Target Details
| UniProt AC | P27448 |
|---|---|
| Gene Symbol | MARK3 |
| Protein Name | MAP/microtubule affinity-regulating kinase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02149 (KA1) PF00069 (Pkinase) PF00627 (UBA) |
Summary
- Multi-target molecules 170
- Clinical molecules 20
- Avg pChEMBL 6.74
Associated Diseases (1)
Active Molecules (170)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HRZOUBQYVUXBNS
|
6.0 | Ki | 38 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
JJJSCYSPSKBQAX
|
6.0 | Ki | 34 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
KNARVZUUCLIBGV
|
6.0 | Ki | 33 | — | |
LGHBDVLAHHANMX
|
6.0 | Ki | 53 | — | |
LYNBNVBMAGDJRW
|
6.0 | Ki | 81 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
MIYRKQLKDQNUKZ
|
6.0 | Ki | 23 | — | |
MQRDVGBWWVWMEN
|
6.0 | Ki | 47 | — | |
NHHQJBCNYHBUSI
|
6.0 | Ki | 220 | — | |
NRGYZNJPCGRCLV
|
6.0 | Ki | 52 | — | |
NZVDDFRUBIEKLV
|
6.0 | Ki | 20 | — | |
OAVGBZOFDPFGPJ
|
6.0 | Ki | 42 | Yes | |
RITAVMQDGBJQJZ
|
6.0 | Ki | 33 | — | |
RQJIDUOCLNMUHR
|
6.0 | Ki | 15 | — | |
RTDSHUGNRVXRHN
|
6.0 | Ki | 51 | — | |
SFPWNTQWFFNJIH
|
6.0 | Ki | 48 | — | |
XOOAAYRIVATZNM
|
6.0 | Ki | 55 | — | |
XSRHBCYNCKAFKS
|
6.0 | Ki | 45 | — |