Target Details
| UniProt AC | P27487 |
|---|---|
| Gene Symbol | DPP4 |
| Protein Name | Dipeptidyl peptidase 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00930 (DPPIV_N) PF00326 (Peptidase_S9) |
Summary
- Multi-target molecules 550
- Clinical molecules 3
- Avg pChEMBL 7.78
KEGG Pathways (2)
Active Molecules (550)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XNYPZBCCPFEFKG
|
7.8 | IC50 | 4 | — | |
YQHVRHHVEWIRMK
|
7.8 | IC50 | 3 | — | |
ZPXUSKUJOYAZDE
|
7.8 | IC50 | 2 | — | |
FWTKUAZIABBHDG
|
7.8 | IC50 | 5 | — | |
QQWAAYVLDUCPCB
|
7.8 | IC50 | 3 | — | |
XIYYLZKLNGSLAJ
|
7.8 | IC50 | 2 | — | |
XIYYLZKLNGSLAJ
|
7.8 | IC50 | 2 | — | |
YQHVRHHVEWIRMK
|
7.8 | IC50 | 3 | — | |
VBUWQVASCOSYOA
|
7.8 | IC50 | 2 | — | |
OKRRCGPMTODYSO
|
7.8 | IC50 | 2 | — | |
KPULQFRFEHKYJN
|
7.8 | IC50 | 2 | — | |
OUTGBEKENIEJSN
|
7.8 | IC50 | 2 | — | |
RYWOUVPMSNURME
|
7.8 | Ki | 3 | — | |
TUHONCVWZIUJQF
|
7.8 | IC50 | 3 | — | |
UFKZUCRYERHLMO
|
7.8 | IC50 | 3 | — | |
ZXZUNWVRSSPWJV
|
7.8 | IC50 | 3 | — | |
PZRVLRRTOLHQPA
|
7.8 | IC50 | 2 | — | |
SUVWKEOODLERME
|
7.7 | IC50 | 2 | — | |
YKYFCUZSEAKDFM
|
7.7 | IC50 | 2 | — | |
ZFPIDBLQXYWDHM
|
7.7 | Ki | 2 | — | |
IOGINJTZTHWKHC
|
7.7 | IC50 | 2 | — | |
IOGINJTZTHWKHC
|
7.7 | IC50 | 2 | — | |
LIFQCANQFXGCDS
|
7.7 | IC50 | 2 | — | |
LIFQCANQFXGCDS
|
7.7 | IC50 | 2 | — | |
PHJKYNSEJIZCAD
|
7.7 | IC50 | 2 | — | |
AKUNMFBNBYVKEQ
|
7.7 | IC50 | 4 | — | |
XTKKBNBCZVXQHF
|
7.7 | IC50 | 2 | — | |
IKUISOBQXBKHEE
|
7.7 | Ki | 4 | — | |
YQHVRHHVEWIRMK
|
7.7 | IC50 | 3 | — | |
AYKSOEXCVFOICI
|
7.7 | IC50 | 2 | — | |
IKPSTJUNXQLLLI
|
7.7 | IC50 | 2 | — | |
IQZGQZRIRWWXMX
|
7.7 | IC50 | 2 | — | |
OOXYFRGBSLUXAB
|
7.7 | IC50 | 2 | — | |
SCKICTTYVVYRPZ
|
7.7 | IC50 | 2 | — | |
SYTNSVGDEHOAHB
|
7.7 | IC50 | 2 | — | |
UBZAWPWRJAUSNK
|
7.7 | Ki | 3 | — | |
AOKRQCIWMGZDDW
|
7.7 | Ki | 2 | — | |
DUQWZJWFTUCARE
|
7.7 | IC50 | 6 | — | |
FKCMADOPPWWGNZ
|
7.7 | IC50 | 3 | — | |
IAXFZVFUACWVDO
|
7.7 | IC50 | 3 | — | |
IEFYZYNWWLPCJV
|
7.7 | IC50 | 2 | — | |
OXWKYGRZWVLPOF
|
7.7 | IC50 | 4 | — | |
LMCNNCISVGRBQK
|
7.6 | IC50 | 3 | — | |
LXEJMHRSZPBLRA
|
7.6 | IC50 | 3 | — | |
RMZXAQNHSDWZDH
|
7.6 | IC50 | 2 | — | |
SYOKIDBDQMKNDQ
|
7.6 | IC50 | 3 | — | |
XBMITRBRBFZWMY
|
7.6 | IC50 | 2 | — | |
BJXIVQVJSPSKQE
|
7.6 | Ki | 2 | — | |
QQNHTINEHANVJY
|
7.6 | IC50 | 2 | — | |
WPLYXFXZTORDCT
|
7.6 | IC50 | 3 | — |