Target Details
| UniProt AC | P27540 |
|---|---|
| Gene Symbol | ARNT |
| Protein Name | Aryl hydrocarbon receptor nuclear translocator |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00010 (HLH) PF00989 (PAS) PF14598 (PAS_11) |
Summary
- Multi-target molecules 30
- Clinical molecules 0
- Avg pChEMBL 7.36
KEGG Pathways (7)
Top Co-occurrence Targets
- EPAS1 30 shared
Active Molecules (30)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ITVHGRMYDUEOHH
|
9.0 | IC50 | 2 | — | |
KYTFUEKZQZLJCC
|
9.0 | IC50 | 2 | — | |
NQHCZTHBPKJWBK
|
9.0 | IC50 | 2 | — | |
ONBSHRSJOPSEGS
|
8.7 | IC50 | 2 | — | |
LLQXGXPLKBHEAI
|
8.5 | IC50 | 2 | — | |
ODNKSLDGFCIXQD
|
8.4 | IC50 | 2 | — | |
UWHUYKGCGHNLEP
|
8.4 | IC50 | 2 | — | |
RBKUARNZLBUCAG
|
8.2 | IC50 | 2 | — | |
XZLDMUNIMNCFCN
|
8.2 | IC50 | 2 | — | |
FWKQVEJQEQRFGU
|
8.2 | IC50 | 2 | — | |
GUJWSWZIXSWLTL
|
7.7 | IC50 | 2 | — | |
KVBRHUQRAWRYAI
|
7.6 | IC50 | 2 | — | |
SSIWQCYLGHKCQZ
|
7.5 | IC50 | 2 | — | |
PHQHXQAFRAVKSP
|
7.1 | IC50 | 2 | — | |
FXUKXNSGAXJPHR
|
7.0 | IC50 | 2 | — | |
CDQUJZKBRAFWNG
|
7.0 | IC50 | 2 | — | |
BSLNBWGCFHYQTJ
|
7.0 | IC50 | 2 | — | |
PCJSWXIBXCRFJH
|
6.9 | IC50 | 2 | — | |
PVQSVWLZGINSSA
|
6.9 | IC50 | 2 | — | |
BFZNXAFREFMQDF
|
6.8 | IC50 | 2 | — | |
FUUWQJVNALIXDT
|
6.8 | IC50 | 2 | — | |
FGCJEVWDLATQGD
|
6.5 | IC50 | 2 | — | |
GJLPBJAKALWNPH
|
6.5 | IC50 | 2 | — | |
PQZKMXPISWCLCU
|
6.4 | IC50 | 2 | — | |
FBLSAINZUURAAQ
|
6.4 | IC50 | 2 | — | |
DDQZGFIXHMUCKK
|
6.4 | IC50 | 2 | — | |
IRUDMTDFNXURLI
|
6.3 | IC50 | 2 | — | |
MSLKJZNCDWDMHK
|
6.3 | IC50 | 2 | — | |
RBKUARNZLBUCAG
|
6.2 | IC50 | 2 | — | |
AHLKPENLDGAISD
|
6.1 | IC50 | 2 | — |