Target Details
| UniProt AC | P27695 |
|---|---|
| Gene Symbol | APEX1 |
| Protein Name | DNA repair nuclease/redox regulator APEX1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF03372 (Exo_endo_phos) |
Summary
- Multi-target molecules 4
- Clinical molecules 0
- Avg pChEMBL 7.09
KEGG Pathways (1)
Active Molecules (4)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GIXWDMTZECRIJT
|
7.3 | IC50 | 9 | — | |
VWTPGUPXPKYBNL
|
7.3 | IC50 | 8 | — | |
MWKSRKSEWLRPBL
|
7.1 | Kd | 1075 | — | |
ZTQRMGDLUGQTTF
|
6.7 | IC50 | 4 | — |