Target Details
| UniProt AC | P27815 |
|---|---|
| Gene Symbol | PDE4A |
| Protein Name | 3',5'-cyclic-AMP phosphodiesterase 4A |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF18100 (PDE4_UCR) PF00233 (PDEase_I) |
Summary
- Multi-target molecules 1,354
- Clinical molecules 3
- Avg pChEMBL 7.5
KEGG Pathways (5)
Active Molecules (1,354)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LROCAZWHWFXPFN
|
7.8 | IC50 | 4 | — | |
NGLYSTCXIRGOIR
|
7.8 | IC50 | 4 | — | |
OEHQEKSCIBKRPE
|
7.8 | IC50 | 4 | — | |
OHASJOLVTWQDCA
|
7.8 | IC50 | 4 | — | |
UJFNOAVXTSKOEP
|
7.8 | IC50 | 4 | — | |
GXYHCJBIWBLNEK
|
7.8 | IC50 | 4 | — | |
WAYXCSKMOOKIDO
|
7.8 | IC50 | 4 | — | |
APHANYYADPNRCL
|
7.8 | IC50 | 4 | — | |
BGARLRUFQVBBEZ
|
7.8 | IC50 | 4 | — | |
CMEUONJHZIAWNP
|
7.8 | IC50 | 4 | — | |
FSIVVLNKOBRHFI
|
7.8 | IC50 | 6 | — | |
GEJPLNWGEJLXJN
|
7.8 | IC50 | 4 | — | |
IAQZKDQBUKXOIW
|
7.8 | IC50 | 4 | — | |
JFIPQLSQEHFZKL
|
7.8 | IC50 | 4 | — | |
KKMHBNSEVLDXRU
|
7.8 | IC50 | 4 | — | |
KUYGTFAVPSRLAO
|
7.8 | IC50 | 4 | — | |
LCFPQNNXKJMNSH
|
7.8 | IC50 | 6 | — | |
MGLGPHGYDFRMFI
|
7.8 | IC50 | 4 | — | |
OCPPCOZBRCBGCK
|
7.8 | IC50 | 4 | — | |
OEGSOWUEEMPITO
|
7.8 | IC50 | 4 | — | |
OGPDSHZLXMVDTO
|
7.8 | IC50 | 6 | — | |
SNKXLTDCGDAPHC
|
7.8 | IC50 | 4 | — | |
ZDSSYIMMEPTDEO
|
7.8 | IC50 | 3 | — | |
ZININGNRPUGNSL
|
7.8 | IC50 | 3 | — | |
NHPLJPOZRUZKND
|
7.8 | IC50 | 3 | — | |
LLKDXLOAXVIBRW
|
7.8 | IC50 | 4 | — | |
GCCPWRCOMQRJON
|
7.8 | IC50 | 4 | — | |
HJSDGVOHRUVZOW
|
7.8 | IC50 | 4 | — | |
OCELOSKSDRCMQK
|
7.8 | IC50 | 4 | — | |
PMXQBXHVHKGVCD
|
7.8 | IC50 | 4 | — | |
UGOZDRKOSSYHBA
|
7.8 | IC50 | 4 | — | |
UGOZDRKOSSYHBA
|
7.8 | IC50 | 3 | — | |
CLHCDDFDRGZJEO
|
7.8 | IC50 | 4 | — | |
CTXZJNXACMKAGH
|
7.8 | IC50 | 4 | — | |
CKDYACSCRUTGHR
|
7.7 | IC50 | 3 | — | |
YFBAOXITVIDIPH
|
7.7 | IC50 | 3 | — | |
PNCIDWSACMQCIG
|
7.7 | IC50 | 3 | — | |
SGDLTWNJVPOTRT
|
7.7 | IC50 | 3 | — | |
ADXIPZNPTFVGDB
|
7.7 | IC50 | 3 | — | |
CQNWMZNUZDLOBT
|
7.7 | IC50 | 4 | — | |
NUMTXTPCPDSVTH
|
7.7 | IC50 | 2 | — | |
PZZXIGQDKGIHNM
|
7.7 | IC50 | 4 | — | |
RAQWULABCGLUNW
|
7.7 | IC50 | 2 | — | |
UPBKTTZHNZAEQA
|
7.7 | IC50 | 2 | — | |
UQCXHZJRNQMJDO
|
7.7 | IC50 | 4 | — | |
MKFKTQOJJMIDOC
|
7.7 | IC50 | 3 | — | |
WMBGBRRUSMUDQB
|
7.7 | IC50 | 4 | — | |
AAWHVDHSXWEWJR
|
7.7 | IC50 | 4 | — | |
AWOFSUFKCXRJMV
|
7.7 | IC50 | 3 | — | |
DITHSWKFXOPMHH
|
7.7 | IC50 | 3 | — |