — | |
FDJPZBHXIZZOLP
|
7.6 | IC50 | 4 | — | |
FZHQFKLHOFLUQF
|
7.6 | IC50 | 4 | — | |
GHPVAQLECQUTMD
|
7.6 | IC50 | 3 | — | |
JWNVKTDNDORZTE
|
7.6 | IC50 | 4 | — | |
KPYILSHDSUADBY
|
7.6 | IC50 | 4 | — | |
LEDSLQCBWQCPEZ
|
7.6 | IC50 | 4 | — | |
NDVMSTHWOUOSMI
|
7.6 | IC50 | 4 | — | |
NDVMSTHWOUOSMI
|
7.6 | IC50 | 4 | — | |
NXQIEDDZYQXLGS
|
7.6 | IC50 | 3 | — | |
VJAHAVJLFBDRIZ
|
7.6 | IC50 | 4 | — | |
VQZLXFXVXIGVSV
|
7.6 | IC50 | 4 | — | |
WDMINEFVSXLMJR
|
7.6 | IC50 | 4 | — | |
WIOFCDPOPOOQNI
|
7.6 | IC50 | 4 | — | |
XBCOPPJJOUTQEB
|
7.6 | IC50 | 4 | — | |
XVPMLCYXSAROSC
|
7.6 | IC50 | 4 | — | |
SNPDIBMAAUTAIH
|
7.6 | IC50 | 4 | — | |
FKAXUOKPFFFYTF
|
7.6 | IC50 | 4 | — | |
LHHMNAHPCIAINQ
|
7.6 | IC50 | 4 | — | |
LOJKHUDVHIIXBA
|
7.6 | IC50 | 4 | — | |
WYVVCFNADZMHEN
|
7.6 | IC50 | 3 | — | |
GRAADZXYCUWZRB
|
7.6 | IC50 | 4 | — | |
LPBBOFAPPVCKTQ
|
7.6 | IC50 | 4 | — | |
VQTBBBGKBIKAAN
|
7.6 | IC50 | 4 | — |