Target Details
UniProt ACP27487
Gene SymbolDPP4
Protein NameDipeptidyl peptidase 4
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF00930 (DPPIV_N) PF00326 (Peptidase_S9)
Summary
  • Multi-target molecules 550
  • Clinical molecules 3
  • Avg pChEMBL 7.78
Top Co-occurrence Targets
Active Molecules (550)
InChIKey pChEMBL Type Targets Clinical
DNVZYSMOLXCOLY 10.1 Ki 2
DTJBLPKYVYTFNJ 9.8 IC50 2
FZCRAZHUTJJBEB 9.7 IC50 2
BYPUTAKAOUIYHF 9.7 Ki 3
OJFSBKDDVWJMOU 9.6 IC50 2
HFUIIUHINNYZIC 9.6 IC50 3
OZVWHEGOMPUFMZ 9.6 Ki 2
CIBRWLRGRGMMMC 9.5 Ki 3
FKCMADOPPWWGNZ 9.5 IC50 3
FKCMADOPPWWGNZ 9.5 IC50 5
GFMFEAABVSLIHJ 9.5 Ki 3
IUBVFVIHMGDKMU 9.5 IC50 3
MPJMFYXQDLKORA 9.5 IC50 3
NPDHHSAKDZBURI 9.5 Ki 2
UWUBKMNCQYTDRI 9.5 IC50 3
SOFQOASLSXGZBR 9.5 Ki 2
MXRXLBDXLGOZNC 9.5 IC50 2
ZEMFLZQUUHJMGT 9.5 IC50 6
JWKZKADFQDTDIU 9.4 IC50 3
DGSUAHCROANBGI 9.4 Ki 3
JXXNQEGNWBPSSV 9.4 Ki 3
SXXTUZFVBVFYTQ 9.4 Ki 3
WDWDEKNARRTAAI 9.4 IC50 2
XIZQTPHCQYNKEB 9.4 Ki 3
HLRKUFDGYOQJCU 9.4 IC50 2
MFMDQBPDMCWAMW 9.4 Ki 2
FNMRYIUQPWAZNO 9.3 IC50 2
QZDNMCJSIHSMDY 9.3 Ki 3
PLSOUKNNDKPEQR 9.3 Ki 2
BODWWFCPUUAGKO 9.2 IC50 2
PBKKSVSTEODBGF 9.2 Ki 4
WGRQANOPCQRCME 9.2 IC50 3
LUKBXSAWLPMMSZ 9.2 IC50 18 Yes
NEGWJHQAWQAHOF 9.2 Ki 5
OQFFZYFZRBISJN 9.2 Ki 3
MKJRNYHUGVCOAT 9.2 IC50 3
QTVNDHFXVZVLIP 9.2 IC50 2
IIGXQPFTWGSNDP 9.2 Ki 3
IXOXZCSVVMIYCV 9.2 Ki 3
WDFZXMUIFGGBQF 9.1 IC50 6
RCUCVXSPMYHBOU 9.1 Ki 3
WDFZXMUIFGGBQF 9.1 IC50 2
QKCRGRBXMIWGEO 9.1 Ki 4
DTSZQBAFUITGDQ 9.1 Ki 4
BVKYXWNXHBSXKO 9.1 Ki 3
FFIPQPHIKAFYCA 9.1 Ki 2
BZTBBVKEKPNNBE 9.0 IC50 4
CXDSYZLZPXATBE 9.0 IC50 3
DUYPYSBUOWVEJT 9.0 Ki 3
JOAPVBJGWDLSMU 9.0 IC50 2
2D structure