Target Details
| UniProt AC | P27487 |
|---|---|
| Gene Symbol | DPP4 |
| Protein Name | Dipeptidyl peptidase 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00930 (DPPIV_N) PF00326 (Peptidase_S9) |
Summary
- Multi-target molecules 550
- Clinical molecules 3
- Avg pChEMBL 7.78
KEGG Pathways (2)
Active Molecules (550)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DVJAMEIQRSHVKC
|
7.6 | IC50 | 2 | — | |
FWAIOMYEQWSGSO
|
7.6 | IC50 | 2 | — | |
IMQBTVOWEGWZTQ
|
7.6 | IC50 | 2 | — | |
MQHXRECXBSFFAH
|
7.6 | IC50 | 6 | — | |
PVJXCUHDUBMQIG
|
7.6 | IC50 | 3 | — | |
GMVMVXIACIVOBR
|
7.6 | IC50 | 2 | — | |
VHFQTXGXXHNCSA
|
7.6 | IC50 | 3 | — | |
ZYXUIWSHYKMKKF
|
7.6 | IC50 | 2 | — | |
BTGXNIALOLYGDP
|
7.6 | IC50 | 2 | — | |
GMVMVXIACIVOBR
|
7.6 | IC50 | 2 | — | |
PEBCJHONXDFPDD
|
7.6 | IC50 | 2 | — | |
PNCYZOJJIHDBQW
|
7.6 | IC50 | 2 | — | |
ZYXUIWSHYKMKKF
|
7.6 | IC50 | 2 | — | |
CDYUFFXWJNHDCH
|
7.6 | IC50 | 3 | — | |
DGFODDFZJTVDBE
|
7.6 | IC50 | 3 | — | |
LHBJCBLEWINWEE
|
7.6 | IC50 | 3 | — | |
SGZSKDAIMPUTKY
|
7.6 | IC50 | 2 | — | |
XXNGRRJMDFPNGD
|
7.6 | IC50 | 2 | — | |
FEFCYILNMDAYPD
|
7.5 | IC50 | 3 | — | |
RUMNOCQXRVXQHH
|
7.5 | IC50 | 3 | — | |
DFYJCRFQTFRQQL
|
7.5 | Ki | 3 | — | |
HEZZWSOOCHPSTM
|
7.5 | Ki | 3 | — | |
ITTGFFWXLHEONY
|
7.5 | IC50 | 2 | — | |
OBBPMZQSYHHZLS
|
7.5 | IC50 | 2 | — | |
ZXZUNWVRSSPWJV
|
7.5 | IC50 | 3 | — | |
CEUHNJVXCHXXJT
|
7.5 | IC50 | 2 | — | |
CPKSIOFLZDEMJS
|
7.5 | IC50 | 2 | — | |
CWYRIAXMURYWCO
|
7.5 | IC50 | 2 | — | |
PUKARVRQDSPFPB
|
7.5 | IC50 | 2 | — | |
KTOZHKKTQSOMAC
|
7.5 | IC50 | 2 | — | |
XKINFADDUXLVQO
|
7.5 | IC50 | 4 | — | |
AYERFFUVGKDBLN
|
7.5 | IC50 | 2 | — | |
BXWYQMPOVCJLIS
|
7.5 | IC50 | 4 | — | |
IQFUBDUMFIQJND
|
7.5 | IC50 | 2 | — | |
JKNMLQBDAFABJN
|
7.5 | IC50 | 3 | — | |
PGJBNBOMGATLCI
|
7.5 | IC50 | 2 | — | |
RGFGJCQSMFQBDA
|
7.5 | IC50 | 3 | — | |
SQFZVFRBKRWUGQ
|
7.5 | IC50 | 2 | — | |
VDFNHBBTFMQIJU
|
7.5 | IC50 | 3 | — | |
WAVJGCCRPYAHLF
|
7.5 | IC50 | 4 | — | |
AIHJWXVXFBJARD
|
7.4 | IC50 | 2 | — | |
AIHJWXVXFBJARD
|
7.4 | IC50 | 2 | — | |
DMEMEVKGKFAOHJ
|
7.4 | IC50 | 2 | — | |
XAXKWKHCLDUGSC
|
7.4 | IC50 | 2 | — | |
KZUMVCZJLNJWHF
|
7.4 | IC50 | 2 | — | |
KZUMVCZJLNJWHF
|
7.4 | IC50 | 2 | — | |
ONRMYFPPPIJZIS
|
7.4 | IC50 | 3 | — | |
NTSXERLNWNEXJZ
|
7.4 | IC50 | 2 | — | |
QNPWPDPAAFHYEL
|
7.4 | IC50 | 2 | — | |
QNPWPDPAAFHYEL
|
7.4 | IC50 | 2 | — |