Target Details
| UniProt AC | P27487 |
|---|---|
| Gene Symbol | DPP4 |
| Protein Name | Dipeptidyl peptidase 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00930 (DPPIV_N) PF00326 (Peptidase_S9) |
Summary
- Multi-target molecules 550
- Clinical molecules 3
- Avg pChEMBL 7.78
KEGG Pathways (2)
Active Molecules (550)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PUKARVRQDSPFPB
|
7.4 | IC50 | 2 | — | |
SBBQYCLBXQJVIG
|
7.4 | IC50 | 4 | — | |
YZYFOKXDBHHJLB
|
7.4 | IC50 | 5 | — | |
IIKCZGQEACUCTC
|
7.3 | Ki | 2 | — | |
QAAMJGGJVHEAAE
|
7.3 | IC50 | 2 | — | |
WJHCPHJMRCWJNR
|
7.3 | IC50 | 3 | — | |
OGWARBNUWZYESR
|
7.3 | IC50 | 2 | — | |
RABCMFOALSUEDW
|
7.3 | IC50 | 2 | — | |
TXDCCDZUBCMPHL
|
7.3 | IC50 | 2 | — | |
DGFODDFZJTVDBE
|
7.3 | IC50 | 3 | — | |
JAWWAXWVCGDCRL
|
7.3 | IC50 | 2 | — | |
SZJRQDUCFNDXRI
|
7.3 | IC50 | 2 | — | |
WDOUSOAMPWULRN
|
7.3 | IC50 | 2 | — | |
PQBMPUQYJGLDHI
|
7.3 | IC50 | 2 | — | |
QTZTUCOZZMQUFY
|
7.3 | IC50 | 2 | — | |
QTZTUCOZZMQUFY
|
7.3 | IC50 | 2 | — | |
QTZTUCOZZMQUFY
|
7.3 | IC50 | 2 | — | |
YQHVRHHVEWIRMK
|
7.3 | IC50 | 3 | — | |
GHVPEVBTYVRTHA
|
7.3 | IC50 | 7 | — | |
GBIOGHVNJXDPTI
|
7.3 | IC50 | 2 | — | |
HTRJNCXDNJEXTE
|
7.3 | IC50 | 2 | — | |
LXSIOBIMXNFAPK
|
7.3 | IC50 | 2 | — | |
ROKKOEGCWJIYBM
|
7.3 | IC50 | 3 | — | |
YWTVUFINLWIWSD
|
7.3 | IC50 | 2 | — | |
RDCOILYSFOFPMK
|
7.3 | IC50 | 3 | — | |
SVXNNKHVIMXUBX
|
7.3 | Ki | 3 | — | |
OPGZDGQAZJNDIL
|
7.3 | IC50 | 3 | — | |
PZADYECUTZNBBF
|
7.3 | IC50 | 2 | — | |
XQBOWELYOBLTAR
|
7.3 | IC50 | 2 | — | |
OJEKLVGMWTUETI
|
7.3 | IC50 | 2 | — | |
SCVRXRIXRGTJCH
|
7.3 | IC50 | 2 | — | |
WEOYJEAONRLZTP
|
7.2 | IC50 | 2 | — | |
DWNYARNMKKSCAV
|
7.2 | IC50 | 2 | — | |
LJDGJZNBWICGDO
|
7.2 | IC50 | 2 | — | |
SWAHNRUQLSQRJA
|
7.2 | IC50 | 3 | — | |
UMYATHACFZUSIJ
|
7.2 | IC50 | 2 | — | |
ZSKIIFIEKWHPCC
|
7.2 | IC50 | 2 | — | |
OPGZDGQAZJNDIL
|
7.2 | IC50 | 3 | — | |
WBCJLZYNWBZUOD
|
7.2 | IC50 | 4 | — | |
MHAGASFEHUMNPA
|
7.2 | IC50 | 2 | — | |
PUTRGMSPWZNXAA
|
7.2 | IC50 | 2 | — | |
YLQGXGBOYJWXBT
|
7.2 | IC50 | 6 | — | |
FYLALFHFEDXUNH
|
7.2 | IC50 | 3 | — | |
CLPMLRHDUWYGIQ
|
7.2 | IC50 | 3 | — | |
IXTYKLRDJPLWOX
|
7.2 | IC50 | 2 | — | |
YDVBKYKVTWRKIY
|
7.2 | Ki | 3 | — | |
ZHBCFUGAJMXZDU
|
7.2 | IC50 | 2 | — | |
BFIKQYQPKFNDJQ
|
7.2 | IC50 | 4 | — | |
BNVVNCVXADUCNT
|
7.2 | IC50 | 2 | — | |
ZYVUFELPRWRHOR
|
7.2 | IC50 | 2 | — |