Target Details
| UniProt AC | P27487 |
|---|---|
| Gene Symbol | DPP4 |
| Protein Name | Dipeptidyl peptidase 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00930 (DPPIV_N) PF00326 (Peptidase_S9) |
Summary
- Multi-target molecules 550
- Clinical molecules 3
- Avg pChEMBL 7.78
KEGG Pathways (2)
Active Molecules (550)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KRTKHGSZOGTURQ
|
9.0 | Ki | 3 | — | |
LTXREWYXXSTFRX
|
9.0 | IC50 | 3 | — | |
UVLAIQGSAPXWHH
|
9.0 | Ki | 3 | — | |
FQLSDZRDGGRNBU
|
9.0 | Ki | 3 | — | |
RREWXFWIJFLGBI
|
9.0 | Ki | 3 | — | |
RWNXMLKAIWDHLU
|
9.0 | IC50 | 2 | — | |
YPMDOGSZRWVDOZ
|
9.0 | Ki | 6 | — | |
ZUXRZVPVHVFNSX
|
9.0 | IC50 | 2 | — | |
OOTQGBQMGZXPSV
|
8.9 | Ki | 4 | — | |
IQCXFICIUMLNPY
|
8.9 | IC50 | 3 | — | |
APAWICYFJOXVSI
|
8.9 | Ki | 3 | — | |
ZRWMIHVRYPKICQ
|
8.9 | IC50 | 2 | — | |
JGJABGSOYWQCSC
|
8.8 | Ki | 3 | — | |
VEWKBTTWHTZHER
|
8.8 | IC50 | 7 | — | |
XBIIDVIXTFCFMM
|
8.8 | IC50 | 5 | — | |
HRPXFEWNYGNBNG
|
8.8 | IC50 | 2 | — | |
LODNLIGCRDVPHF
|
8.8 | Ki | 3 | — | |
QGJUIPDUBHWZPV
|
8.8 | IC50 | 3 | — | |
YSWYESAJMAXMOW
|
8.8 | IC50 | 2 | — | |
YWWWYGQQSBBBEZ
|
8.8 | Ki | 5 | — | |
DYWIFQZBBPGCNX
|
8.8 | IC50 | 2 | — | |
NRTUDFQDPVFTRM
|
8.8 | IC50 | 2 | — | |
XCCSSVMRGIQMGF
|
8.8 | IC50 | 2 | — | |
ZWKWPVARAOYCNW
|
8.8 | IC50 | 2 | — | |
SXJMLLMEFNYEQL
|
8.8 | IC50 | 2 | — | |
HRRDDUUHRLZHKI
|
8.8 | IC50 | 2 | — | |
PVWNTNVPPWCQAH
|
8.8 | IC50 | 2 | — | |
DMTPQYQQHYOTQM
|
8.7 | IC50 | 6 | — | |
DXRCXIFJMBZDLA
|
8.7 | Ki | 3 | — | |
JGIPUZQWGWHNLZ
|
8.7 | IC50 | 3 | — | |
KTOQVDYNVULFMN
|
8.7 | IC50 | 3 | — | |
WRUWEAUEMYXCRS
|
8.7 | IC50 | 2 | — | |
UYXAPGZGTCWPHK
|
8.7 | IC50 | 2 | — | |
AUZSDJGYAUSLSY
|
8.7 | IC50 | 2 | — | |
BJBOAPYAMPEKGS
|
8.7 | IC50 | 2 | — | |
FKCMADOPPWWGNZ
|
8.7 | IC50 | 6 | — | |
HGJBPTYSVMUIKF
|
8.7 | Ki | 3 | — | |
JVPBPORZRDYLOU
|
8.7 | IC50 | 3 | — | |
KQPQOENOYPKDIN
|
8.7 | IC50 | 2 | — | |
LMGYQTFTIFUZCP
|
8.7 | IC50 | 2 | — | |
MQHXRECXBSFFAH
|
8.7 | IC50 | 6 | — | |
SXNUNNAPZNTPQV
|
8.7 | IC50 | 2 | — | |
XBODCTVRQGLZFY
|
8.7 | IC50 | 2 | — | |
XWGIZMOOTLOFBG
|
8.7 | IC50 | 2 | — | |
ZSANYRQZXIRJRH
|
8.7 | Ki | 3 | — | |
CXZGZTKUARYIDS
|
8.7 | Ki | 3 | — | |
DBOZUIVNRDURJJ
|
8.7 | IC50 | 3 | — | |
MNRQGIJBOGTUFQ
|
8.7 | Ki | 3 | — | |
LXEJMHRSZPBLRA
|
8.6 | IC50 | 3 | — | |
RBLWOLKKTLUERQ
|
8.6 | Ki | 3 | — |