Target Details
| UniProt AC | P27448 |
|---|---|
| Gene Symbol | MARK3 |
| Protein Name | MAP/microtubule affinity-regulating kinase 3 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02149 (KA1) PF00069 (Pkinase) PF00627 (UBA) |
Summary
- Multi-target molecules 170
- Clinical molecules 20
- Avg pChEMBL 6.74
Associated Diseases (1)
Active Molecules (170)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XSDJOIOVIMPMHD
|
6.4 | Ki | 44 | — | |
YGJKHDBRTOPTNK
|
6.4 | Ki | 8 | — | |
YWTBGJGMTBHQTM
|
6.4 | Ki | 65 | — | |
WINHZLLDWRZWRT
|
6.4 | Kd | 201 | Yes | |
ZZSBPGIGIUFJRA
|
6.3 | Kd | 46 | — | |
BIKYDWLMTPRSQL
|
6.3 | Ki | 50 | — | |
FDVSOQRNTAPCHB
|
6.3 | Ki | 40 | — | |
GCBJDOWIQHMCMR
|
6.3 | Ki | 84 | — | |
GSXRCPJTNIGKSZ
|
6.3 | Ki | 43 | — | |
JXMYIDZREHNPDO
|
6.3 | Ki | 19 | — | |
MCCCQFAOMZMZKE
|
6.3 | Ki | 52 | — | |
PRRYQINUAIQTFJ
|
6.3 | Ki | 11 | — | |
RKUKAACYUCUJEE
|
6.3 | Ki | 58 | — | |
XJSFDMGICAWQFS
|
6.3 | Ki | 60 | — | |
ZLVOTRRGLSDLPF
|
6.3 | Ki | 36 | — | |
ASUGUQWIHMTFJL
|
6.2 | Kd | 18 | — | |
KDKUVYLMPJIGKA
|
6.2 | Kd | 91 | Yes | |
AOBLBPWPSKBHSI
|
6.2 | Ki | 55 | — | |
FXQWJULRETZHHW
|
6.2 | Ki | 14 | — | |
GVPOWKVWVGYUKF
|
6.2 | Ki | 3 | — | |
OLUKILHGKRVDCT
|
6.2 | Ki | 44 | Yes | |
QNUKRWAIZMBVCU
|
6.2 | Ki | 46 | — | |
QQUXFYAWXPMDOE
|
6.2 | Ki | 31 | — | |
TVLFEDKEAOXRCZ
|
6.2 | Ki | 22 | — | |
UJLAWZDWDVHWOW
|
6.2 | Ki | 11 | — | |
VUHZDNOPEVGHEO
|
6.2 | Ki | 29 | — | |
VXYDJXMHISGSDA
|
6.2 | Ki | 59 | — | |
WUBHCQHBUVGGRX
|
6.2 | Ki | 11 | — | |
WYOMXSAYYXBPMN
|
6.2 | Ki | 24 | — | |
XHORJSJFHVABEA
|
6.2 | Ki | 49 | — | |
YUOWJICKAJQZLS
|
6.2 | Ki | 35 | — | |
ZVWRFVCNQOECJS
|
6.2 | Ki | 71 | — | |
YBYYWUUUGCNAHQ
|
6.2 | IC50 | 8 | — | |
VAARYSWULJUGST
|
6.1 | Kd | 119 | Yes | |
XZXHXSATPCNXJR
|
6.1 | Kd | 165 | Yes | |
AXIVWWPYPSYJLD
|
6.1 | Ki | 7 | Yes | |
FQEODTMNWMDUMD
|
6.1 | Ki | 25 | — | |
GHPFQRTVUDXWCC
|
6.1 | Ki | 35 | — | |
GVMDVMPNOAVKJR
|
6.1 | Ki | 26 | Yes | |
KCKXYZOBGBJZEG
|
6.1 | Ki | 36 | — | |
MASJMHFQMYAPJR
|
6.1 | Ki | 41 | — | |
NLUPJKQOKWBWFC
|
6.1 | Ki | 69 | — | |
NVRXTLZYXZNATH
|
6.1 | Ki | 47 | Yes | |
ULHGAQSVFPOUDY
|
6.1 | Ki | 43 | — | |
UUWNXFJBBYAMDT
|
6.1 | Ki | 46 | — | |
ZRQXCQXWTLVASO
|
6.1 | Ki | 36 | — | |
IOYFYUOBKSQTFF
|
6.1 | IC50 | 3 | — | |
DJLORVJVWIBDME
|
6.0 | Ki | 24 | — | |
DKSNLQYRZJKYOC
|
6.0 | Ki | 51 | — | |
HEUSUIRCBWROMH
|
6.0 | Ki | 64 | — |