Target Details
| UniProt AC | P27487 |
|---|---|
| Gene Symbol | DPP4 |
| Protein Name | Dipeptidyl peptidase 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00930 (DPPIV_N) PF00326 (Peptidase_S9) |
Summary
- Multi-target molecules 550
- Clinical molecules 3
- Avg pChEMBL 7.78
KEGG Pathways (2)
Active Molecules (550)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NQGZMSIGTNYNPY
|
7.2 | IC50 | 2 | — | |
GVCXDPXWUCFOOE
|
7.2 | Ki | 3 | — | |
HTEXKUKUMOZCFK
|
7.2 | IC50 | 2 | — | |
PGHYBEWUAIZJET
|
7.2 | IC50 | 2 | — | |
AAMHEKBKKUYLPS
|
7.2 | IC50 | 2 | — | |
BMCGYCXNUMDZSH
|
7.2 | IC50 | 6 | — | |
DJJDMDCQSLKDBW
|
7.2 | IC50 | 2 | — | |
IQLBIWJJBRDGRO
|
7.2 | IC50 | 2 | — | |
IQLBIWJJBRDGRO
|
7.2 | IC50 | 2 | — | |
BYSBLNSCHBIOLU
|
7.1 | IC50 | 2 | — | |
HHUJSBHWHUGOTO
|
7.1 | IC50 | 2 | — | |
HHUJSBHWHUGOTO
|
7.1 | IC50 | 2 | — | |
LPGHTFZPBWNCQD
|
7.1 | IC50 | 2 | — | |
MOTWXMLKPRYXNR
|
7.1 | IC50 | 2 | — | |
DKYAPNCLSWLGEV
|
7.1 | IC50 | 2 | — | |
SWTQPEVJGWLIDH
|
7.1 | IC50 | 2 | — | |
XCUPYUKEECXEPG
|
7.1 | IC50 | 2 | — | |
YIDAVMZDHIDPFB
|
7.1 | IC50 | 2 | — | |
AOHMCYUGHQMVEI
|
7.1 | IC50 | 2 | — | |
LNDZIFCFUWGUBW
|
7.1 | IC50 | 2 | — | |
NXGCDTBNUXWSGM
|
7.1 | IC50 | 2 | — | |
NYDLAPOYXYVHSC
|
7.1 | IC50 | 3 | — | |
ZOJNVHBDZGHINU
|
7.1 | IC50 | 2 | — | |
XXVBSPRJQMYRKA
|
7.1 | IC50 | 2 | — | |
XXVBSPRJQMYRKA
|
7.1 | IC50 | 2 | — | |
NIDVIGBTBOHQNL
|
7.1 | IC50 | 2 | — | |
ADDDIJIWQWCYSH
|
7.0 | IC50 | 3 | — | |
FLSQVTUPJGNXGP
|
7.0 | IC50 | 2 | — | |
UZZDZARFWLTODD
|
7.0 | IC50 | 5 | — | |
LRINXVSRRIIMQL
|
7.0 | IC50 | 2 | — | |
MPZCONICLYEKDC
|
7.0 | IC50 | 3 | — | |
OQOKNTNHKHWJGC
|
7.0 | IC50 | 2 | — | |
NCKFTUHNPCXRDM
|
7.0 | IC50 | 6 | — | |
YJMLPSBGVRXCPM
|
7.0 | IC50 | 5 | — | |
QLNACVPURHNJCY
|
7.0 | IC50 | 2 | — | |
SYSFQGYFFKSFIC
|
7.0 | IC50 | 2 | — | |
SYSFQGYFFKSFIC
|
7.0 | IC50 | 2 | — | |
YGAZXKNSNKIHFM
|
7.0 | IC50 | 2 | — | |
YGAZXKNSNKIHFM
|
7.0 | IC50 | 2 | — | |
SVXBTHULZGXAEU
|
7.0 | IC50 | 2 | — | |
GKRHKBHELWAKHM
|
7.0 | IC50 | 2 | — | |
KDGSVHGIVBVYFE
|
7.0 | IC50 | 2 | — | |
LNQWGYANQRWXNE
|
7.0 | IC50 | 2 | — | |
LNQWGYANQRWXNE
|
7.0 | IC50 | 2 | — | |
LRINXVSRRIIMQL
|
7.0 | IC50 | 2 | — | |
PKVNQQPGIAQMEH
|
7.0 | IC50 | 4 | — | |
QHNUQBRSRCCURR
|
7.0 | IC50 | 2 | — | |
YZARUVQCPYHDDR
|
7.0 | IC50 | 3 | — | |
DDIZCHCPOMXXRE
|
7.0 | IC50 | 3 | — | |
DRQXWCARABZCPQ
|
6.9 | IC50 | 2 | — |