Target Details
| UniProt AC | P27487 |
|---|---|
| Gene Symbol | DPP4 |
| Protein Name | Dipeptidyl peptidase 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00930 (DPPIV_N) PF00326 (Peptidase_S9) |
Summary
- Multi-target molecules 550
- Clinical molecules 3
- Avg pChEMBL 7.78
KEGG Pathways (2)
Active Molecules (550)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NHUNIBDLWXLRBY
|
8.1 | IC50 | 3 | — | |
XAOOJPSBTBPGLY
|
8.1 | IC50 | 2 | — | |
ANONTXNDTZLCFJ
|
8.1 | IC50 | 2 | — | |
DGGYQQCWHVPZRV
|
8.1 | IC50 | 3 | — | |
LZRNDAKXSHXRJN
|
8.1 | IC50 | 2 | — | |
CIYSGOBBUFBQIH
|
8.1 | IC50 | 3 | — | |
DGFODDFZJTVDBE
|
8.1 | IC50 | 2 | — | |
GEKJAYDKEVECQC
|
8.1 | IC50 | 2 | — | |
KEHDIZISMAQBKX
|
8.1 | IC50 | 2 | — | |
PDSFQJYJMMJUTN
|
8.1 | IC50 | 3 | — | |
PDSFQJYJMMJUTN
|
8.1 | IC50 | 3 | — | |
LJLRZRUHARLSSJ
|
8.1 | IC50 | 4 | — | |
LKKWOSVPEMTNNP
|
8.1 | Ki | 3 | — | |
QZQMHVURPDKZHO
|
8.1 | Ki | 2 | — | |
ITGGEZBXZCTHDU
|
8.1 | IC50 | 4 | — | |
RTQKTWYQOVSVLC
|
8.1 | Ki | 2 | — | |
YIYAUIWJPDJXEC
|
8.1 | IC50 | 2 | — | |
JVPBPORZRDYLOU
|
8.1 | IC50 | 6 | — | |
ZXFWCMGMSOMZFC
|
8.1 | IC50 | 2 | — | |
PJGGRUQCESCOHY
|
8.0 | IC50 | 4 | — | |
AQFAIYNCQTYWSQ
|
8.0 | IC50 | 3 | — | |
DHJQGELJULZCPM
|
8.0 | IC50 | 2 | — | |
HGEQTKWTBCNJEW
|
8.0 | IC50 | 4 | — | |
MTBATCJDNBSLTB
|
8.0 | IC50 | 4 | — | |
OHOPDRRPSWGLIL
|
8.0 | Ki | 2 | — | |
VVVGZTGKMJOGEW
|
8.0 | IC50 | 2 | — | |
NTSFWZVBIVORHZ
|
8.0 | IC50 | 3 | — | |
JSBRNGDYGFBUPK
|
8.0 | Ki | 3 | — | |
LBYXBJFNOYPLBF
|
8.0 | IC50 | 3 | — | |
MLRHWBQYYDVLMQ
|
8.0 | Ki | 3 | — | |
PHCFSFBQEROREL
|
8.0 | IC50 | 6 | — | |
ZWYVWOHOVTWLNH
|
8.0 | IC50 | 3 | — | |
BZOKGOVFXOVEJF
|
7.9 | IC50 | 3 | — | |
CTVCNKIVQXSUSH
|
7.9 | Ki | 2 | — | |
DYWIFQZBBPGCNX
|
7.9 | IC50 | 2 | — | |
HTCIQWGNZAEQKI
|
7.9 | Ki | 3 | — | |
LGHBEIDFUUJBSV
|
7.9 | IC50 | 2 | — | |
PPEROMZIWASUGT
|
7.9 | Ki | 3 | — | |
XCCSSVMRGIQMGF
|
7.9 | IC50 | 2 | — | |
YPGNHGMZLLVIHB
|
7.9 | IC50 | 3 | — | |
ZNNCLYSYFNMXCX
|
7.9 | IC50 | 7 | — | |
CCCCRDFOGIQSFC
|
7.9 | IC50 | 2 | — | |
WFOKSQKLWVYFPZ
|
7.9 | IC50 | 3 | — | |
JFLWTONGCRBODS
|
7.8 | IC50 | 2 | — | |
WDNVNCPECUHEGM
|
7.8 | IC50 | 2 | — | |
CQMFJBQSRKSKOJ
|
7.8 | Ki | 3 | — | |
IPGJEBMBCSCKBX
|
7.8 | IC50 | 2 | — | |
ISAYLDPRTPLQPU
|
7.8 | IC50 | 4 | — | |
JUMMJPACZXTMNS
|
7.8 | IC50 | 3 | — | |
ONEZBKYGJZWXCN
|
7.8 | IC50 | 2 | — |