Target Details
| UniProt AC | P27487 |
|---|---|
| Gene Symbol | DPP4 |
| Protein Name | Dipeptidyl peptidase 4 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00930 (DPPIV_N) PF00326 (Peptidase_S9) |
Summary
- Multi-target molecules 550
- Clinical molecules 3
- Avg pChEMBL 7.78
KEGG Pathways (2)
Active Molecules (550)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HJMXMWNMTNQTDK
|
6.9 | IC50 | 2 | — | |
SIUKGJQBSLZIDB
|
6.9 | IC50 | 3 | — | |
NTCVWJJBXJNPGK
|
6.9 | IC50 | 2 | — | |
SOYGWDUWIWWWAW
|
6.9 | IC50 | 2 | — | |
BBDCFVIVCWDRRA
|
6.9 | IC50 | 3 | — | |
WCRLBFHWFPELKW
|
6.9 | Ki | 2 | — | |
ORKCQLYPJLXJQR
|
6.9 | IC50 | 2 | — | |
UNXLWAPASUFEBS
|
6.9 | IC50 | 2 | — | |
UNXLWAPASUFEBS
|
6.9 | IC50 | 2 | — | |
ANMYGYZKOMNFMD
|
6.9 | IC50 | 2 | — | |
MJHMLQMSLLYYIV
|
6.9 | IC50 | 2 | — | |
CJTOOQZVDDNOCD
|
6.8 | IC50 | 2 | — | |
CJTOOQZVDDNOCD
|
6.8 | IC50 | 2 | — | |
JHKIZAUXJSBIHB
|
6.8 | IC50 | 2 | — | |
KZNIFHPLKGYRTM
|
6.8 | IC50 | 21 | Yes | |
NZASMWDMZPCYQT
|
6.8 | IC50 | 2 | — | |
NZASMWDMZPCYQT
|
6.8 | IC50 | 2 | — | |
JGKLCLPAWVWMML
|
6.8 | IC50 | 2 | — | |
CHHIZIRVLVBGFB
|
6.8 | IC50 | 2 | — | |
DEBKZXMRQCNZLE
|
6.8 | IC50 | 2 | — | |
DEBKZXMRQCNZLE
|
6.8 | IC50 | 2 | — | |
NWHZLDQPCBMVMD
|
6.8 | IC50 | 3 | — | |
SNCGIJIHBJNUMZ
|
6.8 | IC50 | 2 | — | |
XQCDOEXVSJZTAR
|
6.8 | IC50 | 3 | — | |
ZLBZIRLEBXTFAN
|
6.8 | IC50 | 2 | — | |
UUONITSRYVQOGQ
|
6.8 | IC50 | 3 | — | |
UUGZWSRZTMDOEL
|
6.8 | IC50 | 3 | — | |
YHODYDUROZNEBI
|
6.8 | IC50 | 2 | — | |
VHBFFQKBGNRLFZ
|
6.8 | IC50 | 21 | — | |
KDGSVHGIVBVYFE
|
6.7 | IC50 | 2 | — | |
DMZNDCVSESDXQQ
|
6.7 | IC50 | 2 | — | |
KFFWURJBCLXNDL
|
6.7 | IC50 | 2 | — | |
SXTVBRRFCBSWSJ
|
6.7 | IC50 | 2 | — | |
JTKCHMXVNWZDGD
|
6.7 | IC50 | 3 | — | |
UJXXZBKYMMMTOG
|
6.7 | IC50 | 3 | — | |
IWXJNMIPPGJIDW
|
6.7 | IC50 | 2 | — | |
SQWDCNZIYSKJKL
|
6.7 | IC50 | 2 | — | |
BCWHINKEOIUUJT
|
6.7 | IC50 | 3 | — | |
OJNCDAFVKCNDBJ
|
6.7 | IC50 | 3 | — | |
QBERUZDRNWBNOV
|
6.7 | IC50 | 2 | — | |
UNPAMBCPZOAJLB
|
6.7 | IC50 | 2 | — | |
KTNUSPOEGQOANN
|
6.6 | IC50 | 2 | — | |
WLQMEUCBATXXEH
|
6.6 | IC50 | 2 | — | |
FTVWIRXFELQLPI
|
6.6 | IC50 | 6 | — | |
GGFAOTAJDWCMLQ
|
6.6 | IC50 | 2 | — | |
LKYFKLGYIAVFES
|
6.6 | IC50 | 2 | — | |
YUEGKNMSWAXVJP
|
6.6 | IC50 | 2 | — | |
BLQSJTWUUQHVBT
|
6.6 | IC50 | 3 | — | |
OABPNHDJHMUHTK
|
6.6 | IC50 | 2 | — | |
AOYYAWFDWQGJIA
|
6.6 | IC50 | 2 | — |